P-glycoprotein and cytochrome P450 3A4 involvement in risperidone transport using an in vitro Caco-2/TC7 model and an in vivo model.

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Published in Prog Neuropsychopharmacol Biol Psychiatry on February 08, 2007

Authors

Etienne Cousein1, Christine Barthélémy, Stéphanie Poullain, Nicolas Simon, Sophie Lestavel, Virginie Williame, Etienne Joiris, Cécile Danel, Véronique Clavey, Denis Brossard, Hugues Robert, Sylvie Crauste-Manciet, Claude Vaccher, Pascal Odou

Author Affiliations

1: Laboratoire de Biopharmacie, EA 4034, Pharmacie Galénique et Hospitalière et Laboratoire de Chimie Analytique, Faculté des Sciences Pharmaceutiques et Biologiques, Université de Lille 2, 3 rue du Professeur Laguesse, 59006 LILLE Cedex, France.

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