Published in Future Med Chem on June 01, 2012
First three-dimensional structure of Toxoplasma gondii thymidylate synthase-dihydrofolate reductase: insights for catalysis, interdomain interactions, and substrate channeling. Biochemistry (2013) 0.95
Thermodynamic and functional characteristics of deep-sea enzymes revealed by pressure effects. Extremophiles (2013) 0.83
Structure of dihydromethanopterin reductase, a cubic protein cage for redox transfer. J Biol Chem (2014) 0.80
A Focused Screen Identifies Antifolates with Activity on Mycobacterium tuberculosis. ACS Infect Dis (2015) 0.77
Preliminary joint X-ray and neutron protein crystallographic studies of ecDHFR complexed with folate and NADP+. Acta Crystallogr F Struct Biol Commun (2014) 0.76
Structure-based analysis of Bacilli and plasmid dihydrofolate reductase evolution. J Mol Graph Model (2016) 0.75
Synthesis of 2,4,6-trisubstituted pyrimidines as antimalarial agents. Bioorg Med Chem (2005) 1.14
Syntheses of novel antimycobacterial combinatorial libraries of structurally diverse substituted pyrimidines by three-component solid-phase reactions. Bioorg Med Chem Lett (2002) 1.06
Bis and tris indole alkaloids from marine organisms: new leads for drug discovery. Curr Med Chem (2007) 1.04
A small library of trisubstituted pyrimidines as antimalarial and antitubercular agents. Bioorg Med Chem Lett (2005) 1.03
Dihydropyrido[2,3-d]pyrimidines as a new class of antileishmanial agents. Bioorg Med Chem (2005) 0.91
Substituted quinolinyl chalcones and quinolinyl pyrimidines as a new class of anti-infective agents. Eur J Med Chem (2008) 0.88
Antimalarial activity and synthesis of new trisubstituted pyrimidines. Bioorg Med Chem Lett (2005) 0.87
Discovery of new 1,3,5-triazine scaffolds with potent activity against Mycobacterium tuberculosis H37Rv. Eur J Med Chem (2010) 0.87
Synthesis of new 4-aminoquinolines and quinoline-acridine hybrids as antimalarial agents. Bioorg Med Chem Lett (2010) 0.87
Synthesis of 4-pyrido-6-aryl-2-substituted amino pyrimidines as a new class of antimalarial agents. Bioorg Med Chem (2005) 0.86
Synthesis of marine alkaloid: 8,9-dihydrocoscinamide B and its analogues as Novel class of antileishmanial agents. Bioorg Med Chem Lett (2007) 0.86
Discovery of a new class of natural product-inspired quinazolinone hybrid as potent antileishmanial agents. J Med Chem (2013) 0.85
Synthesis and antileishmanial activity of novel 2,4,6-trisubstituted pyrimidines and 1,3,5-triazines. Eur J Med Chem (2009) 0.83
Synthesis of 2-[3-(7-Chloro-quinolin-4-ylamino)-alkyl]-1-(substituted phenyl)-2,3,4,9-tetrahydro-1H-beta-carbolines as a new class of antimalarial agents. Bioorg Med Chem Lett (2008) 0.83
Skeletal diverse synthesis of N-fused polycyclic heterocycles via the sequence of Ugi-type MCR and CuI-catalyzed coupling/tandem Pictet-Spengler reaction. J Org Chem (2012) 0.82
A natural product inspired hybrid approach towards the synthesis of novel pentamidine based scaffolds as potential anti-parasitic agents. Bioorg Med Chem Lett (2012) 0.82
Access to indole- and pyrrole-fused diketopiperazines via tandem Ugi-4CR/intramolecular cyclization and its regioselective ring-opening by intermolecular transamidation. J Org Chem (2012) 0.81
Synthesis of 2-[3,5-substituted pyrazol-1-yl]-4,6-trisubstituted triazine derivatives as antimalarial agents. Bioorg Med Chem Lett (2005) 0.81
Synthesis and biological evaluation of new [1,2,4]triazino[5,6-b]indol-3-ylthio-1,3,5-triazines and [1,2,4]triazino[5,6-b]indol-3-ylthio-pyrimidines against Leishmania donovani. Eur J Med Chem (2010) 0.81
Antimalarial activity of 2,4,6-trisubstituted pyrimidines. Bioorg Med Chem Lett (2005) 0.80
Discovery of novel antileishmanial agents in an attempt to synthesize pentamidine-aplysinopsin hybrid molecule. J Med Chem (2009) 0.80
Synthesis and bioevaluation of novel 4-aminoquinoline-tetrazole derivatives as potent antimalarial agents. Eur J Med Chem (2013) 0.80
Cyanuric chloride catalyzed mild protocol for synthesis of biologically active dihydro/spiro quinazolinones and quinazolinone-glycoconjugates. J Org Chem (2012) 0.79
Synthesis and bioevaluation of hybrid 4-aminoquinoline triazines as a new class of antimalarial agents. Bioorg Med Chem Lett (2008) 0.79
Synthesis and cytotoxicity evaluation of (tetrahydro-beta-carboline)-1,3,5-triazine hybrids as anticancer agents. Eur J Med Chem (2010) 0.78
Molecular cloning and characterization of glucose-6-phosphate dehydrogenase from Brugia malayi. Parasitology (2013) 0.77
Syntheses of new substituted triazino tetrahydroisoquinolines and beta-carbolines as novel antileishmanial agents. Eur J Med Chem (2005) 0.77
Synthesis of oxalamide and triazine derivatives as a novel class of hybrid 4-aminoquinoline with potent antiplasmodial activity. Bioorg Med Chem (2009) 0.77
Synthesis of novel thiourea, thiazolidinedione and thioparabanic acid derivatives of 4-aminoquinoline as potent antimalarials. Bioorg Med Chem Lett (2009) 0.77
Synthesis of 9-anilinoacridine triazines as new class of hybrid antimalarial agents. Bioorg Med Chem Lett (2009) 0.77
Synthesis and biological evaluation of a new class of 4-aminoquinoline-rhodanine hybrid as potent anti-infective agents. Eur J Med Chem (2013) 0.77
Synthesis of substituted indole derivatives as a new class of antimalarial agents. Bioorg Med Chem Lett (2005) 0.76
Trioxaquines: hybrid molecules for the treatment of malaria. Drug News Perspect (2010) 0.76
4-anilinoquinoline triazines: a novel class of hybrid antimalarial agents. Eur J Med Chem (2010) 0.76
Syntheses of 2,4,6-trisubstituted triazines as antimalarial agents. Bioorg Med Chem Lett (2005) 0.76
A ligand-free Pd-catalyzed cascade reaction: an access to the highly diverse isoquinolin-1(2H)-one derivatives via isocyanide and Ugi-MCR synthesized amide precursors. Org Lett (2012) 0.76
Synthesis of 4-amino-5-cyano-2, 6-disubstituted pyrimidines as a potential antifilarial DNA topoisomerase II inhibitors. Med Chem (2008) 0.75
Synthesis and antibacterial evaluation of novel 8-fluoro Norfloxacin derivatives as potential probes for methicillin and vancomycin-resistant Staphylococcus aureus. Eur J Med Chem (2011) 0.75
2-Aminoimidazole, glycociamidine and 2-thiohydantoin-marine alkaloids as molecular inspirations for the development of lead structures. Curr Drug Targets (2011) 0.75
Synthesis of perspicamide A and related diverse analogues: their bioevaluation as potent antileishmanial agents. J Org Chem (2013) 0.75
Design and synthesis of a new class of 4-aminoquinolinyl- and 9-anilinoacridinyl Schiff base hydrazones as potent antimalarial agents. Chem Biol Drug Des (2014) 0.75
Solid support synthesis of 6-aryl-2-substituted pyrimidin-4-yl phenols as anti-infective agents. Bioorg Med Chem Lett (2005) 0.75
Synthesis of 2,4,6-trisubstituted pyrimidine and triazine heterocycles as antileishmanial agents. Bioorg Med Chem (2006) 0.75
Base mediated 7-exo-dig intramolecular cyclization of Ugi-propargyl precursors: a highly efficient and regioselective synthetic approach toward diverse 1,4-benzoxazepine-5(2H)-ones. Org Biomol Chem (2014) 0.75
2,4,6-Trisubstituted pyrimidine derivatives as pregnancy interceptive agents. Bioorg Med Chem (2005) 0.75
Synthesis of 2-(pyrimidin-2-yl)-1-phenyl-2,3,4,9-tetrahydro-1H-beta-carbolines as antileishmanial agents. Eur J Med Chem (2010) 0.75
Synthesis and biological evaluation of indolyl glyoxylamides as a new class of antileishmanial agents. Bioorg Med Chem Lett (2010) 0.75