Combinatorial lead optimization of [1,2]-diamines based on ethambutol as potential antituberculosis preclinical candidates.

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Published in J Comb Chem on March 10, 2003

Authors

Richard E Lee1, Marina Protopopova, Emma Crooks, Richard A Slayden, Marianne Terrot, Clifton E Barry

Author Affiliations

1: Tuberculosis Research Section, NIAID, National Institutes of Health, Rockville, Maryland 20850, USA.

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