Docking studies and ligand recognition in folylpolyglutamate synthetase.

PubWeight™: 0.79‹?›

🔗 View Article (PMID 16302815)

Published in J Med Chem on December 01, 2005

Authors

Xiao-Jian Tan1, Heather A Carlson

Author Affiliations

1: Department of Medicinal Chemistry, College of Pharmacy, University of Michigan, 428 Church St., Ann Arbor, Michigan 48109-1065, USA.

Articles by these authors

Binding MOAD (Mother Of All Databases). Proteins (2005) 2.40

Development of polyphosphate parameters for use with the AMBER force field. J Comput Chem (2003) 2.33

Binding MOAD, a high-quality protein-ligand database. Nucleic Acids Res (2007) 1.99

Chemical screens against a reconstituted multiprotein complex: myricetin blocks DnaJ regulation of DnaK through an allosteric mechanism. Chem Biol (2011) 1.89

CSAR benchmark exercise of 2010: selection of the protein-ligand complexes. J Chem Inf Model (2011) 1.61

Exploring experimental sources of multiple protein conformations in structure-based drug design. J Am Chem Soc (2007) 1.52

Gaussian-weighted RMSD superposition of proteins: a structural comparison for flexible proteins and predicted protein structures. Biophys J (2006) 1.45

CSAR benchmark exercise of 2010: combined evaluation across all submitted scoring functions. J Chem Inf Model (2011) 1.42

Small molecule inhibitors of the MDM2-p53 interaction discovered by ensemble-based receptor models. J Am Chem Soc (2007) 1.28

Binding of a small molecule at a protein-protein interface regulates the chaperone activity of hsp70-hsp40. ACS Chem Biol (2010) 1.28

Full protein flexibility is essential for proper hot-spot mapping. J Am Chem Soc (2010) 1.17

CSAR benchmark exercise 2011-2012: evaluation of results from docking and relative ranking of blinded congeneric series. J Chem Inf Model (2013) 1.17

Solvation influences flap collapse in HIV-1 protease. Proteins (2005) 1.16

Incorporating protein flexibility in structure-based drug discovery: using HIV-1 protease as a test case. J Am Chem Soc (2004) 1.15

Mutagenesis reveals the complex relationships between ATPase rate and the chaperone activities of Escherichia coli heat shock protein 70 (Hsp70/DnaK). J Biol Chem (2010) 1.15

Computational studies and peptidomimetic design for the human p53-MDM2 complex. Proteins (2005) 1.10

A poke in the eye: inhibiting HIV-1 protease through its flap-recognition pocket. Biopolymers (2008) 1.10

Protein flexibility and species specificity in structure-based drug discovery: dihydrofolate reductase as a test system. J Am Chem Soc (2007) 1.09

CSAR data set release 2012: ligands, affinities, complexes, and docking decoys. J Chem Inf Model (2013) 1.02

Exploring protein-ligand recognition with Binding MOAD. J Mol Graph Model (2005) 1.00

Incorporating dynamics in E. coli dihydrofolate reductase enhances structure-based drug discovery. J Chem Inf Model (2007) 0.98

Refining the multiple protein structure pharmacophore method: consistency across three independent HIV-1 protease models. J Med Chem (2006) 0.97

Protein flexibility in docking and surface mapping. Q Rev Biophys (2012) 0.96

Novel deletion of lysine 7 expands the clinical, histopathological and genetic spectrum of TPM2-related myopathies. Brain (2013) 0.93

Exploring the composition of protein-ligand binding sites on a large scale. PLoS Comput Biol (2013) 0.90

Improving protocols for protein mapping through proper comparison to crystallography data. J Chem Inf Model (2013) 0.86

Clarifying allosteric control of flap conformations in the 1TW7 crystal structure of HIV-1 protease. Proteins (2009) 0.85

Conformational behavior of beta-proline oligomers. J Am Chem Soc (2003) 0.83

An allosteric modulator of HIV-1 protease shows equipotent inhibition of wild-type and drug-resistant proteases. J Med Chem (2014) 0.82

Computational methods for predicting sites of functionally important dynamics. J Phys Chem B (2009) 0.82

Chemical probes that selectively recognize the earliest Aβ oligomers in complex mixtures. J Am Chem Soc (2010) 0.82

The role of tyrosine 71 in modulating the flap conformations of BACE1. Proteins (2011) 0.81

Computational methods for identifying a layered allosteric regulatory mechanism for ALS-causing mutations of Cu-Zn superoxide dismutase 1. Proteins (2011) 0.81

Secondary structural preferences of 2,2-disubstituted pyrrolidine-4-carboxylic acid oligomers: beta-peptide foldamers that cannot form internal hydrogen bonds. J Am Chem Soc (2003) 0.81

Parameter choice matters: validating probe parameters for use in mixed-solvent simulations. J Chem Inf Model (2014) 0.80

The role of aspartic acid 143 in E. coli tRNA-guanine transglycosylase: insights from mutagenesis studies and computational modeling. Biophys J (2005) 0.80

Biophysical limits of protein-ligand binding. J Chem Inf Model (2012) 0.79

Binding to the open conformation of HIV-1 protease. Proteins (2011) 0.79

A call to arms: what you can do for computational drug discovery. J Chem Inf Model (2011) 0.78

Automated clustering of probe molecules from solvent mapping of protein surfaces: new algorithms applied to hot-spot mapping and structure-based drug design. J Comput Aided Mol Des (2008) 0.78

Quantum mechanical models of the resting state of the vanadium-dependent haloperoxidase. Inorg Chem (2004) 0.77

Identification of key hinge residues important for nucleotide-dependent allostery in E. coli Hsp70/DnaK. PLoS Comput Biol (2013) 0.76

Overcoming sequence misalignments with weighted structural superposition. Proteins (2012) 0.75

The 12-minute journey. Narrat Inq Bioeth (2014) 0.75