Rank | Title | Journal | Year | PubWeight™‹?› |
---|---|---|---|---|
1 | Synthesis and SAR of pyridazinone-substituted phenylalanine amide alpha4 integrin antagonists. | Bioorg Med Chem Lett | 2008 | 0.80 |
2 | Rationale, design, and synthesis of novel phenyl imidazoles as opioid receptor agonists for gastrointestinal disorders. | J Med Chem | 2004 | 0.80 |
3 | Synthesis and biological evaluation of novel pyridazinone-based alpha4 integrin receptor antagonists. | J Med Chem | 2006 | 0.79 |
4 | Aza-bicyclic amino acid carboxamides as alpha4beta1/alpha4beta7 integrin receptor antagonists. | Bioorg Med Chem | 2005 | 0.77 |
5 | Aza-bicyclic amino acid sulfonamides as alpha(4)beta(1)/alpha(4)beta(7) integrin antagonists. | Bioorg Med Chem Lett | 2004 | 0.75 |