| Rank | Title | Journal | Year | PubWeight™‹?› |
|---|---|---|---|---|
| 1 | Azaindoles: noncovalent DprE1 inhibitors from scaffold morphing efforts, kill Mycobacterium tuberculosis and are efficacious in vivo. | J Med Chem | 2013 | 0.97 |
| 2 | 4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity. | J Med Chem | 2014 | 0.82 |
| 3 | Lead optimization of 1,4-azaindoles as antimycobacterial agents. | J Med Chem | 2014 | 0.82 |
| 4 | A high-throughput absorbance-based assay for methionine produced by methionine aminopeptidase using S-adenosyl-L-methionine synthetase. | J Biomol Screen | 2011 | 0.78 |
| 5 | Diarylthiazole: an antimycobacterial scaffold potentially targeting PrrB-PrrA two-component system. | J Med Chem | 2014 | 0.77 |
| 6 | A homogeneous, high-throughput-compatible, fluorescence intensity-based assay for UDP-N-acetylenolpyruvylglucosamine reductase (MurB) with nanomolar product detection. | J Biomol Screen | 2011 | 0.76 |