Rank | Title | Journal | Year | PubWeight™‹?› |
---|---|---|---|---|
1 | Discovery of a selective M₄ positive allosteric modulator based on the 3-amino-thieno[2,3-b]pyridine-2-carboxamide scaffold: development of ML253, a potent and brain penetrant compound that is active in a preclinical model of schizophrenia. | Bioorg Med Chem Lett | 2012 | 0.95 |