Rank | Title | Journal | Year | PubWeight™‹?› |
---|---|---|---|---|
1 | MEK inhibitors: the chemistry and biological activity of U0126, its analogs, and cyclization products. | Bioorg Med Chem Lett | 1998 | 2.61 |
2 | Nonpeptide angiotensin II receptor antagonists: the discovery of a series of N-(biphenylylmethyl)imidazoles as potent, orally active antihypertensives. | J Med Chem | 1991 | 1.50 |
3 | Pyrazoles, 1,2,4-triazoles, and tetrazoles as surrogates for cis-amide bonds in boronate ester thrombin inhibitors. | Bioorg Med Chem Lett | 1998 | 0.77 |
4 | EXP597, a nonpeptide angiotensin II receptor antagonist with high affinities for the angiotensin AT1 and AT2 receptor subtypes. | Eur J Pharmacol | 1994 | 0.75 |