Safety and Anti-Tumor Study of Oral EPI-506 for Patients With Metastatic Castration-Resistant Prostate Cancer

Clinical Trial ID NCT02606123

PubWeight™ 8.63‹?›

🔗 Visit the ClinicalTrials.gov page for NCT02606123

Top papers

Rank Title Journal Year PubWeight™‹?›
1 Targeting Androgen Receptor Activation Function-1 with EPI to Overcome Resistance Mechanisms in Castration-Resistant Prostate Cancer. Clin Cancer Res 2016 0.87
2 Androgen receptor variant-driven prostate cancer: clinical implications and therapeutic targeting. Prostate Cancer Prostatic Dis 2016 0.83
3 Resistance to Novel Antiandrogen Therapies in Metastatic Castration-Resistant Prostate Cancer. Clin Med Insights Oncol 2016 0.83
4 New drugs in prostate cancer. Prostate Int 2016 0.80
5 EPI-001, A Compound Active against Castration-Resistant Prostate Cancer, Targets Transactivation Unit 5 of the Androgen Receptor. ACS Chem Biol 2016 0.80
6 Sintokamide A Is a Novel Antagonist of Androgen Receptor That Uniquely Binds Activation Function-1 in Its Amino-terminal Domain. J Biol Chem 2016 0.77
7 An imaging agent to detect androgen receptor and its active splice variants in prostate cancer. JCI Insight 2016 0.77
8 Novel Insights into Molecular Indicators of Response and Resistance to Modern Androgen-Axis Therapies in Prostate Cancer. Curr Urol Rep 2016 0.77
9 Novel mechanism-based therapeutics for androgen axis blockade in castration-resistant prostate cancer. Curr Opin Endocrinol Diabetes Obes 2016 0.76
10 A sting in the tail: the N-terminal domain of the androgen receptor as a drug target. Asian J Androl 2016 0.76
11 Advances in hormonal therapies for hormone naïve and castration-resistant prostate cancers with or without previous chemotherapy. Exp Hematol Oncol 2016 0.75
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