|
1
|
Human electrophysiological and pharmacological properties of XEN-D0101: a novel atrial-selective Kv1.5/IKur inhibitor.
|
J Cardiovasc Pharmacol
|
2013
|
0.93
|
|
2
|
Near-thorough QT study as part of a first-in-man study.
|
J Clin Pharmacol
|
2008
|
0.85
|
|
3
|
Identification of selective inhibitors of the potassium channel Kv1.1-1.2((3)) by high-throughput virtual screening and automated patch clamp.
|
ChemMedChem
|
2012
|
0.77
|
|
4
|
Prediction of ion channel activity using binary kernel discrimination.
|
J Chem Inf Model
|
2007
|
0.76
|
|
5
|
Naphthol derivatives as TRPV1 inhibitors for the treatment of urinary incontinence.
|
Bioorg Med Chem Lett
|
2011
|
0.75
|
|
6
|
Tetrahydro-naphthols as orally available TRPV1 inhibitors.
|
Bioorg Med Chem Lett
|
2012
|
0.75
|