Published in Org Lett on September 18, 2003
Formal syntheses of (+/-)-pinnaic acid and (+/-)-halichlorine. Org Lett (2005) 1.15
Concise total synthesis of (+/-)-pseudotabersonine via double ring-closing metathesis strategy. Org Lett (2010) 0.96
Enantioselective synthesis of (+)-isolysergol via ring-closing metathesis. Org Lett (2010) 0.95
Toward the total synthesis of FR901483: concise synthesis of the azatricyclic skeleton. J Org Chem (2007) 0.95
Facile Syntheses of Substituted, Conformationally-Constrained Benzoxazocines and Benzazocines via Sequential Multicomponent Assembly and Cyclization. Tetrahedron Lett (2011) 0.88
Recent Applications of Imines as Key Intermediates in the Synthesis of Alkaloids and Novel Nitrogen Heterocycles. Pure Appl Chem (2009) 0.85
Concise, enantioselective total synthesis of (-)-alstonerine. Org Lett (2007) 0.84
Synthesis of Functionalized Isoindolinones: Addition of In Situ Generated Organoalanes to Acyliminium Ions. J Organomet Chem (2007) 0.83
Retracted Novel approach to the lundurine alkaloids: synthesis of the tetracyclic core. Org Lett (2011) 0.80
Carbamoyl radical-mediated synthesis and semipinacol rearrangement of β-lactam diols. Chemistry (2014) 0.78
The Pauson-Khand Reaction as a New Entry to the Synthesis of Bridged Bicyclic Heterocycles: Application to the Enantioselective Total Synthesis of (-)-Alstonerine. Tetrahedron (2008) 0.77
Applications of Ring Closing Metathesis. Total Synthesis of (±)-Pseudotabersonine. Tetrahedron (2015) 0.75
Synthesis of oxygen- and nitrogen-containing heterocycles by ring-closing metathesis. Chem Rev (2004) 2.41
Applications of multicomponent reactions for the synthesis of diverse heterocyclic scaffolds. Org Lett (2007) 1.68
Applications of multicomponent reactions to the synthesis of diverse heterocyclic scaffolds. Chemistry (2009) 1.60
Enantioselective total syntheses of manzamine a and related alkaloids. J Am Chem Soc (2002) 1.52
Thermodynamic and structural effects of conformational constraints in protein-ligand interactions. Entropic paradoxy associated with ligand preorganization. J Am Chem Soc (2009) 1.37
Synthesis and diversification of 1,2,3-triazole-fused 1,4-benzodiazepine scaffolds. Org Lett (2011) 1.34
Synthesis of Diverse Heterocyclic Scaffolds via Tandem Additions to Imine Derivatives and Ring-Forming Reactions. Tetrahedron (2009) 1.27
Synthesis of bridged azabicyclic structures via ring-closing olefin metathesis. J Org Chem (2003) 1.25
Regioselective synthesis of unsymmetrical C-aryl glycosides using silicon tethers as disposable linkers. J Am Chem Soc (2003) 1.22
General strategy for the syntheses of corynanthe, tacaman, and oxindole alkaloids. J Org Chem (2006) 1.16
Ligand preorganization may be accompanied by entropic penalties in protein-ligand interactions. Angew Chem Int Ed Engl (2006) 1.15
Facile and unified approach to skeletally diverse, privileged scaffolds. Org Lett (2011) 1.15
Formal syntheses of (+/-)-pinnaic acid and (+/-)-halichlorine. Org Lett (2005) 1.15
C-Aryl glycosides via tandem intramolecular benzyne-furan cycloadditions. Total synthesis of vineomycinone B2 methyl ester. J Am Chem Soc (2006) 1.14
Calorimetric and structural studies of 1,2,3-trisubstituted cyclopropanes as conformationally constrained peptide inhibitors of Src SH2 domain binding. J Am Chem Soc (2002) 1.13
Concise, stereoselective approach to the spirooxindole ring system of citrinadin A. Org Lett (2007) 1.13
Diversity-Oriented Synthesis Yields a Novel Lead for the Treatment of Malaria. ACS Med Chem Lett (2011) 1.12
Multicomponent assembly strategies for the synthesis of diverse tetrahydroisoquinoline scaffolds. Org Lett (2011) 1.12
Altering protein specificity: techniques and applications. Bioorg Med Chem (2005) 1.12
Cascade iminium ion reactions for the facile synthesis of quinolizidines. Concise syntheses of (+/-)-epilupinine and (-)-epimyrtine. Org Lett (2005) 1.11
Approaches to N-methylwelwitindolinone C isothiocyanate: facile synthesis of the tetracyclic core. Org Lett (2010) 1.09
Multicomponent assembly and diversification of novel heterocyclic scaffolds derived from 2-arylpiperidines. Org Lett (2011) 1.09
Facile synthesis of 2-substituted 1,2-dihydro-1-naphthols and 2-substituted 1-naphthols. Org Lett (2004) 1.06
Total synthesis of (+)-4,5-deoxyneodolabelline. J Am Chem Soc (2003) 1.05
Enantioselective total synthesis of (-)-citrinadin A and revision of its stereochemical structure. J Am Chem Soc (2013) 1.03
Constraining binding hot spots: NMR and molecular dynamics simulations provide a structural explanation for enthalpy-entropy compensation in SH2-ligand binding. J Am Chem Soc (2010) 1.02
Total synthesis of cribrostatin 6. Angew Chem Int Ed Engl (2009) 1.02
Enantioselective total syntheses of citrinadins A and B. Stereochemical revision of their assigned structures. J Am Chem Soc (2014) 1.01
Tandem Electrocyclic Ring Opening/Radical Cyclization: Application to the Total Synthesis of Cribrostatin 6. Tetrahedron (2011) 1.00
An abiotic strategy for the enantioselective synthesis of erythromycin B. Angew Chem Int Ed Engl (2003) 1.00
Synthesis and properties of cyclopropane-derived peptidomimetics. Acc Chem Res (2006) 0.99
Total synthesis of isokidamycin. J Am Chem Soc (2010) 0.98
Concise total synthesis of (+/-)-pseudotabersonine via double ring-closing metathesis strategy. Org Lett (2010) 0.96
Probing the effect of conformational constraint on phosphorylated ligand binding to an SH2 domain using polarizable force field simulations. J Phys Chem B (2012) 0.96
Structural and energetic aspects of Grb2-SH2 domain-swapping. Arch Biochem Biophys (2007) 0.96
Enantioselective synthesis of (+)-isolysergol via ring-closing metathesis. Org Lett (2010) 0.95
Toward the total synthesis of FR901483: concise synthesis of the azatricyclic skeleton. J Org Chem (2007) 0.95
Concise total synthesis of (+/-)-lycopladine A. Org Lett (2010) 0.95
Tandem Intramolecular Benzyne-Furan Cycloadditions. Total Synthesis of Vineomycinone B(2) Methyl Ester. Tetrahedron (2007) 0.95
Thermodynamic and Structural Effects of Macrocyclization as a Constraining Method in Protein-Ligand Interactions. ACS Med Chem Lett (2010) 0.95
Application of a sequential multicomponent assembly process/huisgen cycloaddition strategy to the preparation of libraries of 1,2,3-triazole-fused 1,4-benzodiazepines. ACS Comb Sci (2012) 0.94
Novel Entry to the Tricyclic Core of Stemofoline and Didehydrostemofoline. Tetrahedron Lett (2011) 0.94
Biomimetic entry to the sarpagan family of indole alkaloids: total synthesis of +-geissoschizine and +-N-methylvellosimine. J Am Chem Soc (2003) 0.94
Bifunctional catalyst promotes highly enantioselective bromolactonizations to generate stereogenic C-Br bonds. J Am Chem Soc (2012) 0.93
Carbonylative cross-coupling of ortho-disubstituted aryl iodides. convenient synthesis of sterically hindered aryl ketones. Org Lett (2008) 0.92
APPLICATIONS OF MULTICOMPONENT ASSEMBLY PROCESSES TO THE FACILE SYNTHESES OF DIVERSELY FUNCTIONALIZED NITROGEN HETEROCYCLES. Heterocycles (2011) 0.92
General and expedient synthesis of 1,4-dioxygenated xanthones. Org Lett (2011) 0.91
Applications of the Ugi reaction with ketones. Tetrahedron Lett (2008) 0.90
Synthesis of β-Heteroaryl Propionates via Trapping of Carbocations with π-Nucleophiles. Tetrahedron Lett (2009) 0.90
Expedient synthesis of norbenzomorphan library via multicomponent assembly process coupled with ring-closing reactions. ACS Comb Sci (2012) 0.89
Toward a total synthesis of the stemofoline alkaloids: Advancement of a 1,3-dipolar cycloaddition strategy. Tetrahedron Lett (2011) 0.89
Facile Syntheses of Substituted, Conformationally-Constrained Benzoxazocines and Benzazocines via Sequential Multicomponent Assembly and Cyclization. Tetrahedron Lett (2011) 0.88
Application of a domino intramolecular enyne metathesis/cross metathesis reaction to the total synthesis of (+)-8-epi-xanthatin. Org Lett (2005) 0.87
Enantioselective syntheses of tremulenediol A and tremulenolide A. Org Lett (2005) 0.86
Studies Toward the Syntheses of Pluramycin Natural Products. The First Total Synthesis of Isokidamycin. Tetrahedron (2011) 0.86
Formal syntheses of naturally occurring welwitindolinones. Org Lett (2012) 0.86
Libraries of 2,3,4,6,7,11b-hexahydro-1H-pyrido[2,1-a]isoquinolin-2-amine derivatives via a multicomponent assembly process/1,3-dipolar cycloaddition strategy. ACS Comb Sci (2011) 0.86
Protein-ligand interactions: thermodynamic effects associated with increasing nonpolar surface area. J Am Chem Soc (2011) 0.85
Enantioselective formal total syntheses of didehydrostemofoline and isodidehydrostemofoline through a catalytic dipolar cycloaddition cascade. Angew Chem Int Ed Engl (2012) 0.85
Concise, enantioselective total synthesis of (-)-alstonerine. Org Lett (2007) 0.84
Altering substrate specificity of phosphatidylcholine-preferring phospholipase C of Bacillus cereus by random mutagenesis of the headgroup binding site. Biochemistry (2003) 0.84
Facile Access to Sterically Hindered Aryl Ketones via Carbonylative Cross-Coupling: Application to the Total Synthesis of Luteolin. Tetrahedron (2011) 0.84
Synthesis of (±)-actinophyllic acid and analogs: applications of cascade reactions and diverted total synthesis. J Am Chem Soc (2013) 0.84
Studies toward welwitindolinones: formal syntheses of N-methylwelwitindolinone C isothiocyanate and related natural products. Tetrahedron (2013) 0.84
Diversity-oriented synthesis-facilitated medicinal chemistry: toward the development of novel antimalarial agents. J Med Chem (2014) 0.83
Studies toward the enantioselective syntheses of oxylipins: total synthesis and structure revision of solandelactone E. J Org Chem (2007) 0.83
Application of intramolecular enyne metathesis to the synthesis of aza[4.2.1]bicyclics: enantiospecific total synthesis of (+)-anatoxin-a. Org Lett (2004) 0.83
Stereoselective total synthesis of dihydrocorynantheol. Org Lett (2002) 0.83
[Rh(CO)2Cl]2-catalyzed domino reactions involving allylic substitution and subsequent carbocyclization reactions. Org Lett (2005) 0.83
Structural studies examining the substrate specificity profiles of PC-PLC(Bc) protein variants. Arch Biochem Biophys (2007) 0.83
Iminium Ion Cascade Reactions: Stereoselective Synthesis of Quinolizidines and Indolizidines. Tetrahedron (2009) 0.83
Diversity Oriented Synthesis: Concise Entry to Novel Derivatives of Yohimbine and Corynanthe Alkaloids. Tetrahedron Lett (2011) 0.82
Concise Approach to 1,4-Dioxygenated Xanthones via Novel Application of the Moore Rearrangement. Tetrahedron (2012) 0.82
Evolution of a strategy for preparing bioactive small molecules by sequential multicomponent assembly processes, cyclizations, and diversification. Org Biomol Chem (2014) 0.82
Multicomponent assembly processes for the synthesis of diverse yohimbine and corynanthe alkaloid analogues. ACS Comb Sci (2013) 0.81
Features and applications of [Rh(CO)(2)Cl](2)-catalyzed alkylations of unsymmetrical allylic substrates. J Org Chem (2007) 0.81
Enantioselective iodolactonization of disubstituted olefinic acids using a bifunctional catalyst. Org Lett (2012) 0.80
Divergent kinetics differentiate the mechanism of action of two HDAC inhibitors. Biochemistry (2014) 0.80
Retracted Novel approach to the lundurine alkaloids: synthesis of the tetracyclic core. Org Lett (2011) 0.80
Binding of flexible and constrained ligands to the Grb2 SH2 domain: structural effects of ligand preorganization. Acta Crystallogr D Biol Crystallogr (2010) 0.80
Enantioselective synthesis of 2,2,5-tri- and 2,2,5,5-tetrasubstituted tetrahydrofurans via [4 + 2] cycloaddition and ring-opening cross-metathesis. Org Lett (2011) 0.79
Approaches to polycyclic 1,4-dioxygenated xanthones. Application to total synthesis of the aglycone of IB-00208. Org Lett (2014) 0.79
Design, synthesis, and evaluation of matrix metalloprotease inhibitors bearing cyclopropane-derived peptidomimetics as P1' and P2' replacements. J Org Chem (2002) 0.79
Asymmetric Formal Total Synthesis of the Stemofoline Alkaloids: The Evolution, Development and Application of a Catalytic Dipolar Cycloaddition Cascade. Tetrahedron (2013) 0.78
Pd-catalyzed ring opening of oxa- and azabicyclic alkenes with aryl and vinyl halides: efficient entry to 2-substituted 1,2-dihydro-1-naphthols and 2-substituted 1-naphthols. J Org Chem (2006) 0.78
Total synthesis of (-)-dihydroprotolichesterenic acid via diastereoselective conjugate addition to chiral fumarates. Tetrahedron Lett (2013) 0.78
Design, synthesis, and evaluation of water-soluble phospholipid analogues as inhibitors of phospholipase C from Bacillus cereus. J Org Chem (2003) 0.77
The Pauson-Khand Reaction as a New Entry to the Synthesis of Bridged Bicyclic Heterocycles: Application to the Enantioselective Total Synthesis of (-)-Alstonerine. Tetrahedron (2008) 0.77
Novel approach to the zaragozic acids. Enantioselective total synthesis of 6,7-dideoxysqualestatin H5. J Org Chem (2002) 0.77
Direct, stereoselective substitution in [Rh(CO)(2)Cl](2)-catalyzed allylic alkylations of unsymmetrical substrates. Org Lett (2004) 0.76
Enantioselective conjugate addition employing 2-heteroaryl titanates and zinc reagents. Org Lett (2009) 0.76
Enantioselective synthesis and structure revision of solandelactone E. J Am Chem Soc (2007) 0.75
Approach toward the total synthesis of 5-hydroxyaloin A. Org Lett (2010) 0.75
Using X-ray crystallography of the Asp55Asn mutant of the phosphatidylcholine-preferring phospholipase C from Bacillus cereus to support the mechanistic role of Asp55 as the general base. Arch Biochem Biophys (2003) 0.75
Enantioselective iodolactonization of disubstituted olefinic acids using a bifunctional catalyst. Org Lett (2013) 0.75