Theranostic pretargeted radioimmunotherapy of colorectal cancer xenografts in mice using picomolar affinity (86)Y- or (177)Lu-DOTA-Bn binding scFv C825/GPA33 IgG bispecific immunoconjugates.

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🔗 View Article (PMID 26596724)

Published in Eur J Nucl Med Mol Imaging on November 24, 2015

Authors

Sarah M Cheal1,2, Hong Xu3, Hong-Fen Guo3, Sang-Gyu Lee1,2, Blesida Punzalan1,2, Sandhya Chalasani1, Edward K Fung2,4, Achim Jungbluth5, Pat B Zanzonico4, Jorge A Carrasquillo1, Joseph O'Donoghue4, Peter M Smith-Jones6,7, K Dane Wittrup8,9,10, Nai-Kong V Cheung2,3, Steven M Larson11,12

Author Affiliations

1: Department of Radiology, Memorial Sloan Kettering Cancer Center, New York, NY, USA.
2: Molecular Pharmacology and Chemistry Program, Memorial Sloan Kettering Cancer Center, 415 E. 68th Street, Z-2064, New York, NY, 10065, USA.
3: Department of Pediatrics, Memorial Sloan Kettering Cancer Center, New York, NY, USA.
4: Department of Medical Physics, Memorial Sloan Kettering Cancer Center, New York, NY, USA.
5: Department of Pathology, Memorial Sloan Kettering Cancer Center, New York, NY, USA.
6: Department of Psychiatry and Behavioral Science, Stony Brook University, Stony Brook, NY, USA.
7: Department of Radiology, Stony Brook University, Stony Brook, NY, USA.
8: Department of Chemical Engineering, Massachusetts Institute of Technology, Cambridge, MA, USA.
9: Department of Biological Engineering, Massachusetts Institute of Technology, Cambridge, MA, USA.
10: Koch Institute for Integrative Cancer Research, Massachusetts Institute of Technology, Cambridge, MA, USA.
11: Department of Radiology, Memorial Sloan Kettering Cancer Center, New York, NY, USA. larsons@mskcc.org.
12: Molecular Pharmacology and Chemistry Program, Memorial Sloan Kettering Cancer Center, 415 E. 68th Street, Z-2064, New York, NY, 10065, USA. larsons@mskcc.org.

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