Rank | Title | Journal | Year | PubWeight™‹?› |
---|---|---|---|---|
1 | Optimization of a tertiary alcohol series of phosphodiesterase-4 (PDE4) inhibitors: structure-activity relationship related to PDE4 inhibition and human ether-a-go-go related gene potassium channel binding affinity. | J Med Chem | 2003 | 1.03 |