Published in Adv Synth Catal on November 01, 2011
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Direct catalytic asymmetric synthesis of pyrazolidine derivatives. ChemistryOpen (2012) 0.75
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Novel immunosuppressive agents. Potent immunological activity of some bensothiopyrano [4,3-c]pyrazol-3-ones. J Med Chem (1981) 1.47
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Kinesin spindle protein (KSP) inhibitors. Part 1: The discovery of 3,5-diaryl-4,5-dihydropyrazoles as potent and selective inhibitors of the mitotic kinesin KSP. Bioorg Med Chem Lett (2005) 1.19
Highly enantioselective michael addition of cyclic 1,3-dicarbonyl compounds to alpha,beta-unsaturated ketones. Org Lett (2007) 1.10
An entry to a chiral dihydropyrazole scaffold: enantioselective [3 + 2] cycloaddition of nitrile imines. J Am Chem Soc (2005) 1.09
Catalytic asymmetric hydroperoxidation of alpha,beta-unsaturated ketones: an approach to enantiopure peroxyhemiketals, epoxides, and aldols. Angew Chem Int Ed Engl (2008) 1.08
Enantioselective synthesis of beta-(3-hydroxypyrazol-1-yl) ketones using an organocatalyzed Michael addition reaction. Org Lett (2009) 1.06
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Readily accessible 9-epi-amino cinchona alkaloid derivatives promote efficient, highly enantioselective additions of aldehydes and ketones to nitroolefins. Org Lett (2007) 1.04
Enantioselective Diels-Alder reaction of simple alpha,beta-unsaturated ketones with a cinchona alkaloid catalyst. J Am Chem Soc (2008) 1.03
Diaryl dihydropyrazole-3-carboxamides with significant in vivo antiobesity activity related to CB1 receptor antagonism: synthesis, biological evaluation, and molecular modeling in the homology model. J Med Chem (2007) 0.98
Enantioselective 1,3-dipolar cycloaddition reaction between diazoacetates and alpha-substituted acroleins: total synthesis of manzacidin A. J Am Chem Soc (2006) 0.98
A convenient synthesis of substituted pyrazolidines and azaproline derivatives through highly regio- and diastereoselective reduction of 2-pyrazolines. J Org Chem (2007) 0.97
Organocatalytic asymmetric Friedel-Crafts alkylation of indoles with simple alpha,beta-unsaturated ketones. Org Lett (2007) 0.96
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Organocatalytic and highly enantioselective direct alpha-amination of aromatic ketones. Org Lett (2007) 0.93
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Enantioselective 1,3-dipolar cycloadditions of diazoacetates with electron-deficient olefins. Org Lett (2007) 0.89
Organocatalytic asymmetric aziridination of enones. Angew Chem Int Ed Engl (2008) 0.88
Organocatalytic enantioselective indole alkylations of alpha,beta-unsaturated ketones. Org Biomol Chem (2007) 0.87
Kinesin spindle protein (KSP) inhibitors. Part 4: Structure-based design of 5-alkylamino-3,5-diaryl-4,5-dihydropyrazoles as potent, water-soluble inhibitors of the mitotic kinesin KSP. Bioorg Med Chem Lett (2006) 0.87
Synthesis, biological properties, and molecular modeling investigations of novel 3,4-diarylpyrazolines as potent and selective CB(1) cannabinoid receptor antagonists. J Med Chem (2004) 0.86
Asymmetric aza-Michael reactions catalyzed by cinchona alkaloids. J Org Chem (2007) 0.85
Asymmetric aza-Michael reactions of alpha,beta-unsaturated ketones with bifunctional organic catalysts. Angew Chem Int Ed Engl (2008) 0.85
Novel 3,4-diarylpyrazolines as potent cannabinoid CB1 receptor antagonists with lower lipophilicity. Bioorg Med Chem Lett (2005) 0.84
A catalytic asymmetric 6 pi electrocyclization: enantioselective synthesis of 2-pyrazolines. Angew Chem Int Ed Engl (2009) 0.82
Synthesis and antidepressant profiles of phenyl-substituted 2-amino- and 2-[(alkoxycarbonyl)amino]-1,4,5,6-tetrahydropyrimidines. J Med Chem (1985) 0.79
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Catalytic enantioselective 1,3-dipolar cycloadditions of alkyl diazoacetates with alpha,beta-disubstituted acroleins. Chem Commun (Camb) (2009) 0.78
Enantioselective phase-transfer catalysis: synthesis of pyrazolines. Angew Chem Int Ed Engl (2010) 0.78
Structural biochemistry. 8. 9-Amino-(9-deoxy)-cinchona alkaloids. J Chem Soc Perkin 1 (1968) 0.77
Kinesin spindle protein (KSP) inhibitors. Part 6: Design and synthesis of 3,5-diaryl-4,5-dihydropyrazole amides as potent inhibitors of the mitotic kinesin KSP. Bioorg Med Chem Lett (2007) 0.76
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TAB2 and TAB3 activate the NF-kappaB pathway through binding to polyubiquitin chains. Mol Cell (2004) 6.00
The TRAF6 ubiquitin ligase and TAK1 kinase mediate IKK activation by BCL10 and MALT1 in T lymphocytes. Mol Cell (2004) 5.08
Prediction of genetic values of quantitative traits in plant breeding using pedigree and molecular markers. Genetics (2010) 4.95
A putative ABC transporter confers durable resistance to multiple fungal pathogens in wheat. Science (2009) 3.85
Differential expression in SAGE: accounting for normal between-library variation. Bioinformatics (2003) 3.06
Association analysis of historical bread wheat germplasm using additive genetic covariance of relatives and population structure. Genetics (2007) 2.39
Act1, a U-box E3 ubiquitin ligase for IL-17 signaling. Sci Signal (2009) 2.05
Overdispersed logistic regression for SAGE: modelling multiple groups and covariates. BMC Bioinformatics (2004) 2.01
A simple and efficient method for concentration of ocean viruses by chemical flocculation. Environ Microbiol Rep (2011) 1.64
An approach to skeletal diversity using functional group pairing of multifunctional scaffolds. Org Lett (2007) 1.56
Towards quantitative metagenomics of wild viruses and other ultra-low concentration DNA samples: a rigorous assessment and optimization of the linker amplification method. Environ Microbiol (2012) 1.52
Association mapping and gene-gene interaction for stem rust resistance in CIMMYT spring wheat germplasm. Theor Appl Genet (2011) 1.39
Highly enantioselective conjugate addition of malonate and beta-ketoester to nitroalkenes: asymmetric C-C bond formation with new bifunctional organic catalysts based on cinchona alkaloids. J Am Chem Soc (2004) 1.39
Stereocontrolled creation of adjacent quaternary and tertiary stereocenters by a catalytic conjugate addition. Angew Chem Int Ed Engl (2004) 1.39
Human DNA ligases I and III, but not ligase IV, are required for microhomology-mediated end joining of DNA double-strand breaks. Nucleic Acids Res (2008) 1.37
Evaluation of methods to concentrate and purify ocean virus communities through comparative, replicated metagenomics. Environ Microbiol (2012) 1.36
Biodiesel production with immobilized lipase: A review. Biotechnol Adv (2010) 1.28
Catalytic enantioselective peroxidation of alpha,beta-unsaturated ketones. J Am Chem Soc (2008) 1.26
Mouse embryonic stem cells, but not somatic cells, predominantly use homologous recombination to repair double-strand DNA breaks. Stem Cells Dev (2010) 1.23
Dual-function cinchona alkaloid catalysis: catalytic asymmetric tandem conjugate addition-protonation for the direct creation of nonadjacent stereocenters. J Am Chem Soc (2006) 1.19
Construction of quaternary stereocenters by efficient and practical conjugate additions to alpha,beta-unsaturated ketones with a chiral organic catalyst. Angew Chem Int Ed Engl (2006) 1.19
Control of diastereoselectivity in tandem asymmetric reactions generating nonadjacent stereocenters with bifunctional catalysis by cinchona alkaloids. J Am Chem Soc (2007) 1.15
Homologous recombination conserves DNA sequence integrity throughout the cell cycle in embryonic stem cells. Stem Cells Dev (2010) 1.15
Gene-specific markers for the wheat gene Lr34/Yr18/Pm38 which confers resistance to multiple fungal pathogens. Theor Appl Genet (2009) 1.15
Modulation of DNA end joining by nuclear proteins. J Biol Chem (2005) 1.14
Enantioselective nitroaldol reaction of alpha-ketoesters catalyzed by cinchona alkaloids. J Am Chem Soc (2006) 1.14
Rice APOPTOSIS INHIBITOR5 coupled with two DEAD-box adenosine 5'-triphosphate-dependent RNA helicases regulates tapetum degeneration. Plant Cell (2011) 1.14
Asymmetric organic catalysis with modified cinchona alkaloids. Acc Chem Res (2004) 1.12
Isolation of mesenchymal stem cells from human placental decidua basalis and resistance to hypoxia and serum deprivation. Stem Cell Rev (2009) 1.11
Vps9p CUE domain ubiquitin binding is required for efficient endocytic protein traffic. J Biol Chem (2003) 1.11
Pellino 3b negatively regulates interleukin-1-induced TAK1-dependent NF kappaB activation. J Biol Chem (2008) 1.10
New slow-rusting leaf rust and stripe rust resistance genes Lr67 and Yr46 in wheat are pleiotropic or closely linked. Theor Appl Genet (2010) 1.09
A rat model for stable chronic obstructive pulmonary disease induced by cigarette smoke inhalation and repetitive bacterial infection. Biol Pharm Bull (2012) 1.07
Repair of infarcted myocardium using mesenchymal stem cell seeded small intestinal submucosa in rabbits. Biomaterials (2009) 1.06
Asymmetric alcoholysis of cyclic anhydrides. Chem Rev (2003) 1.06
From mice to humans: identification of commonly deregulated genes in mammary cancer via comparative SAGE studies. Cancer Res (2004) 1.06
Pneumococcal serotype distribution and antimicrobial resistance in Chinese children hospitalized for pneumonia. Vaccine (2011) 1.06
Asymmetric synthesis of chiral aldehydes by conjugate additions with bifunctional organocatalysis by cinchona alkaloids. Angew Chem Int Ed Engl (2006) 1.06
Hepatoblast-like progenitor cells derived from embryonic stem cells can repopulate livers of mice. Gastroenterology (2010) 1.06
A consensus map for Ug99 stem rust resistance loci in wheat. Theor Appl Genet (2014) 1.05
Porcine urinary bladder matrix-polypropylene mesh: a novel scaffold material reduces immunorejection in rat pelvic surgery. Int Urogynecol J (2012) 1.05
Enantioselective Diels-Alder reaction of simple alpha,beta-unsaturated ketones with a cinchona alkaloid catalyst. J Am Chem Soc (2008) 1.03
The novel mouse Polo-like kinase 5 responds to DNA damage and localizes in the nucleolus. Nucleic Acids Res (2010) 1.02
Dynamic kinetic resolution via dual-function catalysis of modified cinchona alkaloids: asymmetric synthesis of alpha-hydroxy carboxylic acids. J Am Chem Soc (2002) 1.02
Lr68: a new gene conferring slow rusting resistance to leaf rust in wheat. Theor Appl Genet (2012) 1.02
Presence of qnr gene in Escherichia coli and Klebsiella pneumoniae resistant to ciprofloxacin isolated from pediatric patients in China. BMC Infect Dis (2008) 1.02
Catalytic asymmetric conjugate addition of simple alkyl thiols to alpha,beta-unsaturated N-acylated oxazolidin-2-ones with bifunctional catalysts. J Am Chem Soc (2009) 1.01
The Mannich reaction of malonates with simple imines catalyzed by bifunctional cinchona alkaloids: enantioselective synthesis of beta-amino acids. J Am Chem Soc (2006) 1.01
Leaf rust (Puccinia triticina) resistance in wheat (Triticum aestivum) cultivars grown in Northern Europe 1992-2002. Hereditas (2006) 1.00
Molecular characteristics of community-acquired, methicillin-resistant Staphylococcus aureus isolated from Chinese children. FEMS Immunol Med Microbiol (2010) 0.99
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Long-term effects of Tiaobu Feishen therapies on systemic and local inflammation responses in rats with stable chronic obstructive pulmonary disease. Zhong Xi Yi Jie He Xue Bao (2012) 0.98
Asymmetric Friedel-crafts reaction of indoles with imines by an organic catalyst. J Am Chem Soc (2006) 0.97
Lr67/Yr46 confers adult plant resistance to stem rust and powdery mildew in wheat. Theor Appl Genet (2014) 0.96
miR-124 inhibits growth and invasion of gastric cancer by targeting ROCK1. Asian Pac J Cancer Prev (2014) 0.96
Mlh1 mediates tissue-specific regulation of mitotic recombination. Oncogene (2004) 0.96
Antibiotic use in five children's hospitals during 2002-2006: the impact of antibiotic guidelines issued by the Chinese Ministry of Health. Pharmacoepidemiol Drug Saf (2008) 0.96
Catalytic asymmetric cyanosilylation of ketones with chiral Lewis base. J Am Chem Soc (2003) 0.96
Community-acquired, methicillin-resistant Staphylococcus aureus isolated from children with community-onset pneumonia in China. Pediatr Pulmonol (2010) 0.95
Kinetic study of thermal inactivation of potato peroxidase during high-temperature short-time processing. J Food Sci Technol (2010) 0.95
Occurrence of qnr-positive clinical isolates in Klebsiella pneumoniae producing ESBL or AmpC-type beta-lactamase from five pediatric hospitals in China. FEMS Microbiol Lett (2008) 0.95
Asymmetric Diels-Alder reactions of 2-pyrones with a bifunctional organic catalyst. J Am Chem Soc (2007) 0.94
The breast cancer susceptibility allele CHEK2*1100delC promotes genomic instability in a knock-in mouse model. Mutat Res (2006) 0.94
Using Galleria mellonella-Candida albicans infection model to evaluate antifungal agents. Biol Pharm Bull (2013) 0.94
EGFR-specific PEGylated immunoliposomes for active siRNA delivery in hepatocellular carcinoma. Biomaterials (2011) 0.93
Morphological behavior of osteoblast-like cells on surface-modified titanium in vitro. Biomaterials (2002) 0.92
Catalytic enantioselective C-C bond forming conjugate additions with vinyl sulfones. J Am Chem Soc (2005) 0.92
Asymmetric synthesis of trifluoromethylated amines via catalytic enantioselective isomerization of imines. J Am Chem Soc (2012) 0.92
Highly Enantioselective Asymmetric Darzens Reactions with a Phase Transfer Catalyst. Chem Sci (2011) 0.92
Diagnostic and co-dominant PCR markers for wheat stem rust resistance genes Sr25 and Sr26. Theor Appl Genet (2009) 0.91
Hypoxia inhibits the spontaneous calcification of bone marrow-derived mesenchymal stem cells. J Cell Biochem (2012) 0.90
Multidrug-resistant clones of community-associated meticillin-resistant Staphylococcus aureus isolated from Chinese children and the resistance genes to clindamycin and mupirocin. J Med Microbiol (2012) 0.90
Highly enantioselective amination of alpha-substituted alpha-cyanoacetates with chiral catalysts accessible from both quinine and quinidine. Org Lett (2005) 0.89
Development of a rapid, room-temperature dynamic kinetic resolution for efficient asymmetric synthesis of alpha-aryl amino acids. Org Lett (2002) 0.89
[Serotype distribution and resistance to beta-lactams of Streptococcus pneumoniae isolated from children in Beijing, Shanghai and Guangzhou, 2000 - 2002]. Zhonghua Er Ke Za Zhi (2006) 0.89
Pseudogene PTENP1 Suppresses Gastric Cancer Progression by Modulating PTEN. Anticancer Agents Med Chem (2016) 0.89
Spatial variation and contamination assessment of heavy metals in sediments in the Manwan Reservoir, Lancang River. Ecotoxicol Environ Saf (2012) 0.88
Luteolin protects dopaminergic neurons from inflammation-induced injury through inhibition of microglial activation. Neurosci Lett (2008) 0.88
The promotion of siRNA delivery to breast cancer overexpressing epidermal growth factor receptor through anti-EGFR antibody conjugation by immunoliposomes. Biomaterials (2011) 0.88
Asymmetric Mannich reactions with in situ generation of carbamate-protected imines by an organic catalyst. Org Lett (2007) 0.88
Angiogenic and osteogenic potential of platelet-rich plasma and adipose-derived stem cell laden alginate microspheres. Biomaterials (2012) 0.87
Spatio-temporal variation of heavy metals in fresh water after dam construction: a case study of the Manwan Reservoir, Lancang River. Environ Monit Assess (2011) 0.87
Effect of tiotropium bromide on expression of CD(8) (+)CD (25) (+)FoxP (3) (+) regulatory T cells in patients with stable chronic obstructive pulmonary disease. J Huazhong Univ Sci Technolog Med Sci (2011) 0.86
Molecular and clinical characteristics of clonal complex 59 methicillin-resistant Staphylococcus aureus infections in Mainland China. PLoS One (2013) 0.86
Asymmetric olefin isomerization of butenolides via proton transfer catalysis by an organic molecule. J Am Chem Soc (2011) 0.86
The performance of a bone-derived scaffold material in the repair of critical bone defects in a rhesus monkey model. Biomaterials (2007) 0.85
Asymmetric aza-Michael reactions of alpha,beta-unsaturated ketones with bifunctional organic catalysts. Angew Chem Int Ed Engl (2008) 0.85
Elucidation of the active conformation of cinchona alkaloid catalyst and chemical mechanism of alcoholysis of meso anhydrides. Proc Natl Acad Sci U S A (2010) 0.85
QTL mapping of slow-rusting, adult plant resistance to race Ug99 of stem rust fungus in PBW343/Muu RIL population. Theor Appl Genet (2013) 0.85
Structural study-guided development of versatile phase-transfer catalysts for asymmetric conjugate additions of cyanide. Angew Chem Int Ed Engl (2011) 0.85
Tensor deep stacking networks. IEEE Trans Pattern Anal Mach Intell (2013) 0.85
Radiation-induced genetic instability in vivo depends on p53 status. Mutat Res (2002) 0.85
Enantioselective Friedel-Crafts reaction of indoles with carbonyl compounds catalyzed by bifunctional cinchona alkaloids. Org Lett (2006) 0.85
Mesenchymal stem cells transplantation mildly ameliorates experimental diabetic nephropathy in rats. Chin Med J (Engl) (2009) 0.85
Fabrication and detection of tissue-engineered bones with bio-derived scaffolds in a rotating bioreactor. Biotechnol Appl Biochem (2006) 0.84