Ronald J Doll

Author PubWeight™ 5.42^‹?›

Top papers

Rank	Title	Journal	Year	PubWeight™‹?›
1	Versatile templates for the development of novel kinase inhibitors: Discovery of novel CDK inhibitors.	Bioorg Med Chem Lett	2007	1.10
2	Aurora kinase inhibitors based on the imidazo[1,2-a]pyrazine core: fluorine and deuterium incorporation improve oral absorption and exposure.	J Med Chem	2010	0.95
3	Structure-guided discovery of cyclin-dependent kinase inhibitors.	Biopolymers	2008	0.91
4	Analysis of the ERK1,2 transcriptome in mammary epithelial cells.	Biochem J	2004	0.90
5	Pyrazolo[1,5-a]pyrimidines as orally available inhibitors of cyclin-dependent kinase 2.	Bioorg Med Chem Lett	2007	0.82
6	Mass spectrometric studies of potent inhibitors of farnesyl protein transferase--detection of pentameric noncovalent complexes.	J Mass Spectrom	2008	0.76
7	Inhibition of cyclin-dependent kinases - a review of the recent patent literature.	Recent Pat Anticancer Drug Discov	2006	0.76
8	Towards the second generation of Boceprevir: Dithianes as an alternative P2 substituent for 2,2-dimethyl cycloproyl proline in HCV NS3 protease inhibitors.	Bioorg Med Chem Lett	2010	0.75
9	Guiding farnesyltransferase inhibitors from an ECLiPS library to the catalytic zinc.	Bioorg Med Chem Lett	2005	0.75
10	Bioisosteric approach to the discovery of imidazo[1,2-a]pyrazines as potent Aurora kinase inhibitors.	Bioorg Med Chem Lett	2010	0.75
11	Exploring the role of bromine at C(10) of (+)-4-[2-[4-(8-chloro-3,10-dibromo- 6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridin-11(R)-yl)-1-piperidinyl]-2- oxoethyl]-1-piperidinecarboxamide (Sch-66336): the discovery of indolocycloheptapyridine inhibitors of farnesyl protein transferase.	J Med Chem	2002	0.75
12	Discovery of C-imidazole azaheptapyridine FPT inhibitors.	Bioorg Med Chem Lett	2009	0.75