Published in Org Lett on August 14, 2012
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Targeting the prostaglandin F2α receptor for preventing preterm labor with azapeptide tocolytics. J Med Chem (2011) 0.77
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Conformationally constrained dipeptide surrogates with aromatic side-chains: synthesis of 4-aryl indolizidin-9-one amino acids by conjugate addition to a common alpha,omega-diaminoazelate enone intermediate. J Org Chem (2004) 0.75
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Synthesis of protected 2-pyrrolylalanine for peptide chemistry and examination of its influence on prolyl amide isomer equilibrium. J Org Chem (2012) 0.75
Investigation of the active turn geometry for the labour delaying activity of indolizidinone and azapeptide modulators of the prostaglandin F2α receptor. Org Biomol Chem (2015) 0.75
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Solid-phase synthesis of 1,3,5-trisubstituted 1,4-diazepin-2-one peptide mimic. Adv Exp Med Biol (2009) 0.75
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Synthesis of fused heteroarylprolines and pyrrolopyrroles. J Org Chem (2004) 0.75
Multicomponent diversity-oriented synthesis of aza-lysine-peptide mimics. Org Lett (2013) 0.75
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Diversity-oriented synthesis of azapeptides with basic amino acid residues: aza-lysine, aza-ornithine, and aza-arginine. Org Lett (2014) 0.75
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Influences of Histidine-1 and Azaphenylalanine-4 on the Affinity, Anti-inflammatory and Antiangiogenic Activities of Azapeptide Cluster of Differentiation 36 Receptor Modulators. J Med Chem (2017) 0.75
Structure-activity study of the ORL1 antagonist Ac-Arg-D-Cha-Qaa-D-Arg-D-p-ClPhe-NH2. J Med Chem (2004) 0.75
Insertion of multiple alpha-amino gamma-lactam (Agl) residues into a peptide sequence by solid-phase synthesis on synphase lanterns. Biopolymers (2010) 0.75
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Synthesis and alkylation of aza-glycinyl dipeptide building blocks. J Pept Sci (2013) 0.75
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Design, synthesis and biological assessment of biased allosteric modulation of the urotensin II receptor using achiral 1,3,4-benzotriazepin-2-one turn mimics. J Med Chem (2017) 0.75