J T Sisko

Author PubWeight™ 6.20‹?›

Top papers

Rank Title Journal Year PubWeight™‹?›
1 Statins suppress THP-1 cell migration and secretion of matrix metalloproteinase 9 by inhibiting geranylgeranylation. J Leukoc Biol 2001 1.23
2 Design and synthesis of a series of potent and orally bioavailable noncovalent thrombin inhibitors that utilize nonbasic groups in the P1 position. J Med Chem 1998 1.08
3 Characterization of the two-step pathway for inhibition of thrombin by alpha-ketoamide transition state analogs. J Biol Chem 1998 0.91
4 Amide and alpha-keto carbonyl inhibitors of thrombin based on arginine and lysine: synthesis, stability and biological characterization. Bioorg Med Chem 1995 0.82
5 Design of novel, potent, noncovalent inhibitors of thrombin with nonbasic P-1 substructures: rapid structure-activity studies by solid-phase synthesis. J Med Chem 1998 0.81
6 2-Arylindole-3-acetamides: FPP-competitive inhibitors of farnesyl protein transferase. Bioorg Med Chem Lett 2001 0.77
7 Inhibition of thrombin by peptides containing Lysyl-alpha-keto carbonyl derivatives. Thromb Haemost 1995 0.75
8 Synthesis and solution conformation of c(D-Trp-D-Cys(SO3-Na+)-Pro-D-Val-Leu), a potent endothelin-A receptor antagonist. Int J Pept Protein Res 1993 0.75
9 NMR and molecular modeling characterization of RGD containing peptides. Int J Pept Protein Res 1992 0.75
10 Synthesis of a series of potent and orally bioavailable thrombin inhibitors that utilize 3,3-disubstituted propionic acid derivatives in the P3 position. J Med Chem 1997 0.75