Exploiting drug-resistant enzymes as tools to identify thienopyrimidinone inhibitors of human immunodeficiency virus reverse transcriptase-associated ribonuclease H.

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Published in J Med Chem on June 20, 2013

Authors

Takashi Masaoka1, Suhman Chung, Pierluigi Caboni, Jason W Rausch, Jennifer A Wilson, Humeyra Taskent-Sezgin, John A Beutler, Graziella Tocco, Stuart F J Le Grice

Author Affiliations

1: RT Biochemistry Section, HIV Drug Resistance Program, National Cancer Institute , Frederick, Maryland 21702, United States.

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