Published in Angew Chem Int Ed Engl on February 17, 2003
The enantioselective Morita-Baylis-Hillman reaction and its aza counterpart. Angew Chem Int Ed Engl (2007) 1.31
Chiral Brønsted acid-catalyzed enantioselective three-component Povarov reaction. J Am Chem Soc (2009) 1.21
Total synthesis of (±)-aspidophylline A. Angew Chem Int Ed Engl (2014) 1.01
Synthesis of 3-(diarylmethylenyl)oxindole by a palladium-catalyzed domino carbopalladation/C-H activation/C-C bond-forming process. Org Lett (2006) 0.99
Brønsted acid catalyzed enantioselective three-component reaction involving the alpha addition of isocyanides to imines. Angew Chem Int Ed Engl (2009) 0.95
Palladium-catalyzed decarboxylative vinylation of potassium nitrophenyl acetate: application to the total synthesis of (±)-goniomitine. Angew Chem Int Ed Engl (2013) 0.93
Palladium-catalyzed annulation of acyloximes with arynes (or alkynes): synthesis of phenanthridines and isoquinolines. Angew Chem Int Ed Engl (2009) 0.93
Synthesis of protected chiral vicinal diaminoalcohols by diastereoselective intramolecular benzylic substitution from bistrichloroacetimidates. Org Lett (2007) 0.92
Chiral calcium organophosphate-catalyzed enantioselective electrophilic amination of enamides. Org Lett (2010) 0.92
A convergent approach to cyclopeptide alkaloids: total synthesis of sanjoinine G1. J Am Chem Soc (2002) 0.92
Synthesis of DEFG ring of complestatin and chloropeptin I: highly atropdiastereoselective macrocyclization by intramolecular Suzuki-Miyaura reaction. Org Lett (2007) 0.92
Wilkinson's catalyst catalyzed selective hydrogenation of olefin in the presence of an aromatic nitro function: a remarkable solvent effect. J Org Chem (2002) 0.92
Hafnium trifluoromethanesulfonate (hafnium triflate) as a highly efficient catalyst for chemoselective thioacetalization and transthioacetalization of carbonyl compounds. J Org Chem (2008) 0.91
Rapid access to oxindoles by the combined use of an Ugi four-component reaction and a microwave-assisted intramolecular Buchwald-Hartwig amidation reaction. Org Lett (2006) 0.91
Total synthesis of ecteinascidin 743. J Am Chem Soc (2006) 0.90
Catalytic enantioselective Passerini three-component reaction. Angew Chem Int Ed Engl (2008) 0.90
One-pot synthesis of macrocycles by a tandem three-component reaction and intramolecular [3+2] cycloaddition. Org Lett (2006) 0.90
Palladium(II)-catalyzed intramolecular diamination of alkynes under aerobic oxidative conditions: catalytic turnover of an iodide ion. Angew Chem Int Ed Engl (2012) 0.89
Palladium-catalyzed intramolecular C-arylation of benzylic carbon: synthesis of 3-benzoxazolylisoindolinones by a sequence of Ugi-4CR/postfunctionalization. J Org Chem (2008) 0.89
A Unified Strategy toward the Synthesis of Acerogenin-Type Macrocycles: Total Syntheses of Acerogenins A, B, C, and L and Aceroside IV. J Org Chem (1999) 0.89
Synthetic studies toward ecteinascidin 743. J Org Chem (2005) 0.88
Total synthesis of (+)-crocacin C using hidden symmetry. J Org Chem (2010) 0.87
Palladium-catalyzed, modular synthesis of highly functionalized indoles and tryptophans by direct annulation of substituted o-haloanilines and aldehydes. J Org Chem (2006) 0.87
Synthesis of substituted pyridines from cascade [1 + 5] cycloaddition of isonitriles to N-formylmethyl-substituted enamides, aerobic oxidative aromatization, and acyl transfer reaction. J Am Chem Soc (2013) 0.86
Total synthesis of complestatin (chloropeptin II). Angew Chem Int Ed Engl (2010) 0.86
Ammonium chloride-promoted four-component synthesis of pyrrolo[3,4-b]pyridin-5-one. J Am Chem Soc (2002) 0.85
Total synthesis of the marine natural product (-)-cribrostatin 4 (renieramycin H). Angew Chem Int Ed Engl (2007) 0.85
One-pot three-component synthesis of alpha-iminonitriles by IBX/TBAB-mediated oxidative Strecker reaction. Org Lett (2008) 0.85
Catalytic asymmetric Passerini-type reaction: chiral aluminum-organophosphate-catalyzed enantioselective alpha-addition of isocyanides to aldehydes. J Org Chem (2009) 0.85
Palladium- and copper-catalyzed synthesis of medium- and large-sized ring-fused dihydroazaphenanthrenes and 1,4-benzodiazepine-2,5-diones. control of reaction pathway by metal-switching. J Am Chem Soc (2004) 0.85
Synthesis of diastereomers of complestatin and chloropeptin I: substrate-dependent atropstereoselectivity of the intramolecular Suzuki-Miyaura reaction. Angew Chem Int Ed Engl (2008) 0.84
Library generation via postcondensation modifications of isocyanide-based multicomponent reactions. Methods Enzymol (2003) 0.84
Asymmetric synthesis of 5-(1-hydroxyalkyl)tetrazoles by catalytic enantioselective Passerini-type reactions. Angew Chem Int Ed Engl (2008) 0.84
Chiral Brønsted acid-catalyzed enantioselective multicomponent Mannich reaction: synthesis of anti-1,3-diamines using enecarbamates as nucleophiles. Org Lett (2009) 0.84
From natural product to marketed drug: the tiacumicin odyssey. Nat Prod Rep (2013) 0.84
Chiral phosphoric acid-catalyzed enantioselective three-component Povarov reaction using enecarbamates as dienophiles: highly diastereo- and enantioselective synthesis of substituted 4-aminotetrahydroquinolines. J Am Chem Soc (2011) 0.83
Microwave-assisted intramolecular Suzuki-Miyaura reaction to macrocycle, a concise asymmetric total synthesis of biphenomycin B. Org Lett (2005) 0.83
Palladium-catalyzed domino intramolecular N-arylation/intermolecular C-C bond formation for the synthesis of functionalized benzodiazepinediones. Org Lett (2008) 0.83
Modulating the reactivity of alpha-isocyanoacetates: multicomponent synthesis of 5-methoxyoxazoles and furopyrrolones. Angew Chem Int Ed Engl (2007) 0.83
Exploiting the divergent reactivity of α-isocyanoacetate: multicomponent synthesis of 5-alkoxyoxazoles and related heterocycles. Chemistry (2010) 0.83
Copper-mediated N-cyclopropylation of azoles, amides, and sulfonamides by cyclopropylboronic acid. J Org Chem (2008) 0.83
Palladium-catalyzed through-space C(sp(3))-H and C(sp(2))-H bond activation by 1,4-palladium migration: efficient synthesis of [3,4]-fused oxindoles. Angew Chem Int Ed Engl (2013) 0.83
Intramolecular Suzuki-Miyaura reaction for the total synthesis of signal peptidase inhibitors, arylomycins A(2) and B(2). Chemistry (2010) 0.83
Palladium-catalyzed domino process to spirooxindoles: ligand effect on aminopalladation versus carbopalladation. Chemistry (2010) 0.82
Palladium-catalyzed carbo-heterofunctionalization of alkenes for the synthesis of oxindoles and spirooxindoles. Org Lett (2010) 0.82
Unified strategy to monoterpene indole alkaloids: total syntheses of (±)-goniomitine, (±)-1,2-dehydroaspidospermidine, (±)-aspidospermidine, (±)-vincadifformine, and (±)-kopsihainanine A. J Am Chem Soc (2014) 0.81
Cinchona alkaloid amide catalyzed enantioselective formal [2+2] cycloadditions of allenoates and imines: synthesis of 2,4-disubstituted azetidines. Angew Chem Int Ed Engl (2011) 0.81
Copper-promoted N-cyclopropylation of anilines and amines by cyclopropylboronic acid. Chem Commun (Camb) (2010) 0.81
Organocatalytic enantioselective one-pot four-component ugi-type multicomponent reaction for the synthesis of epoxy-tetrahydropyrrolo[3,4-b]pyridin-5-ones. Chemistry (2012) 0.81
Chiral salen-aluminum complex as a catalyst for enantioselective alpha-addition of isocyanides to aldehydes: asymmetric synthesis of 2-(1-hydroxyalkyl)-5-aminooxazoles. Org Lett (2007) 0.81
Ugi-post functionalization, from a single set of ugi-adducts to two distinct heterocycles by microwave-assisted palladium-catalyzed cyclizations: tuning the reaction pathways by ligand switch. J Org Chem (2009) 0.81
Heteroannulation of arynes with N-aryl-α-aminoketones for the synthesis of unsymmetrical N-aryl-2,3-disubstituted indoles: an aryne twist of Bischler-Möhlau indole synthesis. Chem Commun (Camb) (2013) 0.81
Enantioselective total syntheses of leuconolam-leuconoxine-mersicarpine group monoterpene indole alkaloids. J Am Chem Soc (2013) 0.81
Asymmetric total syntheses of (-)-renieramycin M and G and (-)-jorumycin using aziridine as a lynchpin. Org Lett (2009) 0.81
Alcohols in isonitrile-based multicomponent reaction: Passerini reaction of alcohols in the presence of o-iodoxybenzoic acid. Angew Chem Int Ed Engl (2006) 0.80
Plastidic type I signal peptidase 1 is a redox-dependent thylakoidal processing peptidase. Plant J (2014) 0.80
Zinc chloride promoted formal oxidative coupling of aromatic aldehydes and isocyanides to alpha-ketoamides. J Org Chem (2010) 0.80
Synthesis of 3,3-disubstituted oxindoles by one-pot integrated Brønsted base-catalyzed trichloroacetimidation of 3-hydroxyoxindoles and Brønsted acid-catalyzed nucleophilic substitution reaction. Org Biomol Chem (2013) 0.79
Activation of a C(sp3)-H bond by a transient σ-alkylpalladium(II) complex: synthesis of spirooxindoles through a palladium-catalyzed domino carbopalladation/C(sp3)-C(sp3) bond-forming process. Angew Chem Int Ed Engl (2012) 0.79
Highly enantioselective aza Morita-Baylis-Hillman reaction catalyzed by bifunctional beta-isocupreidine derivatives. J Am Chem Soc (2008) 0.79
A New Approach to the Synthesis of Piperazinomycin and Bouvardin: Facile Access to Cycloisodityrosine via an Intramolecular S(N)Ar Reaction. J Org Chem (1996) 0.79
Asymmetric total syntheses of ecteinascidin 597 and ecteinascidin 583. Angew Chem Int Ed Engl (2006) 0.79
Synthetic studies on (-)-lemonomycin: an efficient asymmetric synthesis of lemonomycinone amide. J Org Chem (2009) 0.79
Synthesis of chiral vicinal diamines by highly diastereoselective three-component phenolic Mannich reaction: temperature-dependent stereodivergency. Org Lett (2005) 0.79
Phosphoric acid catalyzed desymmetrization of bicyclic bislactones bearing an all-carbon stereogenic center: total syntheses of (-)-rhazinilam and (-)-leucomidine B. Angew Chem Int Ed Engl (2014) 0.79
Enantioselective synthesis of putative lipiarmycin aglycon related to fidaxomicin/tiacumicin B. Angew Chem Int Ed Engl (2014) 0.79
Trifluoroacetic acid-promoted synthesis of 3-hydroxy, 3-amino and spirooxindoles from α-keto-N-anilides. Org Lett (2011) 0.79
Protecting-group-free total synthesis of (E)- and (Z)-alstoscholarine. Angew Chem Int Ed Engl (2011) 0.79
Passerini three-component reaction of alcohols under catalytic aerobic oxidative conditions. Org Lett (2010) 0.79
Rapid synthesis of cyclodepsipeptides containing a sugar amino acid or a sugar amino alcohol by a sequence of a multicomponent reaction and acid-mediated macrocyclization. J Org Chem (2007) 0.79
Copper catalyzed N-arylation of amidines with aryl boronic acids and one-pot synthesis of benzimidazoles by a Chan-Lam-Evans N-arylation and C-H activation/C-N bond forming process. Org Lett (2012) 0.78
Three-component synthesis of polysubstituted 6-azaindolines and its tricyclic derivatives. Org Lett (2005) 0.78
Copper-catalyzed intermolecular carboetherification of unactivated alkenes by alkyl nitriles and alcohols. Angew Chem Int Ed Engl (2015) 0.78
Synthetic studies on ecteinascidin 743: rapid access to the fully functionalized tetrahydroisoquinoline with a bridged 10-membered sulfur containing macrocycle. Chem Commun (Camb) (2003) 0.78
Palladium-catalyzed three-component synthesis of 3-(diarylmethylene)oxindoles through a domino Sonagashira/carbopalladation/C--H activation/C--C bond-forming sequence. Angew Chem Int Ed Engl (2007) 0.78
Copper-catalyzed cyanomethylation of allylic alcohols with concomitant 1,2-aryl migration: efficient synthesis of functionalized ketones containing an α-quaternary center. Angew Chem Int Ed Engl (2015) 0.78
One-pot synthesis of polyheterocycles by a palladium-catalyzed intramolecular N-arylation/C[bond]H activation/aryl[bond]aryl bond-forming domino process. Angew Chem Int Ed Engl (2003) 0.78
Spirocyclization by palladium-catalyzed domino Heck-direct C-H arylation reactions: synthesis of spirodihydroquinolin-2-ones. Org Lett (2012) 0.77
Importance of the structure of vancomycin binding pocket in designing compounds active against vancomycin-resistant enterococci (VRE). J Antibiot (Tokyo) (2006) 0.77
Synthesis of pyrroles by consecutive multicomponent reaction/[4 + 1] cycloaddition of alpha-iminonitriles with isocyanides. Org Lett (2009) 0.77
A concise total synthesis of (±)-trigonoliimine B. Org Lett (2012) 0.77
IBX-mediated oxidative Ugi-type multicomponent reactions: application to the N and C1 functionalization of tetrahydroisoquinoline. Angew Chem Int Ed Engl (2007) 0.77
Design and synthesis of macrocycles active against vancomycin-resistant enterococci (VRE): the interplay between d-Ala-d-Lac binding and hydrophobic effect. Bioorg Med Chem Lett (2005) 0.76
Exploiting the dual reactivity of o-isocyanobenzamide: three-component synthesis of 4-imino-4H-3,1-benzoxazines. Org Lett (2005) 0.76
Chiral calcium-BINOL phosphate catalyzed diastereo- and enantioselective synthesis of syn-1,2-disubstituted 1,2-diamines: scope and mechanistic studies. Chemistry (2014) 0.76
Chiral phosphoric acid-catalyzed enantioselective three-component Povarov reaction using cyclic enethioureas as dienophiles: stereocontrolled access to enantioenriched hexahydropyrroloquinolines. Chemistry (2012) 0.76
Palladium-catalyzed enantioselective domino heck-cyanation sequence: development and application to the total synthesis of esermethole and physostigmine. Chemistry (2007) 0.76
Design and synthesis of simple macrocycles active against vancomycin-resistant enterococci (VRE). Chemistry (2006) 0.76
Synthesis of polysubstituted 4,5,6,7-tetrahydrofuro[2,3-c]pyridines by a novel multicomponent reaction. Org Lett (2004) 0.76
Copper-mediated/catalyzed oxyalkylation of alkenes with alkylnitriles. Chemistry (2014) 0.76