Katherine A Rouleau

Author PubWeight™ 7.14^‹?›

Rank	Title	Journal	Year	PubWeight™‹?›
1	Acridone-based inhibitors of inosine 5'-monophosphate dehydrogenase: discovery and SAR leading to the identification of N-(2-(6-(4-ethylpiperazin-1-yl)pyridin-3-yl)propan-2-yl)-2- fluoro-9-oxo-9,10-dihydroacridine-3-carboxamide (BMS-566419).	J Med Chem	2007	0.91
2	Rapid synthesis of triazine inhibitors of inosine monophosphate dehydrogenase.	Bioorg Med Chem Lett	2002	0.83
3	Discovery of N-[2-[2-[[3-methoxy-4-(5-oxazolyl)phenyl]amino]-5-oxazolyl]phenyl]-N-methyl-4- morpholineacetamide as a novel and potent inhibitor of inosine monophosphate dehydrogenase with excellent in vivo activity.	J Med Chem	2002	0.83
4	Novel indole-based inhibitors of IMPDH: introduction of hydrogen bond acceptors at indole C-3.	Bioorg Med Chem Lett	2003	0.77
5	Quinolone-based IMPDH inhibitors: introduction of basic residues on ring D and SAR of the corresponding mono, di and benzofused analogues.	Bioorg Med Chem Lett	2003	0.77
6	The TosMIC approach to 3-(oxazol-5-yl) indoles: application to the synthesis of indole-based IMPDH inhibitors.	Bioorg Med Chem Lett	2002	0.77
7	Identification of novel and potent isoquinoline aminooxazole-based IMPDH inhibitors.	Bioorg Med Chem Lett	2003	0.76
8	3-cyanoindole-based inhibitors of inosine monophosphate dehydrogenase: synthesis and initial structure-activity relationships.	Bioorg Med Chem Lett	2003	0.76
9	Inhibitors of inosine monophosphate dehydrogenase: SARs about the N-[3-Methoxy-4-(5-oxazolyl)phenyl moiety.	Bioorg Med Chem Lett	2003	0.76