Re-assessing gallium-67 as a therapeutic radionuclide.

PubWeight™: 0.75‹?›

🔗 View Article (PMID 27915165)

Published in Nucl Med Biol on October 29, 2016

Authors

Muhamad F Bin Othman1, Nabil R Mitry1, Valerie J Lewington2, Philip J Blower1, Samantha Y A Terry3

Author Affiliations

1: King's College London, Department of Imaging Chemistry and Biology, St. Thomas' Hospital, London, SE1 7EH, UK.
2: Guy's & St Thomas' NHS Foundation Trust, Nuclear Medicine Department, London, SE1 9RT, UK.
3: King's College London, Department of Imaging Chemistry and Biology, St. Thomas' Hospital, London, SE1 7EH, UK. Electronic address: samantha.terry@kcl.ac.uk.

Articles cited by this

Radiation spectra for Auger-electron emitting radionuclides: report No. 2 of AAPM Nuclear Medicine Task Group No. 6. Med Phys (1993) 1.63

NODAGATOC, a new chelator-coupled somatostatin analogue labeled with [67/68Ga] and [111In] for SPECT, PET, and targeted therapeutic applications of somatostatin receptor (hsst2) expressing tumors. Bioconjug Chem (2002) 1.12

Indium-111-labeled cellular blood components: mechanism of labeling and intracellular location in human neutrophils. J Nucl Med (1977) 1.10

Comparative gallium-68 labeling of TRAP-, NOTA-, and DOTA-peptides: practical consequences for the future of gallium-68-PET. EJNMMI Res (2012) 1.05

Auger radiation targeted into DNA: a therapy perspective. Eur J Nucl Med Mol Imaging (2006) 1.04

[(68)Ga]FSC-(RGD)3 a trimeric RGD peptide for imaging αvβ3 integrin expression based on a novel siderophore derived chelating scaffold-synthesis and evaluation. Nucl Med Biol (2014) 0.99

Auger electron-induced double-strand breaks depend on DNA topology. Radiat Res (2008) 0.98

111In-labeled EGF is selectively radiotoxic to human breast cancer cells overexpressing EGFR. J Nucl Med (2000) 0.98

Procedure guideline for gallium scintigraphy in the evaluation of malignant disease. Society of Nuclear Medicine. J Nucl Med (1997) 0.96

Efficient bifunctional gallium-68 chelators for positron emission tomography: tris(hydroxypyridinone) ligands. Chem Commun (Camb) (2011) 0.93

Evaluation of bifunctional chelates for the development of gallium-based radiopharmaceuticals. Bioconjug Chem (2010) 0.91

Design and preclinical evaluation of a 99mTc-labelled diabody of mAb J591 for SPECT imaging of prostate-specific membrane antigen (PSMA). EJNMMI Res (2014) 0.91

Radionuclides linked to a CD74 antibody as therapeutic agents for B-cell lymphoma: comparison of Auger electron emitters with beta-particle emitters. J Nucl Med (2000) 0.90

RGD conjugates of the H2dedpa scaffold: synthesis, labeling and imaging with 68Ga. Nucl Med Biol (2012) 0.89

The molecular structure of indium-DTPA. J Nucl Med (1989) 0.89

The mechanism of 67Ga localization in malignant disease. Nucl Med Biol (1996) 0.88

Benefits of NOPO as chelator in gallium-68 peptides, exemplified by preclinical characterization of (68)Ga-NOPO-c(RGDfK). Mol Pharm (2014) 0.88

Uptake of gallium-67 in transfected cells and tumors absent or enriched in the transferrin receptor. J Nucl Med (1998) 0.87

Gallium-67 radiotoxicity in human U937 lymphoma cells. Br J Cancer (1993) 0.86

99mTc-labeled HYNIC-DAPI causes plasmid DNA damage with high efficiency. PLoS One (2014) 0.85

Comparison of two new angiogenesis PET tracers 68Ga-NODAGA-E[c(RGDyK)]2 and (64)Cu-NODAGA-E[c(RGDyK)]2; in vivo imaging studies in human xenograft tumors. Nucl Med Biol (2013) 0.84

A comparison of 4 radionuclides conjugated to antibodies for single-cell kill. J Nucl Med (2003) 0.83

Amplification of DNA damage by a γH2AX-targeted radiopharmaceutical. Nucl Med Biol (2012) 0.83

Radiotoxicity of 67-gallium on myeloid leukemic blasts. Leuk Res (1995) 0.83

Relationship between chromatin structure and sensitivity to molecularly targeted auger electron radiation therapy. Int J Radiat Oncol Biol Phys (2012) 0.82

Therapy of disseminated B-cell lymphoma xenografts in severe combined immunodeficient mice with an anti-CD74 antibody conjugated with (111)indium, (67)gallium, or (90)yttrium. Clin Cancer Res (2001) 0.82

Structure and stability of hexadentate complexes of ligands based on AAZTA for efficient PET labelling with gallium-68. Chem Commun (Camb) (2012) 0.82

H2CHXdedpa and H4CHXoctapa-chiral acyclic chelating ligands for (67/68)Ga and (111)In radiopharmaceuticals. Inorg Chem (2015) 0.81

New Tris(hydroxypyridinone) Bifunctional Chelators Containing Isothiocyanate Groups Provide a Versatile Platform for Rapid One-Step Labeling and PET Imaging with (68)Ga(3.). Bioconjug Chem (2015) 0.81

[The relationship between Ga-67 uptake and transferrin receptors in cultured cells]. Kanagawa Shigaku (1990) 0.80

High-dose gallium-67 therapy in patients with relapsed acute leukaemia: a feasibility study. Br J Cancer (1995) 0.80

The use of SEP-PAK SI cartridges for the preparation of gallium chloride from the citrate solution. Eur J Nucl Med (1993) 0.79

Gallium-68 lipophilic complexes for labeling platelets. J Nucl Med (1985) 0.78

111In-BnDTPA-F3: an Auger electron-emitting radiotherapeutic agent that targets nucleolin. EJNMMI Res (2012) 0.78

The effect of dimethyl sulfoxide on the induction of DNA strand breaks in plasmid DNA and colony formation of PC Cl3 mammalian cells by alpha-, beta-, and Auger electron emitters (223)Ra, (188)Re, and (99m)Tc. EJNMMI Res (2016) 0.77

Transferrin dependence of Ga (NO3)3 inhibition of growth in human-derived small cell lung cancer cells. J Cell Biochem Suppl (1996) 0.77

Gallium-67-labelled red blood cells as a blood-pool marker for dual-isotope imaging. Int J Rad Appl Instrum B (1992) 0.77

Frozen section microautoradiography in the study of radionuclide targeting: application to indium-111-oxine-labeled leukocytes. J Nucl Med (1995) 0.76