Published in Org Biomol Chem on February 11, 2009
Identification of γ-AApeptides with potent and broad-spectrum antimicrobial activity. Chem Commun (Camb) (2011) 1.26
Synthesis of libraries of peptidomimetic compounds containing a 2-oxopiperazine unit in the main chain. Org Biomol Chem (2013) 1.05
Rapid photoassisted access to N,O,S-polyheterocycles with benzoazocine and hydroquinoline cores: intramolecular cycloadditions of photogenerated azaxylylenes. Angew Chem Int Ed Engl (2011) 1.03
Peptoid-based PET imaging of vascular endothelial growth factor receptor (VEGFR) expression. Am J Nucl Med Mol Imaging (2011) 1.01
Adding diverse noncanonical backbones to rosetta: enabling peptidomimetic design. PLoS One (2013) 0.94
Extraordinarily robust polyproline type I peptoid helices generated via the incorporation of α-chiral aromatic N-1-naphthylethyl side chains. J Am Chem Soc (2011) 0.93
Solid-phase submonomer synthesis of peptoid polymers and their self-assembly into highly-ordered nanosheets. J Vis Exp (2011) 0.88
Development of homomultimers and heteromultimers of lung cancer-specific peptoids. Biopolymers (2011) 0.85
In vivo biodistribution and small animal PET of (64)Cu-labeled antimicrobial peptoids. Bioconjug Chem (2012) 0.84
Analogs of the CLV3 peptide: synthesis and structure-activity relationships focused on proline residues. Plant Cell Physiol (2010) 0.83
Novel peptoid building blocks: synthesis of functionalized aromatic helix-inducing submonomers. Org Lett (2010) 0.83
Androgen receptor antagonism by divalent ethisterone conjugates in castrate-resistant prostate cancer cells. ACS Chem Biol (2012) 0.83
End-to-end conformational communication through a synthetic purinergic receptor by ligand-induced helicity switching. Nat Chem (2013) 0.82
A peptoid ribbon secondary structure. Angew Chem Int Ed Engl (2013) 0.80
Targeting the androgen receptor with steroid conjugates. J Med Chem (2014) 0.79
Oxetanyl peptides: novel peptidomimetic modules for medicinal chemistry. Org Lett (2014) 0.79
Design and conformational analysis of peptoids containing N-hydroxy amides reveals a unique sheet-like secondary structure. Biopolymers (2011) 0.78
Unbiased Selection of Peptide-Peptoid Hybrids Specific for Lung Cancer Compared to Normal Lung Epithelial Cells. ACS Chem Biol (2015) 0.78
A chemically synthesized peptoid-based drag-tag enhances free-solution DNA sequencing by capillary electrophoresis. Biopolymers (2011) 0.78
Functional, metal-based crosslinkers for α-helix induction in short peptides. Chem Sci (2013) 0.78
Synthesis and Characterization of Amphiphilic Cyclic Diblock Copolypeptoids from N-Heterocyclic Carbene-Mediated Zwitterionic Polymerization of N-Substituted N-carboxyanhydride. Macromolecules (2011) 0.78
Synthesis of the first examples of iminosugar clusters based on cyclopeptoid cores. Beilstein J Org Chem (2014) 0.77
Identification of lipid-phosphatidylserine (PS) as the target of unbiasedly selected cancer specific peptide-peptoid hybrid PPS1. Oncotarget (2016) 0.77
Construction and conformational behavior of peptoids with cis-amide bond geometry: design of a peptoid with alternate φ, ψ values of inverse PP-II/PP-II and PP-I structures. J Mol Model (2014) 0.76
Consecutive isocyanide-based multicomponent reactions: synthesis of cyclic pentadepsipeptoids. Beilstein J Org Chem (2014) 0.76
NMEGylation: a novel modification to enhance the bioavailability of therapeutic peptides. Biopolymers (2011) 0.75
Molecular Design of Antifouling Polymer Brushes Using Sequence-Specific Peptoids. Adv Mater Interfaces (2015) 0.75
Development of a large peptoid-DOTA combinatorial library. Biopolymers (2016) 0.75
Novel C6-substituted 1,3,4-oxadiazinones as potential anti-cancer agents. Oncotarget (2015) 0.75
Conformational behavior of polyalanine peptides with and without protecting groups of varying chain lengths: population of PP-II structure! J Mol Model (2015) 0.75
Small molecule inhibitors of bacterial quorum sensing and biofilm formation. J Am Chem Soc (2005) 1.90
SIR1, an upstream component in auxin signaling identified by chemical genetics. Science (2003) 1.87
Modulation of bacterial quorum sensing with synthetic ligands: systematic evaluation of N-acylated homoserine lactones in multiple species and new insights into their mechanisms of action. J Am Chem Soc (2007) 1.86
Expanding dialogues: from natural autoinducers to non-natural analogues that modulate quorum sensing in Gram-negative bacteria. Chem Soc Rev (2008) 1.62
N-phenylacetanoyl-L-homoserine lactones can strongly antagonize or superagonize quorum sensing in Vibrio fischeri. ACS Chem Biol (2007) 1.39
Local and tunable n-->pi* interactions regulate amide isomerism in the peptoid backbone. J Am Chem Soc (2007) 1.29
Comparative analyses of N-acylated homoserine lactones reveal unique structural features that dictate their ability to activate or inhibit quorum sensing. Chembiochem (2008) 1.28
New strategies for the design of folded peptoids revealed by a survey of noncovalent interactions in model systems. J Am Chem Soc (2009) 1.27
Small molecules that modulate quorum sensing and control virulence in Pseudomonas aeruginosa. J Org Chem (2010) 1.21
Evaluation of a focused library of N-aryl L-homoserine lactones reveals a new set of potent quorum sensing modulators. Bioorg Med Chem Lett (2008) 1.20
Isovaleryl-homoserine lactone, an unusual branched-chain quorum-sensing signal from the soybean symbiont Bradyrhizobium japonicum. Proc Natl Acad Sci U S A (2011) 1.17
Chemical modification of reactive multilayered films fabricated from poly(2-alkenyl azlactone)s: design of surfaces that prevent or promote mammalian cell adhesion and bacterial biofilm growth. Biomacromolecules (2009) 1.15
Attenuation of quorum sensing in the pathogen Acinetobacter baumannii using non-native N-Acyl homoserine lactones. ACS Chem Biol (2012) 1.14
Highly potent inhibitors of quorum sensing in Staphylococcus aureus revealed through a systematic synthetic study of the group-III autoinducing peptide. J Am Chem Soc (2013) 1.10
Control of quorum sensing by a Burkholderia pseudomallei multidrug efflux pump. J Bacteriol (2007) 1.06
Synthetic ligands that activate and inhibit a quorum-sensing regulator in Pseudomonas aeruginosa. Bioorg Med Chem Lett (2007) 1.03
Characterization of structural elements in native autoinducing peptides and non-native analogues that permit the differential modulation of AgrC-type quorum sensing receptors in Staphylococcus aureus. Org Biomol Chem (2015) 1.03
Diversity-oriented synthesis of biaryl-containing medium rings using a one bead/one stock solution platform. J Am Chem Soc (2002) 1.00
Potent and selective synthetic modulators of a quorum sensing repressor in Pseudomonas aeruginosa identified from second-generation libraries of N-acylated L-homoserine lactones. Chembiochem (2011) 1.00
Design and synthesis of macrocyclic peptomers as mimics of a quorum sensing signal from Staphylococcus aureus. Org Lett (2008) 1.00
Rapid synthesis of diketopiperazine macroarrays via Ugi four-component reactions on planar solid supports. Chem Commun (Camb) (2006) 0.99
Competition studies confirm two major barriers that can preclude the spread of resistance to quorum-sensing inhibitors in bacteria. ACS Chem Biol (2014) 0.98
Expedient synthesis and design strategies for new peptoid construction. Org Lett (2005) 0.98
Rapid identification of antibacterial agents effective against Staphylococcus aureus using small-molecule macroarrays. Chem Biol (2007) 0.97
Construction of peptoids with all trans-amide backbones and peptoid reverse turns via the tactical incorporation of N-aryl side chains capable of hydrogen bonding. J Org Chem (2010) 0.96
Small molecule disruption of quorum sensing cross-regulation in pseudomonas aeruginosa causes major and unexpected alterations to virulence phenotypes. J Am Chem Soc (2015) 0.96
Thiolactone modulators of quorum sensing revealed through library design and screening. Bioorg Med Chem (2011) 0.95
Identification of synthetic inducers and inhibitors of the quorum-sensing regulator LasR in Pseudomonas aeruginosa by high-throughput screening. Appl Environ Microbiol (2010) 0.95
Small molecule macroarray construction via Ugi four-component reactions. Org Lett (2005) 0.94
Microwave-accelerated SPOT-synthesis on cellulose supports. Org Lett (2004) 0.94
Attenuation of virulence in pathogenic bacteria using synthetic quorum-sensing modulators under native conditions on plant hosts. ACS Chem Biol (2011) 0.94
Extraordinarily robust polyproline type I peptoid helices generated via the incorporation of α-chiral aromatic N-1-naphthylethyl side chains. J Am Chem Soc (2011) 0.93
Tuning peptoid secondary structure with pentafluoroaromatic functionality: a new design paradigm for the construction of discretely folded peptoid structures. J Am Chem Soc (2006) 0.93
Design, synthesis, and biological evaluation of abiotic, non-lactone modulators of LuxR-type quorum sensing. Bioorg Med Chem (2011) 0.93
2-Aminobenzimidazole derivatives strongly inhibit and disperse Pseudomonas aeruginosa biofilms. Angew Chem Int Ed Engl (2012) 0.92
Discovery of fluorescent cyanopyridine and deazalumazine dyes using small molecule macroarrays. Org Lett (2006) 0.91
Quorum sensing in bacterial species that use degenerate autoinducers can be tuned by using structurally identical non-native ligands. Chembiochem (2011) 0.91
Quorum-sensing signals in the microbial community of the cabbage white butterfly larval midgut. ISME J (2008) 0.90
Structural characterization of native autoinducing peptides and abiotic analogues reveals key features essential for activation and inhibition of an AgrC quorum sensing receptor in Staphylococcus aureus. J Am Chem Soc (2013) 0.89
Surface-mediated release of a synthetic small-molecule modulator of bacterial quorum sensing: gradual release enhances activity. Chem Commun (Camb) (2010) 0.89
Chemical methods to interrogate bacterial quorum sensing pathways. Org Biomol Chem (2012) 0.89
Efficient synthesis and evaluation of quorum-sensing modulators using small molecule macroarrays. Org Lett (2009) 0.89
Deciphering a protolanguage for bacteria-host communication. Nat Chem Biol (2008) 0.89
Synthesis and characterization of nitroaromatic peptoids: fine tuning peptoid secondary structure through monomer position and functionality. J Org Chem (2009) 0.87
Interception of quorum sensing in Staphylococcus aureus: a new niche for peptidomimetics. Org Biomol Chem (2006) 0.87
New and unexpected insights into the modulation of LuxR-type quorum sensing by cyclic dipeptides. ACS Chem Biol (2009) 0.87
Active efflux influences the potency of quorum sensing inhibitors in Pseudomonas aeruginosa. Chembiochem (2014) 0.86
N-Methyl and peptoid scans of an autoinducing peptide reveal new structural features required for inhibition and activation of AgrC quorum sensing receptors in Staphylococcus aureus. Chem Commun (Camb) (2014) 0.86
Surface coatings that promote rapid release of peptide-based AgrC inhibitors for attenuation of quorum sensing in Staphylococcus aureus. Adv Healthc Mater (2013) 0.83
Introduction to bacterial signals and chemical communication. Chem Rev (2011) 0.83
Improved small-molecule macroarray platform for the rapid synthesis and discovery of antibacterial chalcones. ACS Comb Sci (2011) 0.81
Small molecule macroarray construction via palladium-mediated carbon-carbon bond-forming reactions: highly efficient synthesis and screening of stilbene arrays. Chemistry (2010) 0.81
Plant responses to bacterial N-acyl L-homoserine lactones are dependent on enzymatic degradation to L-homoserine. ACS Chem Biol (2014) 0.81
Synthesis and application of an N-acylated l-homoserine lactone derivatized affinity matrix for the isolation of quorum sensing signal receptors. Bioorg Med Chem Lett (2011) 0.80
A peptoid ribbon secondary structure. Angew Chem Int Ed Engl (2013) 0.80
Efficient construction of diketopiperazine macroarrays through a cyclative-cleavage strategy and their evaluation as luminescence inhibitors in the bacterial symbiont Vibrio fischeri. J Comb Chem (2009) 0.80
Synthesis and biological evaluation of triazole-containing N-acyl homoserine lactones as quorum sensing modulators. Org Biomol Chem (2012) 0.79
Solid-phase and microwave-assisted syntheses of 2,5-diketopiperazines: small molecules with great potential. Comb Chem High Throughput Screen (2007) 0.79
Design and conformational analysis of peptoids containing N-hydroxy amides reveals a unique sheet-like secondary structure. Biopolymers (2011) 0.78
Non-native N-aroyl L-homoserine lactones are potent modulators of the quorum sensing receptor RpaR in Rhodopseudomonas palustris. Chembiochem (2013) 0.78
Surface-mediated release of a small-molecule modulator of bacterial biofilm formation: a non-bactericidal approach to inhibiting biofilm formation in Pseudomonas aeruginosa. Adv Healthc Mater (2013) 0.78
Unraveling the contributions of hydrogen-bonding interactions to the activity of native and non-native ligands in the quorum-sensing receptor LasR. Org Biomol Chem (2015) 0.76
Expedient construction of small molecule macroarrays via sequential palladium- and copper-mediated reactions and their ex situ biological testing. Chem Sci (2012) 0.75
N-[1-(Pentafluorophenyl)ethyl]acetamide. Acta Crystallogr C (2006) 0.75
Microwave-Facilitated SPOT-Synthesis of Antibacterial Dipeptoids. ACS Comb Sci (2017) 0.75