Robert A Domaoal

Author PubWeight™ 15.21^‹?›

Top papers

Rank	Title	Journal	Year	PubWeight™‹?›
1	Computationally-guided optimization of a docking hit to yield catechol diethers as potent anti-HIV agents.	J Med Chem	2011	1.68
2	Optimization of azoles as anti-human immunodeficiency virus agents guided by free-energy calculations.	J Am Chem Soc	2008	1.39
3	Optimization of pyrimidinyl- and triazinyl-amines as non-nucleoside inhibitors of HIV-1 reverse transcriptase.	Bioorg Med Chem Lett	2006	1.38
4	FEP-guided selection of bicyclic heterocycles in lead optimization for non-nucleoside inhibitors of HIV-1 reverse transcriptase.	J Am Chem Soc	2006	1.36
5	From docking false-positive to active anti-HIV agent.	J Med Chem	2007	1.16
6	An antibody-recruiting small molecule that targets HIV gp120.	J Am Chem Soc	2009	1.15
7	Efficient discovery of potent anti-HIV agents targeting the Tyr181Cys variant of HIV reverse transcriptase.	J Am Chem Soc	2011	1.10
8	Eastern extension of azoles as non-nucleoside inhibitors of HIV-1 reverse transcriptase; cyano group alternatives.	Bioorg Med Chem Lett	2010	1.06
9	Discovery of wild-type and Y181C mutant non-nucleoside HIV-1 reverse transcriptase inhibitors using virtual screening with multiple protein structures.	J Chem Inf Model	2009	0.96
10	Discovery of dimeric inhibitors by extension into the entrance channel of HIV-1 reverse transcriptase.	Bioorg Med Chem Lett	2012	0.94
11	Identification of a beta3-peptide HIV fusion inhibitor with improved potency in live cells.	Bioorg Med Chem Lett	2009	0.87
12	Quasi-Biomimetic Ring Contraction Catalyzed by a Cysteine-Based Nucleophile: Total Synthesis of Sch-642305, Some Analogs and their Putative anti-HIV Activities.	Chem Sci	2011	0.82
13	K65R and K65A substitutions in HIV-1 reverse transcriptase enhance polymerase fidelity by decreasing both dNTP misinsertion and mispaired primer extension efficiencies.	J Mol Biol	2010	0.81
14	L12 enhances gonococcal transcytosis of polarized Hec1B cells via the lutropin receptor.	Microb Pathog	2002	0.79