|
1
|
4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity.
|
J Med Chem
|
2014
|
0.82
|
|
2
|
Lead optimization of 1,4-azaindoles as antimycobacterial agents.
|
J Med Chem
|
2014
|
0.82
|
|
3
|
Thiazolopyridine ureas as novel antitubercular agents acting through inhibition of DNA Gyrase B.
|
J Med Chem
|
2013
|
0.78
|
|
4
|
Discovery of efficacious Pseudomonas aeruginosa-targeted siderophore-conjugated monocarbams by application of a semi-mechanistic pharmacokinetic/pharmacodynamic model.
|
J Med Chem
|
2015
|
0.75
|