Structure-activity relationships of progesterone derivatives that bind to the digitalis receptor: modifications in A and B rings.

PubWeight™: 0.75‹?›

🔗 View Article (PMID 3455050)

Published in Steroids on September 30, 1988

Authors

J F Templeton1, V P Kumar, R S Kim, F S LaBella

Author Affiliations

1: Faculty of Pharmacy, University of Manitoba, Winnipeg, Canada.

Articles by these authors

Enhanced cancer growth in mice administered daily human-equivalent doses of some H1-antihistamines: predictive in vitro correlates. J Natl Cancer Inst (1994) 3.79

The Temple-Wisconsin Cognitive Vulnerability to Depression Project: lifetime history of axis I psychopathology in individuals at high and low cognitive risk for depression. J Abnorm Psychol (2000) 2.64

Isolation of nerve endings from the posterior pituitary gland. Electron microscopy of fractions obtained by centrifugation. J Cell Biol (1965) 1.87

Comparison of analytical methods for monitoring autoxidation profiles of authentic lipids. J Lipid Res (1987) 1.50

The long head of the triceps brachii as a free functioning muscle transfer. Plast Reconstr Surg (2001) 1.49

Stimulation of malignant growth in rodents by antidepressant drugs at clinically relevant doses. Cancer Res (1992) 1.48

The unrecognized giants. Plast Reconstr Surg (1996) 1.41

The first description of the free vascularized bone transplant. Plast Reconstr Surg (1997) 1.38

On the specificity of naloxone as an opiate antagonist. Life Sci (1979) 1.33

Drainage versus nondrainage in simultaneous bilateral total knee arthroplasties. Clin Orthop Relat Res (1998) 1.32

Histamine as an intracellular messenger. Biochem Pharmacol (1990) 1.13

Drainage versus nondrainage in simultaneous bilateral total hip arthroplasties. J Arthroplasty (1998) 1.13

Resection of vascular malformations. J Hand Surg Br (1993) 1.10

Distribution of primary motor nerve branches and terminal nerve entry points to the forearm muscles. Anat Rec (1997) 1.07

Histamine is an intracellular messenger mediating platelet aggregation. Science (1989) 1.04

Surgical management of non-union of neglected fractures of the patella. Injury (1991) 1.02

Elbow dislocation with ipsilateral radial shaft fracture. An unusual outcome. Clin Orthop Relat Res (1996) 1.01

Snapping hip--an unusual cause. J Bone Joint Surg Br (1990) 1.00

Enhanced autoxidation of dopamine as a possible basis of manganese neurotoxicity. Neurotoxicology (1981) 0.99

The course of the inferior gluteal nerve in the posterior approach to the hip. J Bone Joint Surg Br (2006) 0.98

Progesterone derivative binds to cardiac ouabain receptor and shows dissociation between sodium pump inhibition and increased contractile force. Nature (1979) 0.98

High risk HPV types in southern Iranian patients with cervical cancer. Pathol Oncol Res (2003) 0.97

Autonomous proliferation of colon cancer cells that coexpress transforming growth factor alpha and its receptor. Variable effects of receptor-blocking antibody. Gastroenterology (1992) 0.96

On the involvement of GABA in the analgesia produced by baclofen, muscimol and morphine. Neuropharmacology (1982) 0.95

Free vascularised epiphyseal transplantation in upper extremity reconstruction. J Hand Surg Br (1988) 0.95

Modified Sihler's technique for studying the distribution of intramuscular nerve branches in mammalian skeletal muscle. Anat Rec (1997) 0.94

Increased apoptosis, changes in intracellular Ca2+, and functional alterations in lymphocytes and macrophages after in vitro exposure to static magnetic field. J Toxicol Environ Health A (1998) 0.93

Amino acid composition of human aortic elastin as influenced by age. J Gerontol (1966) 0.91

Anterior cruciate ligament injuries. To counsel or to operate? J Bone Joint Surg Br (1986) 0.89

Stress fractures of the tibia in osteoarthritis of the knee. J Bone Joint Surg Br (1987) 0.89

Characterization and localization of adenosine receptors in rat spinal cord. J Neurosci (1984) 0.89

Histamine and growth: interaction of antiestrogen binding site ligands with a novel histamine site that may be associated with calcium channels. Cancer Res (1987) 0.88

Histamine and calcium are independently regulated intracellular mediators of lymphocyte mitogenesis. Biochem Biophys Res Commun (1992) 0.87

Contractile characteristics on electrical stimulation of muscle with multiple motor points. An in vivo study in rabbits. Clin Orthop Relat Res (1995) 0.87

Pregnanes that bind to the digitalis receptor: synthesis of 14-hydroxy-5 beta,14 beta-pregnane glycosides from digitoxin and digitoxigenin. J Med Chem (1991) 0.87

Transforming growth factor-beta inhibits apoptosis induced by beta-amyloid peptide fragment 25-35 in cultured neuronal cells. Brain Res Mol Brain Res (1998) 0.86

Opiate-like naloxone-reversible actions of somatostatin given intracerebrally. Can J Physiol Pharmacol (1978) 0.86

Myofascial compartments of the hand in relation to compartment syndrome: a cadaveric study. Plast Reconstr Surg (2009) 0.86

Peptidase inhibitors reduce opiate narcotic withdrawal signs, including seizure activity, in the rat. Brain Res (1982) 0.85

Classic bioassay statistical procedures applied to radioimmunoassay of bovine thyrotropin, growth hormone and prolactin. J Clin Endocrinol Metab (1971) 0.84

The antiproliferative potency of histamine antagonists correlates with inhibition of binding of [3H]-histamine to novel intracellular receptors (HIC) in microsomal and nuclear fractions of rat liver. Agents Actions Suppl (1991) 0.84

Ulnar fractures with bisphosphonate therapy: a systematic review of published case reports. Osteoporos Int (2014) 0.83

The natural history of spontaneous osteonecrosis of the medial tibial plateau. J Bone Joint Surg Br (2003) 0.83

Amino acid composition of neurohypophysial secretory granules and Van Dyke protein. Biochem Pharmacol (1967) 0.83

Transforming growth factor-beta protects human hNT cells from degeneration induced by beta-amyloid peptide: involvement of the TGF-beta type II receptor. Brain Res Mol Brain Res (1997) 0.83

Cloning of the triosephosphate isomerase gene of Plasmodium falciparum and expression in Escherichia coli. Mol Biochem Parasitol (1993) 0.83

The myofascial compartments of the foot: a cadaver study. J Bone Joint Surg Br (2008) 0.82

Dermatitis complicating operatively induced anesthetic regions around the knee. A report of four cases. J Bone Joint Surg Am (1993) 0.82

ACTH receptors in nervous tissue. High affinity binding-sequestration of [125I]Phe2,Nle4]ACTH 1-24 in homogenates and slices from rat brain. Can J Physiol Pharmacol (1989) 0.82

Adrenocorticotropin(1-10) and -(11-24) promote adrenal steroidogenesis by different mechanisms. Endocrinology (1989) 0.81

Ontogenesis of adenosine receptors in the central nervous system of the rat. Brain Res (1984) 0.81

Opiate receptor binding activity of 17-alpha estrogenic steroids. Life Sci (1978) 0.81

Is there a general anesthesia receptor. Can J Physiol Pharmacol (1981) 0.81

The relationship between elastin and an acidic protein in mammalian uterus. Connect Tissue Res (1973) 0.81

Progesterone derivatives that bind to the digitalis receptor: synthesis of 14 beta-hydroxyprogesterone. A novel steroid with positive inotropic activity. J Med Chem (1987) 0.81

Characterization of nitrobenzylthioinosine binding to nucleoside transport sites selective for adenosine in rat brain. J Neurosci (1985) 0.81

Osteoarticular allografts for reconstruction in the proximal part of the humerus after excision of a musculoskeletal tumor. J Bone Joint Surg Am (1992) 0.81

Storage and secretion of neurohypophyseal hormones. Can J Physiol Pharmacol (1968) 0.81

Neuroanatomical basis for the tarsal tunnel syndrome. Foot Ankle Int (2012) 0.81

Infection of vascularized fibular grafts. Clin Orthop Relat Res (1996) 0.80

Postprandial 2-hr C-peptide concentration as a guide for insulin treatment in patient with NIDDM. Korean J Intern Med (1986) 0.80

Extremity osteosarcoma--a Southeast Asian experience. Ann Acad Med Singapore (2002) 0.80

Oxidation of 14-C-1 and 14-C-6-glucose by hormone synthesizing and hormone secreting portions of neurohypophysial neurons. Mol Pharmacol (1965) 0.80

Inhibition of nitric oxide synthase by straight chain and cyclic alcohols. Eur J Pharmacol (1997) 0.80

The role of atmospheric pressure in stabilising the shoulder. An experimental study. J Bone Joint Surg Br (1985) 0.79

Osteochondritis dissecans following Perthes' disease. Arthroscopic-operative treatment. Clin Orthop Relat Res (1986) 0.79

Progesterone derivatives that bind to the digitalis receptor: effects on 86Rb uptake and contractility in the isolated guinea pig heart. Can J Physiol Pharmacol (1984) 0.79

Progesterone derivatives that bind to the digitalis receptor: effects on Na+,K+-ATPase and isolated tissues. Fed Proc (1985) 0.79

Ouabain receptor binding of hydroxyprogesterone derivatives. Br J Pharmacol (1979) 0.79

Tenodesis of the long head of the biceps brachii for chronic bicipital tendinitis. Long-term results. J Bone Joint Surg Am (1990) 0.79

Ultrastructural localization of acid phosphatase in the posterior pituitary of the dehydrated rat. Z Zellforsch Mikrosk Anat (1972) 0.79

Correlation of the antiproliferative action of diphenylmethane-derivative antiestrogen binding site ligands with antagonism of histamine binding but not of protein kinase C-mediated phosphorylation. Cancer Res (1988) 0.79

The neuromuscular compartments of the flexor carpi ulnaris. Plast Reconstr Surg (1999) 0.79

Increased therapeutic index of antineoplastic drugs in combination with intracellular histamine antagonists. J Natl Cancer Inst (1991) 0.79

Intracellular histamine and liver regeneration: high affinity binding of histamine to chromatin, low affinity binding to matrix, and depletion of a nuclear storage pool following partial hepatectomy. Biochem Biophys Res Commun (1992) 0.79

Intraventricular Met5-enkephalin causes unexpected lowering of pain threshold and narcotic withdrawal signs in rats. Nature (1976) 0.79

The effect of linoleic and arachidonic acid derivatives on calcium transport in vesicles from cardiac sarcoplasmic reticulum. J Mol Cell Cardiol (1988) 0.79

Chlormadinone acetate, a progesterone derivative that binds to the digitalis receptor, inhibits the sodium pump in the isolated rat diaphragm. Can J Physiol Pharmacol (1985) 0.79

Digitaloid pregnanes promote potassium-sparing diuresis in the guinea pig. Can J Physiol Pharmacol (1992) 0.78

Split flexor carpi radialis muscle. Plast Reconstr Surg (1999) 0.78

Chlorotyrosine exerts renal effects and antagonizes renal and gastric responses to atrial natriuretic peptide. J Pharmacol Exp Ther (1994) 0.78

Estimation of cholinesterase and choline acetyltransferase in bovine anterior pituitary, posterior pituitary, and pineal body. J Neurochem (1968) 0.78

Opiate-like excitatory effects of steroid sulfates and calcium-complexing agents given cerebroventricularly. Brain Res (1979) 0.78

Independent function in a tendon transfer of the split flexor carpi ulnaris. Plast Reconstr Surg (1999) 0.78

Arterial mesenchyme and arteriosclerosis. Enzymic vs non-enzymic factors in the deterioration of connective tissue. Adv Exp Med Biol (1974) 0.78

Effect of synthetic TRF on hormone release from bovine anterior pituitary in vitro. Endocrinology (1971) 0.78

Opiate properties of SKF 525A. Can J Physiol Pharmacol (1978) 0.78

Agonist-induced regulation of adrenoceptor subtypes in cerebral cortical slices. J Neurochem (1987) 0.78

Long head of the triceps transfer for elbow flexion. Plast Reconstr Surg (2007) 0.77

Electrocardiographic changes in catastrophic abdominal illness mimicking acute myocardial infarction. Am J Cardiol (1987) 0.77

Digitalis-like pregnanes. Cardiac and renal effects of a glycoside of 14 beta-hydroxyprogesterone. Can J Physiol Pharmacol (1988) 0.77

Calcium translocation by fatty acid derivatives in a two-phase partition model. Structure-activity relationships. Biochim Biophys Acta (1985) 0.77