PubRank

Dalibor Sames

Author PubWeight™ 61.47‹?›

Top papers

Rank Title Journal Year PubWeight™‹?›
1 C-H bond functionalization in complex organic synthesis. Science 2006 3.76
2 Direct palladium-catalyzed C-2 and C-3 arylation of indoles: a mechanistic rationale for regioselectivity. J Am Chem Soc 2005 1.82
3 sp3 C-H bond arylation directed by amidine protecting group: alpha-arylation of pyrrolidines and piperidines. J Am Chem Soc 2006 1.40
4 Fluorescent false neurotransmitters visualize dopamine release from individual presynaptic terminals. Science 2009 1.39
5 Fully synthetic carbohydrate-based vaccines in biochemically relapsed prostate cancer: clinical trial results with alpha-N-acetylgalactosamine-O-serine/threonine conjugate vaccine. J Clin Oncol 2003 1.37
6 C-C bond formation via C-H bond activation: synthesis of the core of teleocidin B4. J Am Chem Soc 2002 1.35
7 Direct C-arylation of free (NH)-indoles and pyrroles catalyzed by Ar-Rh(III) complexes assembled in situ. J Am Chem Soc 2005 1.32
8 Room temperature hydroalkylation of electron-deficient olefins: sp3 C-H functionalization via a lewis acid-catalyzed intramolecular redox event. J Am Chem Soc 2005 1.31
9 Pt(IV)-catalyzed cyclization of arene-alkyne substrates via intramolecular electrophilic hydroarylation. Org Lett 2003 1.29
10 Catalytic C-H arylation of SEM-protected azoles with palladium complexes of NHCs and phosphines. Org Lett 2006 1.25
11 Reactivity of functional groups on the protein surface: development of epoxide probes for protein labeling. J Am Chem Soc 2003 1.25
12 Fluorescent dopamine tracer resolves individual dopaminergic synapses and their activity in the brain. Proc Natl Acad Sci U S A 2012 1.20
13 Retracted C-C bond formation via C-H bond activation: catalytic arylation and alkenylation of alkane segments. J Am Chem Soc 2002 1.18
14 C-H bond functionalization via hydride transfer: Lewis acid catalyzed alkylation reactions by direct intramolecular coupling of sp3 C-H bonds and reactive alkenyl oxocarbenium intermediates. J Am Chem Soc 2009 1.14
15 Room temperature intramolecular hydro-O-alkylation of aldehydes: sp3 C-H functionalization via a Lewis acid catalyzed tandem 1,5-hydride transfer/cyclization. Org Lett 2005 1.13
16 Principles of mucin architecture: structural studies on synthetic glycopeptides bearing clustered mono-, di-, tri-, and hexasaccharide glycodomains. J Am Chem Soc 2002 1.13
17 Cross-coupling of sp(3) C-H bonds and alkenes: catalytic cyclization of alkene-amide substrates. J Am Chem Soc 2004 1.09
18 Total synthesis of (-)-rhazinilam: asymmetric C[bond]H bond activation via the use of a chiral auxiliary. J Am Chem Soc 2002 1.05
19 Ru(III)-catalyzed cyclization of arene-alkene substrates via intramolecular electrophilic hydroarylation. Org Lett 2004 1.04
20 Retracted Oxidative C-arylation of free (NH)-heterocycles via direct (sp3) C-H bond functionalization. J Am Chem Soc 2004 1.03
21 Direct C-H bond arylation: selective palladium-catalyzed C2-arylation of N-substituted indoles. Org Lett 2004 1.00
22 Retracted Selective and catalytic arylation of N-phenylpyrrolidine: sp3 C-H bond functionalization in the absence of a directing group. J Am Chem Soc 2005 0.99
23 Phosphine-free palladium-catalyzed C-H bond arylation of free (N-H)-indoles and pyrroles. J Org Chem 2007 0.99
24 Selective and catalytic arylation of N-phenylpyrrolidine: (sp3) C-H bond functionalization in the absence of a directing group [J. Am. Chem. Soc. 2005, 127, 5284-5285]. J Am Chem Soc 2006 0.97
25 C-H bond functionalization via hydride transfer: synthesis of dihydrobenzopyrans from ortho-vinylaryl akyl ethers. Org Lett 2009 0.97
26 Oxidative C-arylation of free (NH)-heterocycles via direct sp3 C-H bond functionalization [J. Am. Chem. Soc. 2004, 126, 13244-13246]. J Am Chem Soc 2006 0.96
27 Development of pH-responsive fluorescent false neurotransmitters. J Am Chem Soc 2010 0.94
28 Imaging induction of cytoprotective enzymes in intact human cells: coumberone, a metabolic reporter for human AKR1C enzymes reveals activation by panaxytriol, an active component of red ginseng. J Am Chem Soc 2008 0.93
29 Retracted Diversity synthesis via C-H bond functionalization: concept-guided development of new C-arylation methods for imidazoles. J Am Chem Soc 2003 0.93
30 A luminescent sensor for tyrosine phosphorylation. Org Lett 2007 0.90
31 C-H arylation of pyridines: high regioselectivity as a consequence of the electronic character of C-H bonds and heteroarene ring. J Am Chem Soc 2011 0.90
32 Design of optical switches as metabolic indicators: new fluorogenic probes for monoamine oxidases (MAO A and B). J Am Chem Soc 2005 0.90
33 Retracted Selective C-arylation of free (NH)-heteroarenes via catalytic C-H bond functionalization. J Am Chem Soc 2003 0.89
34 C-H bond functionalization via hydride transfer: direct coupling of unactivated alkynes and sp(3) C-H bonds catalyzed by platinum tetraiodide. J Am Chem Soc 2009 0.88
35 Complementation of biotransformations with chemical C-H oxidation: copper-catalyzed oxidation of tertiary amines in complex pharmaceuticals. J Am Chem Soc 2013 0.88
36 Cocktails of Tb(3+) and Eu(3+) complexes: a general platform for the design of ratiometric optical probes. J Am Chem Soc 2007 0.87
37 Ruthenium catalyzed decarbonylative arylation at sp3 carbon centers in pyrrolidine and piperidine heterocycles. J Am Chem Soc 2007 0.87
38 C-H bonds as ubiquitous functionality: a general approach to complex arylated pyrazoles via sequential regioselective C-arylation and N-alkylation enabled by SEM-group transposition. J Am Chem Soc 2009 0.87
39 New tools for molecular imaging of redox metabolism: development of a fluorogenic probe for 3 alpha-hydroxysteroid dehydrogenases. J Am Chem Soc 2004 0.86
40 Harnessing functional plasticity of enzymes: a fluorogenic probe for imaging 17beta-HSD10 dehydrogenase, an enzyme involved in Alzheimer's and Parkinson's diseases. J Am Chem Soc 2007 0.85
41 A new fluorogenic transformation: development of an optical probe for coenzyme Q. Org Lett 2005 0.84
42 Concise synthesis of the chemopreventitive agent (+/-)-deguelin via a key 6-endo hydroarylation. Org Lett 2003 0.84
43 Transposing molecular fluorescent switches into the near-IR: development of luminogenic reporter substrates for redox metabolism. J Am Chem Soc 2007 0.84
44 New fluorescent substrate enables quantitative and high-throughput examination of vesicular monoamine transporter 2 (VMAT2). ACS Chem Biol 2013 0.84
45 Synthetic and Receptor Signaling Explorations of the Mitragyna Alkaloids: Mitragynine as an Atypical Molecular Framework for Opioid Receptor Modulators. J Am Chem Soc 2016 0.84
46 C-H bonds as ubiquitous functionality: a general approach to complex arylated imidazoles via regioselective sequential arylation of all three C-H bonds and regioselective N-alkylation enabled by SEM-group transposition. J Org Chem 2010 0.83
47 APP+, a fluorescent analogue of the neurotoxin MPP+, is a marker of catecholamine neurons in brain tissue, but not a fluorescent false neurotransmitter. ACS Chem Neurosci 2013 0.83
48 NeuO: a fluorescent chemical probe for live neuron labeling. Angew Chem Int Ed Engl 2015 0.82
49 Fluorogenic metabolic probes for direct activity readout of redox enzymes: Selective measurement of human AKR1C2 in living cells. Proc Natl Acad Sci U S A 2006 0.81
50 Catalytic coupling of arene C-H bonds and alkynes for the synthesis of coumarins: substrate scope and application to the development of neuroimaging agents. J Org Chem 2012 0.79
51 Phosphorylation state-responsive lanthanide peptide conjugates: a luminescence switch based on reversible complex reorganization. Org Lett 2006 0.79
52 C-H bond functionalization via hydride transfer: formation of α-arylated piperidines and 1,2,3,4-tetrahydroisoquinolines via stereoselective intramolecular amination of benzylic C-H bonds. J Org Chem 2012 0.78
53 Fluoromorphic substrates for fatty acid metabolism: highly sensitive probes for mammalian medium-chain acyl-CoA dehydrogenase. Angew Chem Int Ed Engl 2006 0.78
54 (-)-CHANA, a fluorogenic probe for detecting amyloid binding alcohol dehydrogenase HSD10 activity in living cells. ACS Chem Biol 2010 0.78
55 Site-specific phenylation of pyridine catalyzed by phosphido-bridged ruthenium dimer complexes: a prototype for C-H arylation of electron-deficient heteroarenes. J Am Chem Soc 2005 0.77
56 Paradoxical abatement of striatal dopaminergic transmission by cocaine and methylphenidate. J Biol Chem 2013 0.77
57 Two-photon induced uncaging of a reactive intermediate. Multiphoton in situ detection of a potentially valuable label for biological applications. J Org Chem 2005 0.76
58 Expanding the use of fluorogenic enzyme reporter substrates to imaging metabolic flux changes: the activity measurement of 5α-steroid reductase in intact mammalian cells. ACS Chem Biol 2010 0.76
59 C-H bonds as ubiquitous functionality: preparation of multiple regioisomers of arylated 1,2,4-triazoles via C-H arylation. J Org Chem 2012 0.75
60 Dopamine release at individual presynaptic terminals visualized with FFNs. J Vis Exp 2009 0.75
61 Constructing Iboga alkaloids via C-H bond functionalization: examination of the direct and catalytic union of heteroarenes and isoquinuclidine alkenes. J Org Chem 2015 0.75
62 Cobalt-catalyzed arylation of azole heteroarenes via direct C-H bond functionalization. Org Lett 2003 0.75
63 Identification of fluorescent small molecule compounds for synaptic labeling by image-based, high-content screening. ACS Chem Neurosci 2017 0.75
64 Synthesis of luminescent heterometallic bis-lanthanide complexes via selective, sequential metallation. Chem Commun (Camb) 2006 0.75
65 Intermolecular energy transfer from Tb3+ to Eu3+ in aqueous aggregates and on the surface of human cells. Org Lett 2011 0.75