PubRank

Pravin S Iyer

Author PubWeight™ 10.77‹?›

Top papers

Rank Title Journal Year PubWeight™‹?›
1 Discovery of novel PI3-kinase δ specific inhibitors for the treatment of rheumatoid arthritis: taming CYP3A4 time-dependent inhibition. J Med Chem 2012 1.03
2 Azaindoles: noncovalent DprE1 inhibitors from scaffold morphing efforts, kill Mycobacterium tuberculosis and are efficacious in vivo. J Med Chem 2013 0.97
3 Solution-phase synthesis of a tricyclic pyrrole-2-carboxamide discovery library applying a stetter-Paal-Knorr reaction sequence. J Comb Chem 2006 0.87
4 Aminoazabenzimidazoles, a novel class of orally active antimalarial agents. J Med Chem 2014 0.83
5 Lead optimization of 1,4-azaindoles as antimycobacterial agents. J Med Chem 2014 0.82
6 4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity. J Med Chem 2014 0.82
7 N-aryl-2-aminobenzimidazoles: novel, efficacious, antimalarial lead compounds. J Med Chem 2014 0.82
8 Microwave-assisted "libraries from libraries" approach toward the synthesis of allyl- and C-cyclopropylalkylamides. J Comb Chem 2005 0.81
9 Design, synthesis, and biological evaluation of new monoamine reuptake inhibitors with potential therapeutic utility in depression and pain. Bioorg Med Chem Lett 2010 0.79
10 2-Substituted N-aryl piperazines as novel triple reuptake inhibitors for the treatment of depression. Bioorg Med Chem Lett 2010 0.77
11 Synthesis of privileged scaffolds by using diversity-oriented synthesis. Chem Asian J 2013 0.77
12 Reagent-based DOS: developing a diastereoselective methodology to access spirocyclic- and fused heterocyclic ring systems. Chem Asian J 2012 0.77
13 Novel 3,3-disubstituted pyrrolidines as selective triple serotonin/norepinephrine/dopamine reuptake inhibitors. Bioorg Med Chem Lett 2008 0.76
14 Novel, achiral aminoheterocycles as selective monoamine reuptake inhibitors. Bioorg Med Chem Lett 2009 0.75