|
1
|
In vitro activities of position 2 substitution-bearing 6-nitro- and 6-amino-benzothiazoles and their corresponding anthranilic acid derivatives against Leishmania infantum and Trichomonas vaginalis.
|
Antimicrob Agents Chemother
|
2002
|
1.41
|
|
2
|
Synthesis and biological evaluation of new heterocyclic quinolinones as anti-parasite and anti-HIV drug candidates.
|
Bioorg Med Chem Lett
|
2009
|
1.21
|
|
3
|
TDAE-assisted synthesis of new imidazo[2,1-b]thiazole derivatives as anti-infectious agents.
|
Eur J Med Chem
|
2009
|
0.95
|
|
4
|
Antimalarial activity of sesquiterpene lactones from Vernonia cinerea.
|
Chem Pharm Bull (Tokyo)
|
2006
|
0.93
|
|
5
|
1,3-Diphenylpyrazoles: synthesis and antiparasitic activities of azomethine derivatives.
|
Eur J Med Chem
|
2002
|
0.92
|
|
6
|
Antimalarial activity of alkaloids isolated from Stephania rotunda.
|
J Ethnopharmacol
|
2007
|
0.89
|
|
7
|
Lowering of 5-nitroimidazole's mutagenicity: towards optimal antiparasitic pharmacophore.
|
Eur J Med Chem
|
2008
|
0.88
|
|
8
|
Interaction forces drive the environmental transmission of pathogenic protozoa.
|
Appl Environ Microbiol
|
2011
|
0.87
|
|
9
|
Synthesis and antiprotozoal activity of 4-arylcoumarins.
|
Eur J Med Chem
|
2009
|
0.87
|
|
10
|
Phytochemical and pharmacological study of roots and leaves of Guiera senegalensis J.F. Gmel (Combretaceae).
|
J Ethnopharmacol
|
2006
|
0.87
|
|
11
|
Screening of selected indigenous plants of Cambodia for antiplasmodial activity.
|
J Ethnopharmacol
|
2006
|
0.86
|
|
12
|
Antimalarial activity of crude extracts from nine African medicinal plants.
|
J Ethnopharmacol
|
2007
|
0.86
|
|
13
|
In vitro activities of 7-substituted 9-chloro and 9-amino-2-methoxyacridines and their bis- and tetra-acridine complexes against Leishmania infantum.
|
Antimicrob Agents Chemother
|
2003
|
0.86
|
|
14
|
Antiplasmodial activity and toxicity of crude extracts from alternatives parts of plants widely used for the treatment of malaria in Burkina Faso: contribution for their preservation.
|
Parasitol Res
|
2009
|
0.83
|
|
15
|
A new, rapid and sensitive bioluminescence assay for drug screening on Leishmania.
|
J Microbiol Methods
|
2013
|
0.80
|
|
16
|
Original quinazoline derivatives displaying antiplasmodial properties.
|
Eur J Med Chem
|
2009
|
0.79
|
|
17
|
Mechanics of the Toxoplasma gondii oocyst wall.
|
Proc Natl Acad Sci U S A
|
2013
|
0.78
|
|
18
|
New amide alkaloid from the aerial part of Piper capense L.f. (Piperaceae).
|
Fitoterapia
|
2010
|
0.78
|
|
19
|
Synthesis and antiplasmodial activity of new 4-aryl-2-trichloromethylquinazolines.
|
Bioorg Med Chem Lett
|
2007
|
0.77
|
|
20
|
4-Thiophenoxy-2-trichloromethyquinazolines display in vitro selective antiplasmodial activity against the human malaria parasite Plasmodium falciparum.
|
Bioorg Med Chem Lett
|
2011
|
0.77
|
|
21
|
A decade of Plasmodium falciparum metabolic pathways of therapeutic interest to develop new selective antimalarial drugs.
|
Mini Rev Med Chem
|
2013
|
0.77
|
|
22
|
In vitro antiplasmodial activity of some medicinal plants of Burkina Faso.
|
Parasitol Res
|
2013
|
0.76
|
|
23
|
Preparation and antiprotozoal evaluation of promising β-carboline alkaloids.
|
Biomed Pharmacother
|
2012
|
0.76
|
|
24
|
HPLC quantification of uncarine D and the anti-plasmodial activity of alkaloids from leaves of Mitragyna inermis (Willd.) O. Kuntze.
|
Phytochem Anal
|
2005
|
0.76
|
|
25
|
Discovery of a new antileishmanial hit in 8-nitroquinoline series.
|
Eur J Med Chem
|
2012
|
0.75
|
|
26
|
Anti-HIV and antiplasmodial activity of original flavonoid derivatives.
|
Bioorg Med Chem
|
2010
|
0.75
|
|
27
|
Synthesis and evaluation of original amidoximes as antileishmanial agents.
|
Bioorg Med Chem
|
2010
|
0.75
|
|
28
|
Targeting the human parasite Leishmania donovani: discovery of a new promising anti-infectious pharmacophore in 3-nitroimidazo[1,2-a]pyridine series.
|
Bioorg Med Chem
|
2013
|
0.75
|
|
29
|
Synthesis and evaluation of monoamidoxime derivatives: toward new antileishmanial compounds.
|
Eur J Med Chem
|
2011
|
0.75
|
|
30
|
A new synthetic route to original sulfonamide derivatives in 2-trichloromethylquinazoline series: a structure-activity relationship study of antiplasmodial activity.
|
Molecules
|
2012
|
0.75
|
|
31
|
Tools and methods for detecting and characterizing giardia, cryptosporidium, and toxoplasma parasites in marine mollusks.
|
J Food Prot
|
2013
|
0.75
|
|
32
|
New antiplasmodial alkaloids from Stephania rotunda.
|
J Ethnopharmacol
|
2012
|
0.75
|
|
33
|
Fagraldehyde, a secoiridoid isolated from Fagraea fragrans.
|
J Nat Prod
|
2008
|
0.75
|
|
34
|
HPLC analysis of Stephania rotunda extracts and correlation with antiplasmodial activity.
|
Phytother Res
|
2012
|
0.75
|
|
35
|
Antiplasmodial activity of three bisbenzylisoquinoline alkaloids from the tuber of Stephania rotunda.
|
Nat Prod Res
|
2010
|
0.75
|
|
36
|
Synthesis and promising in vitro antiproliferative activity of sulfones of a 5-nitrothiazole series.
|
Molecules
|
2012
|
0.75
|
|
37
|
Synthesis and in vitro antiplasmodial evaluation of 4-anilino-2-trichloromethylquinazolines.
|
Bioorg Med Chem
|
2009
|
0.75
|
|
38
|
Antimalarial compounds from the aerial parts of Flacourtia indica (Flacourtiaceae).
|
J Ethnopharmacol
|
2010
|
0.75
|
|
39
|
Tandem synthesis and in vitro antiplasmodial evaluation of new naphtho[2,1-d]thiazole derivatives.
|
Eur J Med Chem
|
2012
|
0.75
|
|
40
|
Targeting the human malaria parasite Plasmodium falciparum: in vitro identification of a new antiplasmodial hit in 4-phenoxy-2-trichloromethylquinazoline series.
|
Eur J Med Chem
|
2011
|
0.75
|