Dihydropyrrolo[2,3-d]pyrimidines: Selective Toll-Like Receptor 9 Antagonists from Scaffold Morphing Efforts.

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🔗 View Article (PMC 4233361)

Published in ACS Med Chem Lett on October 02, 2014

Authors

Manabu Watanabe1, Mai Kasai1, Hideyuki Tomizawa1, Masamitsu Aoki1, Kazuo Eiho1, Yoshiaki Isobe1, Shigehiro Asano2

Author Affiliations

1: Sumitomo Dainippon Pharma Co., Ltd. , 3-1-98 Kasugade Naka, Konohana-ku, Osaka 554-0022, Japan.
2: Sumitomo Dainippon Pharma Co., Ltd. , 33-94 Enoki-cho, Suita, Osaka 564-0053, Japan.

Associated clinical trials:

First Safety Study in Humans of a Single Dose of CPG 52364 | NCT00547014

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