Published in Org Lett on March 22, 2008
Palladium(II)-catalyzed C-H activation/C-C cross-coupling reactions: versatility and practicality. Angew Chem Int Ed Engl (2009) 5.09
Palladium(II)-catalyzed ortho alkylation of benzoic acids with alkyl halides. Angew Chem Int Ed Engl (2009) 1.22
A copper-catalyzed, pH-neutral construction of high-enantiopurity peptidyl ketones from peptidic s-acylthiosalicylamides in air at room temperature. Angew Chem Int Ed Engl (2009) 0.96
Chemo- and regioselective C(sp³)-H arylation of unactivated allylarenes by deprotonative cross-coupling. Angew Chem Int Ed Engl (2014) 0.93
Chemoselective Palladium-Catalyzed Deprotonative Arylation/[1,2]-Wittig Rearrangement of Pyridylmethyl Ethers. Chem Sci (2015) 0.82
Synthesis of (diarylmethyl)amines using Ni-catalyzed arylation of C(sp(3))-H bonds. Chem Sci (2015) 0.82
Palladium-Catalyzed Benzylic C-H Arylation of Azaarylmethylamines. Org Lett (2015) 0.79
Palladium-Catalyzed Benzylic Arylation of Pyridylmethyl Silyl Ethers: One-Pot Synthesis of Aryl(pyridyl)methanols. Org Lett (2016) 0.77
Aryl Bromides and Aryl Chlorides for the Direct Arylation of Benzylic Amines Mediated by Ruthenium(II). European J Org Chem (2013) 0.77
Stereoselective cyclopropanation reactions. Chem Rev (2003) 3.15
Synthesis of pyridine and dihydropyridine derivatives by regio- and stereoselective addition to N-activated pyridines. Chem Rev (2012) 1.63
Nucleophilic addition to 3-substituted pyridinium salts: expedient syntheses of (-)-L-733,061 and (-)-CP-99,994. Org Lett (2004) 1.13
Nucleophilic addition of phenol derivatives to methyl 1-nitrocyclopropanecarboxylates. J Org Chem (2008) 1.09
Palladium-catalyzed direct C-h arylation of N-iminopyridinium ylides: application to the synthesis of (+/-)-anabasine. J Am Chem Soc (2007) 1.08
Experimental evidence for the all-up reactive conformation of chiral rhodium(II) carboxylate catalysts: enantioselective synthesis of cis-cyclopropane alpha-amino acids. J Am Chem Soc (2009) 1.06
Asymmetric, catalytic synthesis of alpha-chiral amines using a novel bis(phosphine) monoxide chiral ligand. J Am Chem Soc (2003) 1.04
Stereoselective synthesis of pyridinones: application to the synthesis of (-)-barrenazines. Org Lett (2006) 1.01
Cycloadditions of aromatic azomethine imines with 1,1-cyclopropane diesters. Org Lett (2008) 0.99
Controlled and chemoselective reduction of secondary amides. J Am Chem Soc (2010) 0.99
Total synthesis of (+)-cystothiazole A. Org Lett (2003) 0.97
Highly chemoselective metal-free reduction of tertiary amides. J Am Chem Soc (2007) 0.97
trans-Directing ability of amide groups in cyclopropanation: application to the asymmetric cyclopropanation of alkenes with diazo reagents bearing two carboxy groups. Angew Chem Int Ed Engl (2008) 0.95
TfNH2 as achiral hydrogen-bond donor additive to enhance the selectivity of a transition metal catalyzed reaction. Highly enantio- and diastereoselective rhodium-catalyzed cyclopropanation of alkenes using alpha-cyano diazoacetamide. J Am Chem Soc (2009) 0.95
Chemoselective synthesis of ketones and ketimines by addition of organometallic reagents to secondary amides. Nat Chem (2012) 0.94
Catalytic asymmetric addition of diorganozinc reagents to N-phosphinoylalkylimines. Proc Natl Acad Sci U S A (2004) 0.93
Convenient one-pot synthesis of (E)-beta-aryl vinyl halides from benzyl bromides and dihalomethanes. Org Lett (2008) 0.93
Stereoselective synthesis of 2,6-disubstituted 3-piperidinols: application to the expedient synthesis of (+)-julifloridine. Org Lett (2005) 0.89
Complexation promoted additions to N-benzoyliminopyridinium ylides. A novel and highly regioselective approach to polysubstituted piperidines. J Am Chem Soc (2003) 0.88
Total synthesis of (+)-lepadin B: stereoselective synthesis of nonracemic polysubstituted hydroquinolines using an RC-ROM process. J Am Chem Soc (2008) 0.88
Catalytic asymmetric synthesis of alpha,alpha,alpha-trifluoromethylamines by the copper-catalyzed nucleophilic addition of diorganozinc reagents to imines. Org Lett (2006) 0.88
A mild procedure for the Lewis acid-catalyzed ring-opening of activated cyclopropanes with amine nucleophiles. Org Lett (2008) 0.87
Highly efficient synthesis of O-(2,4-dinitrophenyl)hydroxylamine. Application to the synthesis of substituted N-benzoyliminopyridinium ylides. J Org Chem (2003) 0.87
Tetraarylphosphonium salts as solubility-control groups: phosphonium-supported triphenylphosphine and azodicarboxylate reagents. Angew Chem Int Ed Engl (2006) 0.87
Catalytic enantioselective addition of dialkylzinc to N-diphenylphosphinoylimines. A practical synthesis of alpha-chiral amines. J Am Chem Soc (2003) 0.87
Improved procedure for the synthesis of gem-diiodoalkanes by the alkylation of diiodomethane. scope and limitations. J Org Chem (2008) 0.87
Iron-catalyzed direct arylation through an aryl radical transfer pathway. J Am Chem Soc (2010) 0.86
Structure and reactivity of "unusual" N-heterocyclic carbene (NHC) palladium complexes synthesized from imidazolium salts. J Am Chem Soc (2004) 0.86
Diastereoselective zinco-cyclopropanation of chiral allylic alcohols with gem-dizinc carbenoids. J Am Chem Soc (2005) 0.86
General method for the expedient synthesis of salt-free diorganozinc reagents using zinc methoxide. J Am Chem Soc (2008) 0.85
Expedient synthesis of cyclopropane alpha-amino acids by the catalytic asymmetric cyclopropanation of alkenes using iodonium ylides derived from methyl nitroacetate. J Am Chem Soc (2005) 0.85
Catalytic asymmetric hydrogenation of N-iminopyridinium ylides: expedient approach to enantioenriched substituted piperidine derivatives. J Am Chem Soc (2005) 0.85
Iodomethylzinc phosphates: powerful reagents for the cyclopropanation of alkenes. J Am Chem Soc (2005) 0.85
Asymmetric Rh(II)-catalyzed cyclopropanation of alkenes with diacceptor diazo compounds: p-methoxyphenyl ketone as a general stereoselectivity controlling group. J Am Chem Soc (2011) 0.85
Electrolytic macrocyclizations: scalable synthesis of a diazonamide-based drug development candidate. Angew Chem Int Ed Engl (2015) 0.85
Dual role of silanol groups in cyclopropanation and Hiyama-Denmark cross-coupling reactions. Org Lett (2010) 0.84
Intramolecular pyridine activation-dearomatization reaction: highly stereoselective synthesis of polysubstituted indolizidines and quinolizidines. Org Lett (2009) 0.84
A Diels-Alder approach to the stereoselective synthesis of 2,3,5,6-tetra- and 2,3,4,5,6-pentasubstituted piperidines. Org Lett (2005) 0.84
Probing the importance of the hemilabile site of bis(phosphine) monoxide ligands in the copper-catalyzed addition of diethylzinc to N-phosphinoylimines: discovery of new effective chiral ligands. J Org Chem (2008) 0.84
Grob fragmentation of 2-azabicyclo[2.2.2]oct-7-ene: tool for the stereoselective synthesis of polysubstituted piperidines. J Org Chem (2012) 0.83
Formal synthesis of belactosin A and hormaomycin via a diastereoselective intramolecular cyclopropanation of an alpha-nitro diazoester. Org Lett (2010) 0.83
Direct functionalization processes: a journey from palladium to copper to iron to nickel to metal-free coupling reactions. Acc Chem Res (2012) 0.83
Enantioselective synthesis of 1,2,3-trisubstituted cyclopropanes using gem-dizinc reagents. J Am Chem Soc (2009) 0.83
Asymmetric total synthesis of (+)-luciduline: toward a general approach to related Lycopodium alkaloids. J Org Chem (2011) 0.82
Doubly activated cyclopropanes as synthetic precursors for the preparation of 4-nitro- and 4-cyano-dihydropyrroles and pyrroles. Org Lett (2005) 0.82
General method for the synthesis of phenyliodonium ylides from malonate esters: easy access to 1,1-cyclopropane diesters. J Org Chem (2009) 0.82
New methodology toward chiral, non-racemic 2,5-cis-substituted piperidines via Suzuki cross-coupling. Org Lett (2006) 0.82
An expedient and practical method for the synthesis of a diverse series of cyclopropane alpha-amino acids and amines. J Org Chem (2004) 0.82
Stereoselective Rh2(S-IBAZ)4-catalyzed cyclopropanation of alkenes, alkynes, and allenes: asymmetric synthesis of diacceptor cyclopropylphosphonates and alkylidenecyclopropanes. J Am Chem Soc (2013) 0.81
Intramolecular Simmons-Smith cyclopropanation. Studies into the reactivity of alkyl-substituted zinc carbenoids, effect of directing groups and synthesis of bicyclo[n.1.0]alkanes. J Am Chem Soc (2010) 0.81
Synthesis of 2-substituted pyrazolo[1,5-a]pyridines through cascade direct alkenylation/cyclization reactions. Org Lett (2010) 0.81
trans-Directing ability of the amide group: enabling the enantiocontrol in the synthesis of 1,1-dicarboxy cyclopropanes. Reaction development, scope, and synthetic applications. J Org Chem (2009) 0.81
Stereoselective synthesis of 2,3,6-trisubstituted tetrahydropyridines via Tf(2)O-mediated Grob fragmentation: access to indolizidines (-)-209I and (-)-223J. J Org Chem (2010) 0.81
Umpolung direct arylation reactions: facile process requiring only catalytic palladium and substoichiometric amount of silver salts. J Am Chem Soc (2010) 0.80
Potassium tert-butoxide promoted intramolecular arylation via a radical pathway. Org Lett (2011) 0.80
Highly regioselective intermolecular arylation of 1,2,3,4-tetrahydropyridines. Org Lett (2008) 0.80
Expedient stereoselective synthesis of coronafacic acid through intramolecular Diels-Alder cyclization. J Org Chem (2007) 0.80
Nickel(0)/NaHMDS adduct-mediated intramolecular alkylation of unactivated arenes via a homolytic aromatic substitution mechanism. Chem Commun (Camb) (2012) 0.79
Synthesis of enantioenriched allenes from 1,1-cyclopropanediesters. Org Lett (2010) 0.79
Catalytic enantioselective reduction of beta,beta-disubstituted vinyl phenyl sulfones by using bisphosphine monoxide ligands. Angew Chem Int Ed Engl (2007) 0.79
Evidence for the structure of the enantioactive ligand in the phosphine-copper-catalyzed addition of diorganozinc reagents to imines. Angew Chem Int Ed Engl (2004) 0.79
Application of the chiral bis(phosphine) monoxide ligand to catalytic enantioselective addition of dialkylzinc reagents to beta-nitroalkenes. Org Lett (2007) 0.78
Silver-promoted, palladium-catalyzed direct arylation of cyclopropanes: facile access to spiro 3,3'-cyclopropyl oxindoles. Org Lett (2013) 0.78
In situ generation of zinc carbenoids from diazo compounds and zinc salts: asymmetric synthesis of 1,2,3-substituted cyclopropanes. J Am Chem Soc (2009) 0.78
Hypervalent iodine(III) reagents as safe alternatives to alpha-nitro-alpha-diazocarbonyls. Org Lett (2003) 0.78
Removal, recovery, and recycling of triarylphosphonium-supported tin reagents for various organic transformations. Org Lett (2007) 0.78
Stereoselective syntheses of L-pipecolic acid and (2S,3S)-3-hydroxypipecolic acid from a chiral N-imino-2-phenyl-1,2-dihydropyridine intermediate. J Org Chem (2010) 0.78
C-H functionalization of cyclopropanes: a practical approach employing a picolinamide auxiliary. Org Lett (2013) 0.78
[4+2] Cycloaddition of 2-substituted 1,2-dihydropyridines with nitrosobenzene: asymmetric synthesis of trans-2-substituted 3-amino-1,2,3,6-tetrahydropyridines. J Org Chem (2005) 0.78
Catalytic enantioselective addition of diorganozinc reagents to vinyl sulfones. Org Lett (2008) 0.78
Silver ion-induced Grob fragmentation of gamma-amino iodides: highly stereoselective synthesis of polysubstituted piperidines. Org Lett (2008) 0.77
Palladium-catalyzed synthesis of functionalized tetraarylphosphonium salts. J Org Chem (2007) 0.77
Enantio- and diastereoselective iodocyclopropanation of allylic alcohols by using a substituted zinc carbenoid. Chemistry (2009) 0.76
Improved zinc-catalyzed Simmons-Smith reaction: access to various 1,2,3-trisubstituted cyclopropanes. Org Lett (2014) 0.76
Tetraarylphosphonium-supported carbodiimide reagents: synthesis, structure optimization and applications. J Org Chem (2008) 0.76
Transition metal-catalyzed cyclopropanation of alkenes in water: catalyst efficiency and in situ generation of the diazo reagent. Org Lett (2002) 0.76
Highly efficient two-step synthesis of C-sp3-centered geminal diiodides. Org Lett (2004) 0.76
Highly enantioselective synthesis of 1,2,3-substituted cyclopropanes by using α-Iodo- and α-chloromethylzinc carbenoids. Chemistry (2012) 0.76
Organic chemistry: Short cuts to complexity. Nature (2008) 0.75
Copper-catalyzed direct alkenylation of N-iminopyridinium ylides. Angew Chem Int Ed Engl (2010) 0.75
Orthoacylimines: a new class of chiral auxiliaries for nucleophilic addition of organolithium reagents to imines. J Org Chem (2003) 0.75
One-pot synthesis of 3,4,5-trisubstituted 1,2,4-triazoles via the addition of hydrazides to activated secondary amides. Org Lett (2015) 0.75
Tetraarylphosphonium salts as soluble supports for the synthesis of small molecules. Angew Chem Int Ed Engl (2007) 0.75
One-pot synthesis of 1-iodoalkynes and trisubstituted alkenes from benzylic and allylic bromides. Org Lett (2012) 0.75
Tetraarylphosphonium salts as soluble supports for oxidative catalysts and reagents. J Org Chem (2009) 0.75
Triflic anhydride mediated synthesis of imidazo[1,5-a]azines. Org Lett (2013) 0.75
Synthesis of N-diphenylphosphinoylimines using the Kresze reaction. J Org Chem (2005) 0.75
Multicomponent one-pot procedure for the synthesis of free alpha-chiral amines from aldehydes. J Org Chem (2005) 0.75
Directed functionalization of 1,2-dihydropyridines: stereoselective synthesis of 2,6-disubstituted piperidines. Chem Commun (Camb) (2014) 0.75
Highly enantioselective Simmons-Smith fluorocyclopropanation of allylic alcohols via the halogen scrambling strategy of zinc carbenoids. J Am Chem Soc (2013) 0.75
Use of achiral additives to increase the stereoselectivity in Rh(II)-catalyzed cyclopropanations. Chem Commun (Camb) (2010) 0.75
Structure and reactivity of a new anionic N-heterocyclic carbene silver(I) complex. Chem Commun (Camb) (2005) 0.75
Preparation of a storable zinc carbenoid species and its application in cyclopropanation, chain extension, and [2,3]-sigmatropic rearrangement reactions. J Org Chem (2010) 0.75
Defying ring strain: new approaches to cyclopropanes. Angew Chem Int Ed Engl (2010) 0.75