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Safety and Anti-Tumor Study of Oral EPI-506 for Patients With Metastatic Castration-Resistant Prostate Cancer
Clinical Trial ID NCT02606123
PubWeight™ 8.63
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🔗 Visit the ClinicalTrials.gov page for NCT02606123
Top papers
Rank
Title
Journal
Year
PubWeight™
‹?›
1
Targeting Androgen Receptor Activation Function-1 with EPI to Overcome Resistance Mechanisms in Castration-Resistant Prostate Cancer.
Clin Cancer Res
2016
0.87
2
Androgen receptor variant-driven prostate cancer: clinical implications and therapeutic targeting.
Prostate Cancer Prostatic Dis
2016
0.83
3
Resistance to Novel Antiandrogen Therapies in Metastatic Castration-Resistant Prostate Cancer.
Clin Med Insights Oncol
2016
0.83
4
New drugs in prostate cancer.
Prostate Int
2016
0.80
5
EPI-001, A Compound Active against Castration-Resistant Prostate Cancer, Targets Transactivation Unit 5 of the Androgen Receptor.
ACS Chem Biol
2016
0.80
6
Sintokamide A Is a Novel Antagonist of Androgen Receptor That Uniquely Binds Activation Function-1 in Its Amino-terminal Domain.
J Biol Chem
2016
0.77
7
An imaging agent to detect androgen receptor and its active splice variants in prostate cancer.
JCI Insight
2016
0.77
8
Novel Insights into Molecular Indicators of Response and Resistance to Modern Androgen-Axis Therapies in Prostate Cancer.
Curr Urol Rep
2016
0.77
9
Novel mechanism-based therapeutics for androgen axis blockade in castration-resistant prostate cancer.
Curr Opin Endocrinol Diabetes Obes
2016
0.76
10
A sting in the tail: the N-terminal domain of the androgen receptor as a drug target.
Asian J Androl
2016
0.76
11
Advances in hormonal therapies for hormone naïve and castration-resistant prostate cancers with or without previous chemotherapy.
Exp Hematol Oncol
2016
0.75
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