Functional efficacy of adenosine A₂A receptor agonists is positively correlated to their receptor residence time.

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Published in Br J Pharmacol on July 01, 2012

Authors

Dong Guo1, Thea Mulder-Krieger, Adriaan P IJzerman, Laura H Heitman

Author Affiliations

1: Division of Medicinal Chemistry, Leiden/Amsterdam Centre for Drug Research, Leiden University, Leiden, the Netherlands.

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