Published in J Org Chem on April 12, 2007
Copper(II)-catalyzed enantioselective intramolecular carboamination of alkenes. J Am Chem Soc (2007) 1.94
Copper catalyzed enantioselective intramolecular aminooxygenation of alkenes. J Am Chem Soc (2008) 1.75
Copper(II) carboxylate promoted intramolecular diamination of terminal alkenes: improved reaction conditions and expanded substrate scope. Org Lett (2007) 1.49
Mild conditions for Pd-catalyzed carboamination of N-protected hex-4-enylamines and 1-, 3-, and 4-substituted pent-4-enylamines. Scope, limitations, and mechanism of pyrrolidine formation. J Org Chem (2008) 1.33
Copper-catalyzed enantioselective intramolecular alkene amination/intermolecular Heck-type coupling cascade. J Am Chem Soc (2012) 1.25
Catalytic enantioselective alkene aminohalogenation/cyclization involving atom transfer. Angew Chem Int Ed Engl (2012) 1.22
The enantioselective intramolecular aminative functionalization of unactivated alkenes, dienes, allenes and alkynes for the synthesis of chiral nitrogen heterocycles. Org Biomol Chem (2009) 1.20
Diastereoselective pyrrolidine synthesis via copper promoted intramolecular aminooxygenation of alkenes: formal synthesis of (+)-monomorine. Org Lett (2009) 1.20
A concise asymmetric synthesis of cis-2,6-disubstituted N-aryl piperazines via Pd-catalyzed carboamination reactions. Org Lett (2007) 1.19
Copper(II) carboxylate-promoted intramolecular carboamination of alkenes for the synthesis of polycyclic lactams. Org Lett (2007) 1.13
Copper-promoted and copper-catalyzed intermolecular alkene diamination. Angew Chem Int Ed Engl (2010) 1.08
Evidence for alkene cis-aminocupration, an aminooxygenation case study: kinetics, EPR spectroscopy, and DFT calculations. Chemistry (2012) 1.03
Copper-catalyzed intramolecular alkene carboetherification: synthesis of fused-ring and bridged-ring tetrahydrofurans. J Am Chem Soc (2012) 1.00
Total synthesis of (S)-(+)-tylophorine via enantioselective intramolecular alkene carboamination. J Org Chem (2008) 0.99
Mechanistic studies of Wacker-type intramolecular aerobic oxidative amination of alkenes catalyzed by Pd(OAc)2/pyridine. J Org Chem (2011) 0.97
Copper(II)-Catalyzed Aminooxygenation and Carboamination of N-Aryl-2-allylanilines. Adv Synth Catal (2009) 0.94
Diastereo- and enantioselective copper-catalyzed intramolecular carboamination of alkenes for the synthesis of hexahydro-1H-benz[f]indoles. Org Lett (2010) 0.94
Low temperature organocopper-mediated two-component cross coupling/cycloisomerization approach toward N-fused heterocycles. Org Lett (2008) 0.91
Mechanistic analysis and optimization of the copper-catalyzed enantioselective intramolecular alkene aminooxygenation. J Org Chem (2012) 0.89
Palladium-catalyzed alkene carboamination reactions for the synthesis of substituted piperazines. Tetrahedron (2009) 0.88
Chiral Indoline Synthesis Via Enantioselective Intramolecular Copper-Catalyzed Alkene Hydroamination. Organometallics (2012) 0.84
Intramolecular aminocyanation of alkenes by N-CN bond cleavage. Angew Chem Int Ed Engl (2014) 0.80
Palladium-Catalyzed Alkene Carboamination Reactions of Electron-Poor Nitrogen Nucleophiles. Adv Synth Catal (2015) 0.80
6-Azabicyclo[3.2.1]octanes Via Copper-Catalyzed Enantioselective Alkene Carboamination. Adv Synth Catal (2014) 0.77
Synthesis of substituted tetrahydroindoloisoquinoline derivatives via intramolecular Pd-catalyzed alkene carboamination reactions. J Org Chem (2014) 0.77
Stereoselective Synthesis of Saturated Heterocycles via Pd-Catalyzed Alkene Carboetherification and Carboamination Reactions. Synlett (2006) 0.76
Copper-catalyzed aminooxygenation of styrenes with N-fluorobenzenesulfonimide and N-hydroxyphthalimide derivatives. Beilstein J Org Chem (2015) 0.75
ORGANOCOPPER-MEDIATED TWO-COMPONENT SN2'-SUBSTITUTION CASCADE TOWARDS N-FUSED HETEROCYCLES. Chem Heterocycl Compd (N Y) (2012) 0.75
Intermolecular addition reactions of N-alkyl-N-chlorosulfonamides to unsaturated compounds. Beilstein J Org Chem (2015) 0.75
Bioconjugation by copper(I)-catalyzed azide-alkyne [3 + 2] cycloaddition. J Am Chem Soc (2003) 5.34
Modern synthetic methods for copper-mediated C(aryl)[bond]O, C(aryl)[bond]N, and C(aryl)[bond]S bond formation. Angew Chem Int Ed Engl (2003) 3.81
Aryl-aryl bond formation one century after the discovery of the Ullmann reaction. Chem Rev (2002) 3.65
Metal-Initiated Amination of Alkenes and Alkynes. Chem Rev (1998) 2.64
Palladium-catalyzed synthesis of N-aryl pyrrolidines from gamma-(N-Arylamino) alkenes: evidence for chemoselective alkene insertion into Pd--N bonds. Angew Chem Int Ed Engl (2004) 2.40
Transition-metal-catalyzed reactions in heterocyclic synthesis. Chem Rev (2004) 2.23
Palladium(II)-catalyzed intramolecular diamination of unfunctionalized alkenes. J Am Chem Soc (2005) 2.04
Synthesis of heterocycles via palladium pi-olefin and pi-alkyne chemistry. Chem Rev (2004) 2.04
Pd(II)-catalyzed enantioselective oxidative tandem cyclization reactions. Synthesis of indolines through C-N and C-C bond formation. J Am Chem Soc (2006) 1.86
Copper(II) acetate promoted intramolecular diamination of unactivated olefins. J Am Chem Soc (2005) 1.82
Palladium-catalyzed ring-forming aminoacetoxylation of alkenes. J Am Chem Soc (2005) 1.82
Organolanthanide-catalyzed hydroamination. Acc Chem Res (2004) 1.77
Palladium-catalyzed synthesis of N-aryl-2-benzylindolines via tandem arylation of 2-allylaniline: control of selectivity through in situ catalyst modification. J Am Chem Soc (2004) 1.67
Brønsted acid-catalyzed intramolecular hydroamination of protected alkenylamines. Synthesis of pyrrolidines and piperidines. Org Lett (2002) 1.66
Copper(II) acetate promoted oxidative cyclization of arylsulfonyl-o-allylanilines. Org Lett (2004) 1.65
Cu(II)-catalyzed functionalizations of aryl C-H bonds using O2 as an oxidant. J Am Chem Soc (2006) 1.62
Microwave-accelerated homogeneous catalysis in organic chemistry. Acc Chem Res (2002) 1.58
Synthesis of the azaphilones using copper-mediated enantioselective oxidative dearomatization. J Am Chem Soc (2005) 1.43
Palladium-catalyzed oxidative wacker cyclizations in nonpolar organic solvents with molecular oxygen: a stepping stone to asymmetric aerobic cyclizations. Angew Chem Int Ed Engl (2003) 1.39
Synthesis of biaryls via catalytic decarboxylative coupling. Science (2006) 1.37
Intramolecular Pd-catalyzed carboetherification and carboamination. Influence of catalyst structure on reaction mechanism and product stereochemistry. J Am Chem Soc (2006) 1.35
Efficient intramolecular oxidative amination of olefins through direct dioxygen-coupled palladium catalysis. Angew Chem Int Ed Engl (2002) 1.32
Direct coupling of indoles with carbonyl compounds: short, enantioselective, gram-scale synthetic entry into the hapalindole and fischerindole alkaloid families. J Am Chem Soc (2004) 1.27
A concise stereoselective synthesis of Preussin, 3-epi-Preussin, and analogues. Org Lett (2006) 1.25
Heterocycle synthesis by copper facilitated addition of heteroatoms to alkenes, alkynes and arenes. Chem Soc Rev (2007) 1.21
Enantioselective oxidative biaryl coupling reactions catalyzed by 1,5-diazadecalin metal complexes: efficient formation of chiral functionalized BINOL derivatives. J Org Chem (2003) 1.20
N-sulfonyloxy carbamates as reoxidants for the tethered aminohydroxylation reaction. J Am Chem Soc (2006) 1.12
Synthesis of N-Aryl-2-allyl Pyrrolidines via Palladium-catalyzed Carboamination Reactions of γ-(N-Arylamino)alkenes with Vinyl Bromides. Adv Synth Catal (2005) 1.10
Domino cu-catalyzed C--N coupling/hydroamidation: a highly efficient synthesis of nitrogen heterocycles. Angew Chem Int Ed Engl (2006) 1.09
Iodine(V) reagents in organic synthesis. Part 3. New routes to heterocyclic compounds via o-iodoxybenzoic acid-mediated cyclizations: generality, scope, and mechanism. J Am Chem Soc (2002) 1.09
Catalytic diboration of aldehydes via insertion into the copper-boron bond. J Am Chem Soc (2006) 1.04
A facile access to 2-methylthio/alkoxy/amino-3-acylimidazo[1, 2-a]pyridines based on cupric chloride promoted oxidative ring closure of alpha-oxoketene N,S-, N,O-, and N,N-acetals. J Org Chem (2000) 1.02
Room temperature hydroamination of N-alkenyl ureas catalyzed by a gold(i) N-heterocyclic carbene complex. Org Lett (2006) 1.00
Double reduction of cyclic aromatic sulfonamides: a novel method for the synthesis of 2- and 3-aryl-substituted cyclic amines. Org Lett (2005) 0.99
Stereoselective synthesis of pyrrolidines: catalytic oxidative cyclizations mediated by osmium. Angew Chem Int Ed Engl (2006) 0.98
Synthesis of imidazoles through the copper-catalyzed cross-cycloaddition between two different isocyanides. J Am Chem Soc (2006) 0.95
A new tin-free source of amidyl radicals. Org Lett (2002) 0.92
A short total synthesis of (+/-)-aspidospermidine. Org Lett (2006) 0.91
Palladium-catalyzed intramolecular asymmetric hydroamination of alkynes. J Am Chem Soc (2004) 0.90
Copper(II) complexes of inverted porphyrin and its methylated derivatives. Inorg Chem (2000) 0.90
Catalytic asymmetric intramolecular aminopalladation: enantioselective synthesis of vinyl-substituted 2-oxazolidinones, 2-imidazolidinones, and 2-pyrrolidinones. J Am Chem Soc (2002) 0.90
Efficient acyclic stereocontrol using the tethered aminohydroxylation reaction. Org Lett (2004) 0.89
Copper-catalyzed intermolecular hydroamination of alkenes. Org Lett (2006) 0.89
Hydroamination/cyclization of aminoalkenes using cationic zirconocene and titanocene catalysts. Angew Chem Int Ed Engl (2004) 0.88
The tertiary sulfonamide as a latent directed-metalation group: Ni0-catalyzed reductive cleavage and cross-coupling reactions of aryl sulfonamides with grignard reagents. Angew Chem Int Ed Engl (2004) 0.85
Radical [3+2] annulation of N-allyl-N-chlorotosylamide with alkenes via atom-transfer process. Org Lett (2001) 0.84
Et3B-induced radical addition of N,N-dichlorosulfonamide to alkenes and pyrrolidine formation via radical annulation. J Org Chem (2003) 0.83
Development of an efficient procedure for indole ring synthesis from 2-ethynylaniline derivatives catalyzed by CuII salts and its application to natural product synthesis. J Org Chem (2004) 0.81
Chelating diamide based rate enhancement of intramolecular alkene hydroaminations catalyzed by a neutral Sc(III) complex. Org Lett (2005) 0.80
Intramolecular hydrogen abstraction promoted by amidyl radicals. Evidence for electronic factors in the nucleophilic cyclization of ambident amides to oxocarbenium ions. Org Lett (2005) 0.78
[(18)F]T807, a novel tau positron emission tomography imaging agent for Alzheimer's disease. Alzheimers Dement (2013) 2.31
Copper(II)-catalyzed enantioselective intramolecular carboamination of alkenes. J Am Chem Soc (2007) 1.94
Copper(II) acetate promoted intramolecular diamination of unactivated olefins. J Am Chem Soc (2005) 1.82
Copper catalyzed enantioselective intramolecular aminooxygenation of alkenes. J Am Chem Soc (2008) 1.75
Copper(II) acetate promoted oxidative cyclization of arylsulfonyl-o-allylanilines. Org Lett (2004) 1.65
A highly selective and specific PET tracer for imaging of tau pathologies. J Alzheimers Dis (2012) 1.56
Copper(II) carboxylate promoted intramolecular diamination of terminal alkenes: improved reaction conditions and expanded substrate scope. Org Lett (2007) 1.49
Copper-catalyzed enantioselective intramolecular alkene amination/intermolecular Heck-type coupling cascade. J Am Chem Soc (2012) 1.25
Catalytic enantioselective alkene aminohalogenation/cyclization involving atom transfer. Angew Chem Int Ed Engl (2012) 1.22
Heterocycle synthesis by copper facilitated addition of heteroatoms to alkenes, alkynes and arenes. Chem Soc Rev (2007) 1.21
Diastereoselective pyrrolidine synthesis via copper promoted intramolecular aminooxygenation of alkenes: formal synthesis of (+)-monomorine. Org Lett (2009) 1.20
Copper(II) carboxylate-promoted intramolecular carboamination of alkenes for the synthesis of polycyclic lactams. Org Lett (2007) 1.13
Copper-promoted and copper-catalyzed intermolecular alkene diamination. Angew Chem Int Ed Engl (2010) 1.08
Evidence for alkene cis-aminocupration, an aminooxygenation case study: kinetics, EPR spectroscopy, and DFT calculations. Chemistry (2012) 1.03
Copper-catalyzed intramolecular alkene carboetherification: synthesis of fused-ring and bridged-ring tetrahydrofurans. J Am Chem Soc (2012) 1.00
Total synthesis of (S)-(+)-tylophorine via enantioselective intramolecular alkene carboamination. J Org Chem (2008) 0.99
Stereoselective Copper-Catalyzed Intramolecular Alkene Aminooxygenation: Effects of Substrate and Ligand Structure on Selectivity. European J Org Chem (2011) 0.96
Diastereo- and enantioselective copper-catalyzed intramolecular carboamination of alkenes for the synthesis of hexahydro-1H-benz[f]indoles. Org Lett (2010) 0.94
Copper(II)-Catalyzed Aminooxygenation and Carboamination of N-Aryl-2-allylanilines. Adv Synth Catal (2009) 0.94
Stereoselective isoxazolidine synthesis via copper-catalyzed alkene aminooxygenation. J Org Chem (2012) 0.89
Mechanistic analysis and optimization of the copper-catalyzed enantioselective intramolecular alkene aminooxygenation. J Org Chem (2012) 0.89
Copper-catalyzed oxidative amination and allylic amination of alkenes. Chemistry (2013) 0.89
Multigram Synthesis of a Chiral Substituted Indoline Via Copper-Catalyzed Alkene Aminooxygenation. Synthesis (Stuttg) (2012) 0.88
Design and synthesis of a 3,4-dehydroproline amide discovery library. J Comb Chem (2007) 0.88
Stereoselective synthesis of morpholines via copper-promoted oxyamination of alkenes. Org Lett (2012) 0.88
Synthesis of hydroxylated bicyclic amino acids from L-tyrosine: octahydro-1H-indole carboxylates. J Org Chem (2008) 0.86
Copper-catalyzed oxidative Heck reactions between alkyltrifluoroborates and vinyl arenes. Org Lett (2013) 0.85
Chiral Indoline Synthesis Via Enantioselective Intramolecular Copper-Catalyzed Alkene Hydroamination. Organometallics (2012) 0.84
Cellular and molecular effects of alpha-tocopheryloxybutyrate: lessons for the design of vitamin E analog for cancer prevention. Anticancer Res (2005) 0.81
A computational study of the copper(II)-catalyzed enantioselective intramolecular aminooxygenation of alkenes. J Org Chem (2013) 0.79
Enantioselective copper-catalyzed carboetherification of unactivated alkenes. Angew Chem Int Ed Engl (2014) 0.78
Alpha-vitamin E derivative, RRR-alpha-tocopheryloxybutyric acid inhibits the proliferation of prostate cancer cells. Asian J Androl (2007) 0.76
In vitro and in vivo anticancer effects of the novel vitamin E ether analogue RRR-alpha-tocopheryloxybutyl sulfonic acid in prostate cancer. Clin Cancer Res (2009) 0.76