The discovery and optimization of hexahydro-2H-pyrano[3,2-c]quinolines (HHPQs) as potent and selective inhibitors of the mitotic kinesin-5.

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🔗 View Article (PMID 20149654)

Published in Bioorg Med Chem Lett on January 25, 2010

Authors

Kai Schiemann1, Dirk Finsinger, Frank Zenke, Christiane Amendt, Thorsten Knöchel, David Bruge, Hans-Peter Buchstaller, Ulrich Emde, Wolfgang Stähle, Soheila Anzali

Author Affiliations

1: MS-RTC-MedChem DA35, Merck Serono, Merck KGaA, Frankfurter Strasse 250, D-64293 Darmstadt, Germany. kai.schiemann@merck.de

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