Published in Chem Rev on August 10, 2011
Enantioselective Synthesis of Tetrahydroquinolines, Tetrahydroquinoxalines, and Tetrahydroisoquinolines via Pd-Catalyzed Alkene Carboamination Reactions. Chem Sci (2014) 0.94
Microwave-assisted Expeditious and Efficient Synthesis of Cyclopentene Ring-fused Tetrahydroquinoline Derivatives Using Three-component Povarov Reaction. Tetrahedron Lett (2013) 0.85
Enantioselective annulations for dihydroquinolones by in situ generation of azolium enolates. J Am Chem Soc (2014) 0.85
Application of a catalytic asymmetric Povarov reaction using chiral ureas to the synthesis of a tetrahydroquinoline library. ACS Comb Sci (2012) 0.83
Palladium-catalyzed picolinamide-directed iodination of remote ortho-C-H bonds of arenes: Synthesis of tetrahydroquinolines. Beilstein J Org Chem (2016) 0.82
Asymmetric Methods for the Synthesis of Flavanones, Chromanones, and Azaflavanones. European J Org Chem (2011) 0.82
A combined continuous microflow photochemistry and asymmetric organocatalysis approach for the enantioselective synthesis of tetrahydroquinolines. Beilstein J Org Chem (2013) 0.81
Adaptation of a small-molecule hydrogen-bond donor catalyst to an enantioselective hetero-Diels-Alder reaction hypothesized for brevianamide biosynthesis. Org Lett (2015) 0.77
A one-pot multicomponent strategy for stereospecific construction of tricyclic pyrrolo[1,2-a]quinolines. Chem Commun (Camb) (2012) 0.77
Asymmetric Brønsted acid-catalyzed aza-Diels-Alder reaction of cyclic C-acylimines with cyclopentadiene. Beilstein J Org Chem (2012) 0.77
Practical synthetic strategies towards lipophilic 6-iodotetrahydroquinolines and -dihydroquinolines. Beilstein J Org Chem (2016) 0.75
Dual C-H functionalization of N-aryl amines: synthesis of polycyclic amines via an oxidative Povarov approach. Org Lett (2014) 0.75
Synthesis and fungicidal activity of pyrazole derivatives containing 1,2,3,4-tetrahydroquinoline. Chem Cent J (2016) 0.75
Novel N-allyl/propargyl tetrahydroquinolines: Synthesis via Three-component Cationic Imino Diels-Alder Reaction, Binding Prediction, and Evaluation as Cholinesterase Inhibitors. Chem Biol Drug Des (2016) 0.75
Catalytic, Enantioselective, Intramolecular Sulfenoamination of Alkenes with Anilines. J Org Chem (2017) 0.75
(S)-Benzyl 3-phenyl-carbamoyl-1,2,3,4-tetra-hydro-isoquinoline-2-carboxyl-ate. Acta Crystallogr Sect E Struct Rep Online (2012) 0.75
Development of Novel 1,2,3,4-Tetrahydroquinoline Scaffolds as Potent NF-κB Inhibitors and Cytotoxic Agents. ACS Med Chem Lett (2016) 0.75
6-Methyl-2-oxo-N-(quinolin-6-yl)-2H-chromene-3-carboxamide: crystal structure and Hirshfeld surface analysis. Acta Crystallogr E Crystallogr Commun (2016) 0.75
Kinetic resolution of racemic 2-substituted 1,2-dihydroquinolines via asymmetric Cu-catalyzed borylation. Chem Sci (2017) 0.75
Selective cobalt nanoparticles for catalytic transfer hydrogenation of N-heteroarenes. Chem Sci (2017) 0.75
Concise and very efficient synthesis of the N-methylwelwistatin tetracyclic core based on an anionic domino process. Org Biomol Chem (2010) 1.06
Cerium(IV) ammonium nitrate is an excellent, general catalyst for the Friedländer and Friedländer-Borsche quinoline syntheses: very efficient access to the antitumor alkaloid luotonin A. J Org Chem (2009) 1.05
Cerium(IV) ammonium nitrate as a catalyst in organic synthesis. Chem Rev (2010) 0.99
Multicomponent reactions for the synthesis of pyrroles. Chem Soc Rev (2010) 0.97
Inhibitors of multidrug resistance to antitumor agents (MDR). Curr Med Chem (2002) 0.94
Brief total synthesis of the cell cycle inhibitor tryprostatin B and related preparation of its alanine analogue. J Org Chem (2003) 0.91
Discovery of a class of diketopiperazines as antiprion compounds. ChemMedChem (2010) 0.84
Efficient synthesis of N-prenylpyrroloindoline and N-prenylindole alkaloids based on a new four-reaction anionic domino process. Org Lett (2006) 0.84
Synthesis of benzo- and naphtho-fused bicyclo[n.3.1]alkane frameworks with a bridgehead nitrogen function by palladium-catalyzed intramolecular α'-arylation of α-nitroketones. Org Biomol Chem (2011) 0.81
Recent advances in the synthesis of pyrroles by multicomponent reactions. Chem Soc Rev (2014) 0.81
Privileged scaffolds in synthesis: 2,5-piperazinediones as templates for the preparation of structurally diverse heterocycles. Chem Soc Rev (2012) 0.79
Expedient, one-pot preparation of fused indoles via CAN-catalyzed three-component domino sequences and their transformation into polyheterocyclic compounds containing pyrrolo[1,2-a]azepine fragments. Org Biomol Chem (2010) 0.79
Environmental effects on the fluorescence behaviour of carbazole derivatization reagents. Luminescence (2005) 0.78
L-proline-catalyzed three-component domino [3+2+1] annulation for the regio- and diastereoselective synthesis of highly substituted thienothiopyrans containing three or four stereocenters. J Org Chem (2010) 0.78
Axial chirality of 4-arylpyrazolo[3,4-b]pyridines. Conformational analysis and absolute configuration. J Org Chem (2014) 0.78
Imaging of β-amyloid plaques by near infrared fluorescent tracers: a new frontier for chemical neuroscience. Chem Soc Rev (2015) 0.78
Domino reactions for the synthesis of bridged bicyclic frameworks: fast access to bicyclo[n.3.1]alkanes. Chem Soc Rev (2011) 0.78
Synthesis and structure-activity relationships of 1,5-diazaanthraquinones as antitumour compounds. Bioorg Med Chem Lett (2004) 0.78
Vinylation of nitro-substituted indoles, quinolinones, and anilides with grignard reagents. Chemistry (2009) 0.77
New types of reactivity of α,β-unsaturated N,N-dimethylhydrazones: chemodivergent diastereoselective synthesis of functionalized tetrahydroquinolines and hexahydropyrrolo[3,2-b]indoles. Chemistry (2012) 0.77
Three-component access to pyrroles promoted by the CAN-silver nitrate system under high-speed vibration milling conditions: a generalization of the Hantzsch pyrrole synthesis. Chem Commun (Camb) (2012) 0.76
New 5-unsubstituted dihydropyridines with improved CaV1.3 selectivity as potential neuroprotective agents against ischemic injury. J Med Chem (2014) 0.76
The first aza Diels-Alder reaction involving an alpha,beta-unsaturated hydrazone as the dienophile: stereoselective synthesis of C-4 functionalized 1,2,3,4-tetrahydroquinolines containing a quaternary stereocenter. Org Biomol Chem (2007) 0.76
Efficient generation of highly functionalized fused oxazepine frameworks based on a CAN-catalyzed four-component tetrahydropyridine synthesis/ring-closing metathesis sequence. J Org Chem (2009) 0.75
Modulation of prion by small molecules: from monovalent to bivalent and multivalent ligands. Curr Top Med Chem (2013) 0.75
Diastereoselective, multicomponent access to trans-2-aryl-4-arylamino-1,2,3,4-tetrahydroquinolines via an AA'BC sequential four-component reaction and their application to 2-arylquinoline synthesis. Org Biomol Chem (2012) 0.75
A one-pot sequence for the efficient synthesis of highly functionalized macrocarbocycles or bridged 2,8-dioxabicyclo[3.2.1]octanes from 1-nitrobicyclic compounds. Org Biomol Chem (2012) 0.75
A heavy metal- and oxidant-free, one-pot synthesis of pyridines and fused pyridines based on a Lewis acid-catalyzed multicomponent reaction. Chem Commun (Camb) (2014) 0.75
Synthesis of polysubstituted, functionalized quinolines through a metal-free domino process involving a C4–C3 functional group rearrangement. Org Lett (2012) 0.75
Unique Michael addition-initiated domino reaction for the stereoselective synthesis of functionalized macrolactones from alpha-nitroketones in water. Org Lett (2005) 0.75
A β-enaminone-initiated multicomponent domino reaction for the synthesis of indoloquinolizines and benzoquinolizines from acyclic precursors. Chemistry (2013) 0.75
1,3-dipolar cycloadditions from tricyclic hemiaminals. Synthesis of the quinocarcin core through catalyst-free generation of azomethine ylides. Org Biomol Chem (2011) 0.75
Antimycobacterial activity of novel 1,2,4-oxadiazole-pyranopyridine/chromene hybrids generated by chemoselective 1,3-dipolar cycloadditions of nitrile oxides. Bioorg Med Chem (2011) 0.75
Fully diastereoselective synthesis of polysubstituted, functionalized piperidines and decahydroquinolines based on multicomponent reactions catalyzed by cerium(IV) ammonium nitrate. Chemistry (2014) 0.75
Addition to "ITH14001, a CGP37157-Nimodipine Hybrid Designed to Regulate Calcium Homeostasis and Oxidative Stress, Exerts Neuroprotection in Cerebral Ischemia". ACS Chem Neurosci (2016) 0.75
Stereoselective synthesis of bicyclo[4.2.1]nonane skeletons by ring-closing metathesis: a new versatile methodology for the efficient assembly of functionalized cyclooctanoids. Org Lett (2004) 0.75
Synthesis of 1,4-diazepanes and benzo[b][1,4]diazepines by a domino process involving the in situ generation of an aza-Nazarov reagent. J Org Chem (2020) 0.75
Synthesis of a library of 5,6-unsubstituted 1,4-dihydropyridines based on a one-pot 4CR/elimination process and their application to the generation of structurally diverse fused nitrogen heterocycles. J Comb Chem (2010) 0.75
A very efficient cerium(IV) ammonium nitrate catalyzed, four-component synthesis of tetrahydropyridines and its application in the concise generation of functionalized homoquinolizine frameworks. Chemistry (2009) 0.75
Brief, efficient and highly diastereoselective synthesis of (±)-pumiliotoxin C based on the generation of an octahydroquinoline precursor via a four-component reaction. Chem Commun (Camb) (2011) 0.75
One-pot access to a library of structurally diverse nicotinamide derivatives via a three-component formal aza [3 + 3] cycloaddition. ACS Comb Sci (2012) 0.75
Palladium(II)-catalyzed intramolecular carboxypalladation-olefin insertion cascade: direct access to indeno[1,2-b]furan-2-ones. Org Biomol Chem (2015) 0.75