| Rank | Title | Journal | Year | PubWeight™‹?› |
|---|---|---|---|---|
| 1 | Potentiation of cytotoxic drug activity in human tumour cell lines, by amine-substituted 2-arylbenzimidazole-4-carboxamide PARP-1 inhibitors. | Bioorg Med Chem Lett | 2004 | 1.17 |
| 2 | Tricyclic benzimidazoles as potent poly(ADP-ribose) polymerase-1 inhibitors. | J Med Chem | 2003 | 0.98 |
| 3 | Structure-based design of a parallel synthetic array directed toward the discovery of irreversible inhibitors of human rhinovirus 3C protease. | J Med Chem | 2002 | 0.79 |
| 4 | 3-[3-Fluoro-5-(5-pyridin-2-yl-2H-tetrazol-2-yl)phenyl]-4-methylpyridine: a highly potent and orally bioavailable metabotropic glutamate subtype 5 (mGlu5) receptor antagonist. | Bioorg Med Chem Lett | 2004 | 0.76 |