Rank | Title | Journal | Year | PubWeight™‹?› |
---|---|---|---|---|
1 | In vitro and in vivo efficacy of β-lactams against replicating and slowly growing/nonreplicating Mycobacterium tuberculosis. | Antimicrob Agents Chemother | 2013 | 1.10 |
2 | Azaindoles: noncovalent DprE1 inhibitors from scaffold morphing efforts, kill Mycobacterium tuberculosis and are efficacious in vivo. | J Med Chem | 2013 | 0.97 |
3 | Optimization of pyrrolamides as mycobacterial GyrB ATPase inhibitors: structure-activity relationship and in vivo efficacy in a mouse model of tuberculosis. | Antimicrob Agents Chemother | 2013 | 0.87 |
4 | 4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity. | J Med Chem | 2014 | 0.82 |