Published in Org Biomol Chem on October 21, 2014
Role of the clathrin terminal domain in regulating coated pit dynamics revealed by small molecule inhibition. Cell (2011) 2.56
Clathrin-independent carriers form a high capacity endocytic sorting system at the leading edge of migrating cells. J Cell Biol (2010) 1.84
Modified norcantharidins; synthesis, protein phosphatases 1 and 2A inhibition, and anticancer activity. Bioorg Med Chem Lett (2004) 1.67
Norcantharimides, synthesis and anticancer activity: Synthesis of new norcantharidin analogues and their anticancer evaluation. Bioorg Med Chem (2007) 1.63
Ozone-induced dissociation: elucidation of double bond position within mass-selected lipid ions. Anal Chem (2007) 1.43
Myristyl trimethyl ammonium bromide and octadecyl trimethyl ammonium bromide are surface-active small molecule dynamin inhibitors that block endocytosis mediated by dynamin I or dynamin II. Mol Pharmacol (2007) 1.33
Inhibition of dynamin mediated endocytosis by the dynoles--synthesis and functional activity of a family of indoles. J Med Chem (2009) 1.30
Dynamin inhibition blocks botulinum neurotoxin type A endocytosis in neurons and delays botulism. J Biol Chem (2011) 1.27
Protein phosphatase inhibition: structure based design. Towards new therapeutic agents. Curr Pharm Des (2004) 1.12
Anti-malarial, anti-algal, anti-tubercular, anti-bacterial, anti-photosynthetic, and anti-fouling activity of diterpene and diterpene isonitriles from the tropical marine sponge Cymbastela hooperi. Org Biomol Chem (2010) 1.12
Elucidation of double bond position in unsaturated lipids by ozone electrospray ionization mass spectrometry. Anal Chem (2007) 1.12
Norcantharidin analogues: synthesis, anticancer activity and protein phosphatase 1 and 2A inhibition. ChemMedChem (2008) 1.08
Heterocyclic substituted cantharidin and norcantharidin analogues--synthesis, protein phosphatase (1 and 2A) inhibition, and anti-cancer activity. Bioorg Med Chem Lett (2007) 1.06
The dynamin inhibitors MiTMAB and OcTMAB induce cytokinesis failure and inhibit cell proliferation in human cancer cells. Mol Cancer Ther (2010) 1.01
A novel class of anticancer compounds targets the actin cytoskeleton in tumor cells. Cancer Res (2013) 0.99
Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activity. Bioorg Med Chem Lett (2004) 0.95
Analysis of synaptic vesicle endocytosis in synaptosomes by high-content screening. Nat Protoc (2012) 0.94
Calcineurin activity is required for the completion of cytokinesis. Cell Mol Life Sci (2010) 0.94
Targeting membrane trafficking in infection prophylaxis: dynamin inhibitors. Trends Cell Biol (2012) 0.94
An FTIR spectroscopic study on the effect of molecular structural variations on the CO2 absorption characteristics of heterocyclic amines. Chemphyschem (2011) 0.93
Inhibition of dynamin by dynole 34-2 induces cell death following cytokinesis failure in cancer cells. Mol Cancer Ther (2011) 0.93
Small molecule inhibitors of dynamin I GTPase activity: development of dimeric tyrphostins. J Med Chem (2005) 0.91
New impurity profiles of recent Australian imported 'ice': methamphetamine impurity profiling and the identification of (pseudo)ephedrine and Leuckart specific marker compounds. Forensic Sci Int (2006) 0.90
Norcantharidin analogues with nematocidal activity in Haemonchus contortus. Bioorg Med Chem Lett (2011) 0.87
The pthaladyns: GTP competitive inhibitors of dynamin I and II GTPase derived from virtual screening. J Med Chem (2010) 0.87
Serine/threonine phosphatases in socioeconomically important parasitic nematodes--prospects as novel drug targets? Biotechnol Adv (2010) 0.86
Anticancer activity and protein phosphatase 1 and 2A inhibition of a new generation of cantharidin analogues. Invest New Drugs (2002) 0.86
Iminochromene inhibitors of dynamins I and II GTPase activity and endocytosis. J Med Chem (2010) 0.86
Actin- and dynamin-dependent maturation of bulk endocytosis restores neurotransmission following synaptic depletion. PLoS One (2012) 0.86
Synthesis and evaluation of novel ellipticines as potential anti-cancer agents. Org Biomol Chem (2013) 0.84
The role of the HPA axis in psychiatric disorders and CRF antagonists as potential treatments. Arch Pharm (Weinheim) (2006) 0.84
Clathrin terminal domain-ligand interactions regulate sorting of mannose 6-phosphate receptors mediated by AP-1 and GGA adaptors. J Biol Chem (2014) 0.84
Dynamin regulates specific membrane fusion events necessary for acrosomal exocytosis in mouse spermatozoa. J Biol Chem (2012) 0.83
Synthesis and anticancer activity of a series of norcantharidin analogues. Eur J Med Chem (2012) 0.82
Azido and diazarinyl analogues of bis-tyrphostin as asymmetrical inhibitors of dynamin GTPase. ChemMedChem (2009) 0.82
Inhibition of clathrin by pitstop 2 activates the spindle assembly checkpoint and induces cell death in dividing HeLa cancer cells. Mol Cancer (2013) 0.82
Synthesis and biological activity of Delta-5,6-norcantharimides: importance of the 5,6-bridge. Eur J Med Chem (2010) 0.81
Synthesis and biological evaluation of norcantharidin analogues: towards PP1 selectivity. Bioorg Med Chem (2007) 0.81
Molecular dynamics approaches to the design and synthesis of PCB targeting molecularly imprinted polymers: interference to monomer-template interactions in imprinting of 1,2,3-trichlorobenzene. Org Biomol Chem (2013) 0.81
Australian Federal Police seizures of illicit crystalline methamphetamine ('ice') 1998-2002: impurity analysis. Forensic Sci Int (2006) 0.80
Cytotoxic 2-phenyacrylnitriles, the importance of the cyanide moiety and discovery of potent broad spectrum cytotoxic agents. Eur J Med Chem (2012) 0.80
The expanding utility of continuous flow hydrogenation. Org Biomol Chem (2015) 0.79
Development of 1,8-naphthalimides as clathrin inhibitors. J Med Chem (2013) 0.79
Direct observation of the gas phase reaction of the cyclohexyl radical with dioxygen using a distonic radical ion approach. J Phys Chem A (2010) 0.79
Steroids from an Australian sponge Psammoclema sp. J Nat Prod (2009) 0.78
Development of second-generation indole-based dynamin GTPase inhibitors. J Med Chem (2012) 0.78
Investigation of the one-pot synthesis of quinolin-2-(1H)-ones and the discovery of a variation of the three-component Ugi reaction. Org Biomol Chem (2011) 0.78
A 'cold synthesis' of heroin and implications in heroin signature analysis utility of trifluoroacetic/acetic anhydride in the acetylation of morphine. Forensic Sci Int (2006) 0.77
The antiplasmodial activity of norcantharidin analogs. Bioorg Med Chem Lett (2010) 0.77
Pyrimidyn compounds: dual-action small molecule pyrimidine-based dynamin inhibitors. ACS Chem Biol (2013) 0.77
Anti-inflammatory activity of cinnamon (C. zeylanicum and C. cassia) extracts - identification of E-cinnamaldehyde and o-methoxy cinnamaldehyde as the most potent bioactive compounds. Food Funct (2015) 0.77
Ionic liquids as porogens for molecularly imprinted polymers: propranolol, a model study. Org Biomol Chem (2014) 0.76
Does the metal influence non-covalent binding of complexes to DNA? Dalton Trans (2008) 0.76
An ATR-FTIR study on the effect of molecular structural variations on the CO2 absorption characteristics of heterocyclic amines, part II. Chemphyschem (2012) 0.75
1,8-Naphthalimide derivatives: new leads against dynamin I GTPase activity. Org Biomol Chem (2015) 0.75
Isolation and identification of unique marker compounds from the Tasmanian poppy Papaver somniferum N. Implications for the identification of illicit heroin of Tasmanian origin. Forensic Sci Int (2007) 0.75
An optimized method to quantify dopamine turnover in the mammalian retina. Anal Chem (2017) 0.75
Efficient preparation and improved sensitivity of molecularly imprinted polymers using room temperature ionic liquids. Chem Commun (Camb) (2006) 0.75
The use of effective fragment potentials in the design and synthesis of molecularly imprinted polymers for the group recognition of PCBs. Org Biomol Chem (2013) 0.75
An extreme vertices mixture design approach to the optimisation of 1,2,3-trichlorobenzene specific molecularly imprinted polymers. Org Biomol Chem (2013) 0.75
The discovery of allyltyrosine based tripeptides as selective inhibitors of the HIV-1 integrase strand-transfer reaction. Org Biomol Chem (2016) 0.75
Molecularly imprinted films of acrylonitrile/methyl methacrylate/acrylic acid terpolymers: influence of methyl methacrylate in the binding performance of L-ephedrine imprinted films. Org Biomol Chem (2013) 0.75
A tribute to a living legend. Med Chem (2012) 0.75
Self-assembly of a unique 3d/4f heterometallic square prismatic box-like coordination cage. Dalton Trans (2016) 0.75
Molecular and Silica-Supported Molybdenum Alkyne Metathesis Catalysts: Influence of Electronics and Dynamics on Activity Revealed by Kinetics, Solid-State NMR and Chemical Shift Analysis. J Am Chem Soc (2017) 0.75
Evaluation of 4-substituted styrenes as functional monomers for the synthesis of theophylline-specific molecularly imprinted polymers. Org Biomol Chem (2014) 0.75
Isolation and characterization of charge-tagged phenylperoxyl radicals in the gas phase: direct evidence for products and pathways in low temperature benzene oxidation. Phys Chem Chem Phys (2012) 0.75
Focused library development of 2-phenylacrylamides as broad spectrum cytotoxic agents. Bioorg Med Chem (2012) 0.75
Norcantharimide analogues possessing terminal phosphate esters and their anti-cancer activity. Bioorg Med Chem (2011) 0.75
Serine/threonine protein phosphatase inhibition enhances the effect of thymidylate synthase inhibition. Cancer Chemother Pharmacol (2003) 0.75
Quinolone-1-(2H)-ones as hedgehog signalling pathway inhibitors. Org Biomol Chem (2016) 0.75