PubRank

Dawei Ma

Author PubWeight™ 91.20‹?›

Top papers

Rank Title Journal Year PubWeight™‹?›
1 A selective inhibitor of eIF2alpha dephosphorylation protects cells from ER stress. Science 2005 7.98
2 Small molecule regulators of autophagy identified by an image-based high-throughput screen. Proc Natl Acad Sci U S A 2007 3.37
3 Beclin1 controls the levels of p53 by regulating the deubiquitination activity of USP10 and USP13. Cell 2011 2.58
4 Design of wide-spectrum inhibitors targeting coronavirus main proteases. PLoS Biol 2005 1.73
5 Andrographolide attenuates inflammation by inhibition of NF-kappa B activation through covalent modification of reduced cysteine 62 of p50. J Immunol 2004 1.58
6 Amino acid promoted CuI-catalyzed C-N bond formation between aryl halides and amines or N-containing heterocycles. J Org Chem 2005 1.56
7 Control of basal autophagy by calpain1 mediated cleavage of ATG5. Autophagy 2010 1.51
8 Enantioselective arylation of 2-methylacetoacetates catalyzed by CuI/trans-4-hydroxy-L-proline at low reaction temperatures. J Am Chem Soc 2006 1.16
9 Asymmetric, protecting-group-free total synthesis of (-)-englerin A. Angew Chem Int Ed Engl 2010 1.15
10 CuI/N,N-dimethylglycine-catalyzed coupling of vinyl halides with amides or carbamates. Org Lett 2004 1.10
11 Synthesis of aryl azides and vinyl azides via proline-promoted CuI-catalyzed coupling reactions. Chem Commun (Camb) 2004 1.10
12 Cyclodepsipeptide toxin promotes the degradation of Hsp90 client proteins through chaperone-mediated autophagy. J Cell Biol 2009 1.09
13 Co-recycling of MT1-MMP and MT3-MMP through the trans-Golgi network. Identification of DKV582 as a recycling signal. J Biol Chem 2003 1.06
14 Total synthesis and absolute stereochemical assignment of (-)-communesin F. J Am Chem Soc 2010 1.03
15 Total synthesis of cyclic tetrapeptide FR235222, a potent immunosuppressant that inhibits mammalian histone deacetylases. Org Lett 2005 1.02
16 Total synthesis of the monoterpenoid indole alkaloid (±)-aspidophylline A. Angew Chem Int Ed Engl 2014 1.01
17 A novel small molecule regulator of guanine nucleotide exchange activity of the ADP-ribosylation factor and golgi membrane trafficking. J Biol Chem 2008 1.00
18 Total synthesis of Akuammiline alkaloid (-)-vincorine via intramolecular oxidative coupling. J Am Chem Soc 2012 1.00
19 Elaboration of 2-(trifluoromethyl)indoles via a cascade coupling/condensation/deacylation process. Org Lett 2008 0.98
20 CuI/L-proline-catalyzed coupling reactions of aryl halides with activated methylene compounds. Org Lett 2005 0.97
21 Design, synthesis, and evaluation of potent, nonpeptidic mimetics of second mitochondria-derived activator of caspases. J Med Chem 2009 0.96
22 Total synthesis and structure assignment of papuamide B, a potent marine cyclodepsipeptide with anti-HIV properties. Angew Chem Int Ed Engl 2008 0.95
23 Enantioselective total syntheses of communesins A and B. Angew Chem Int Ed Engl 2011 0.94
24 Total synthesis of microsclerodermin E. Angew Chem Int Ed Engl 2003 0.94
25 Enantioselective addition of activated terminal alkynes to 1-acylpyridinium salts catalyzed by Cu-Bis(oxazoline) complexes. J Am Chem Soc 2007 0.93
26 Highly enantioselective bromocyclization of tryptamines and its application in the synthesis of (-)-chimonanthine. Angew Chem Int Ed Engl 2013 0.92
27 Assembly of isoquinolines via CuI-catalyzed coupling of beta-keto esters and 2-halobenzylamines. Org Lett 2008 0.92
28 PIM kinase inhibitors downregulate STAT3(Tyr705) phosphorylation. Mol Cancer Ther 2010 0.92
29 Total synthesis of lepadins B, d, e, and h; determination of the configuration of the latter three alkaloids. Angew Chem Int Ed Engl 2004 0.91
30 Facile entry to substituted decahydroquinoline alkaloids. Total synthesis of lepadins A-E and H. J Org Chem 2006 0.91
31 Total synthesis of salinamide A: a potent anti-inflammatory bicyclic depsipeptide. Angew Chem Int Ed Engl 2008 0.89
32 Synthesis of 3-substituted and 2,3-disubstituted quinazolinones via Cu-catalyzed aryl amidation. Org Lett 2012 0.87
33 Mild Ullmann-type biaryl ether formation reaction by combination of ortho-substituent and ligand effects. Angew Chem Int Ed Engl 2006 0.86
34 Synthesis of 1,2-disubstituted benzimidazoles by a Cu-catalyzed cascade aryl amination/condensation process. Angew Chem Int Ed Engl 2007 0.86
35 Palladium-catalyzed direct functionalization of 2-aminobutanoic acid derivatives: application of a convenient and versatile auxiliary. Angew Chem Int Ed Engl 2013 0.86
36 Synthesis of an oxazoline analogue of apratoxin A. Org Lett 2003 0.85
37 Formation of arylboronates by a CuI-catalyzed coupling reaction of pinacolborane with aryl iodides at room temperature. Org Lett 2006 0.84
38 Cyclobutane derivatives as novel nonpeptidic small molecule agonists of glucagon-like peptide-1 receptor. J Med Chem 2011 0.84
39 A one-pot coupling/hydrolysis/condensation process to pyrrolo[1,2-a]quinoxaline. J Org Chem 2008 0.84
40 Organocatalytic approach to polysubstituted piperidines and tetrahydropyrans. Org Lett 2011 0.84
41 Organocatalytic approach for the syntheses of corynantheidol, dihydrocorynantheol, protoemetinol, protoemetine, and mitragynine. Chem Asian J 2011 0.83
42 Asymmetric total syntheses of marine cyclic depsipeptide halipeptins A-D. Chemistry 2006 0.82
43 Structure-activity relationship studies of salubrinal lead to its active biotinylated derivative. Bioorg Med Chem Lett 2005 0.82
44 Assembly of substituted 1H-benzimidazoles and 1,3-dihydrobenzimidazol-2-ones via CuI/L-proline catalyzed coupling of aqueous ammonia with 2-iodoacetanilides and 2-iodophenylcarbamates. J Org Chem 2009 0.82
45 Asymmetric total synthesis of (-)-alkaloid 223A and its 6-epimer. J Org Chem 2003 0.81
46 An efficient sequential reaction process to polysubstituted indolizidines and quinolizidines and its application to the total synthesis of indolizidine 223A. Org Lett 2005 0.81
47 Synthesis of aryl sulfones via L-proline-promoted CuI-catalyzed coupling reaction of aryl halides with sulfinic acid salts. J Org Chem 2005 0.81
48 Organocatalytic Michael addition of aldehydes to protected 2-amino-1-nitroethenes: the practical syntheses of oseltamivir (Tamiflu) and substituted 3-aminopyrrolidines. Angew Chem Int Ed Engl 2010 0.80
49 CuI/DMPAO-catalyzed N-arylation of acyclic secondary amines. Org Lett 2012 0.80
50 Assembly of substituted 3-methyleneisoindolin-1-ones via a CuI/l-proline-catalyzed domino reaction process of 2-bromobenzamides and terminal alkynes. Org Lett 2009 0.80
51 Synthetic studies toward galbulimima alkaloid (-)-GB 13 and (+)-GB 16 and (-)-himgaline. Chem Asian J 2010 0.80
52 Transition-metal and organocatalysis in natural product synthesis. Beilstein J Org Chem 2013 0.79
53 A concise route to the proposed structure of lydiamycin B, an antimycobacterial depsipeptide. Org Lett 2009 0.79
54 Structural basis of RasGRP binding to high-affinity PKC ligands. J Med Chem 2002 0.79
55 A general and efficient approach to aryl thiols: CuI-catalyzed coupling of aryl iodides with sulfur and subsequent reduction. Org Lett 2009 0.79
56 Identification of a small molecule activator of novel PKCs for promoting glucose-dependent insulin secretion. Cell Res 2010 0.79
57 CuI/4-hydro-L-proline as a more effective catalytic system for coupling of aryl bromides with N-boc hydrazine and aqueous ammonia. J Org Chem 2009 0.79
58 Synthesis of symmetrical and unsymmetrical N,N'-diaryl guanidines via copper/N-methylglycine-catalyzed arylation of guanidine nitrate. J Org Chem 2012 0.79
59 Retracted The N-aryl aminocarbonyl ortho-substituent effect in Cu-catalyzed aryl amination and its application in the synthesis of 5-substituted 11-oxo-dibenzodiazepines. Org Lett 2011 0.79
60 Enantioselective synthesis of polysubstituted cyclopentanones by organocatalytic double Michael addition reactions. Org Lett 2010 0.79
61 Mild and nonracemizing conditions for Ullmann-type diaryl ether formation between aryl iodides and tyrosine derivatives. J Org Chem 2006 0.78
62 Identification, biochemical and structural evaluation of species-specific inhibitors against type I methionine aminopeptidases. J Med Chem 2013 0.78
63 Cu(I)/L-proline-catalyzed coupling of substituted 3-iodoprop-2-en-1-ols with 1-alkynes and subsequent cyclization: a convenient approach for synthesizing polysubstituted furans. Chem Asian J 2010 0.78
64 Total synthesis of clavepictines A and B and pictamine. Org Lett 2006 0.78
65 Facile access to polysubstituted indoles via a cascade Cu-catalyzed arylation-condensation process. J Org Chem 2007 0.78
66 Total synthesis of the indole alkaloid (±)- and (+)-methyl N-decarbomethoxychanofruticosinate. Angew Chem Int Ed Engl 2013 0.78
67 CuI-catalyzed domino process to 2,3-disubstituted benzofurans from 1-bromo-2-iodobenzenes and beta-keto esters. J Org Chem 2007 0.78
68 Cascade coupling/cyclization process to N-substituted 1,3-dihydrobenzimidazol-2-ones. Org Lett 2007 0.78
69 Total synthesis of piperazimycin A: a cytotoxic cyclic hexadepsipeptide. Angew Chem Int Ed Engl 2009 0.77
70 Total synthesis and cytotoxicity studies of a cyclic depsipeptide with proposed structure of palau'amide. Org Lett 2005 0.77
71 Metal-catalyzed derivatization of C(alpha)-tetrasubstituted amino acids and their use in the synthesis of cyclic peptides. Chem Asian J 2009 0.77
72 Organocatalytic Michael addition of aldehydes to gamma-keto-alpha,beta-unsaturated esters. an efficient entry to versatile chiral building blocks. Org Lett 2008 0.77
73 Studies on the structure-activity relationship of 1,3,3,4-tetra-substituted pyrrolidine embodied CCR5 receptor antagonists. Part 2: Discovery of highly potent anti-HIV agents. Bioorg Med Chem Lett 2010 0.77
74 A convergent route to the Galbulimima alkaloids (-)-GB 13 and (+)-GB 16. Angew Chem Int Ed Engl 2010 0.77
75 Assembly of N,N-disubstituted hydrazines and 1-aryl-1H-indazoles via copper-catalyzed coupling reactions. Org Lett 2012 0.77
76 Assembly of conjugated enynes and substituted indoles via CuI/amino acid-catalyzed coupling of 1-alkynes with vinyl iodides and 2-bromotrifluoroacetanilides. J Org Chem 2007 0.77
77 Enantioselective assembly of substituted dihydropyrones via organocatalytic reaction in water media. Org Lett 2008 0.77
78 Pyridinylpyrimidines selectively inhibit human methionine aminopeptidase-1. Bioorg Med Chem 2013 0.77
79 Pyridinylquinazolines selectively inhibit human methionine aminopeptidase-1 in cells. J Med Chem 2013 0.77
80 A one-pot formal [4 + 2] cycloaddition approach to substituted piperidines, indolizidines, and quinolizidines. total synthesis of indolizidine (-)-209I. J Org Chem 2005 0.77
81 A copper-catalyzed coupling reaction of vinyl halides and carbazates: application in the assembly of polysubstituted pyrroles. Chem Commun (Camb) 2014 0.76
82 Investigation on novel chitosan nanoparticle-aptamer complexes targeting TGF-β receptor II. Int J Pharm 2013 0.76
83 Highly convergent route to cyclopeptide alkaloids: total synthesis of ziziphine N. Org Lett 2007 0.76
84 Highly asymmetric bromocyclization of tryptophol: unexpected accelerating effect of DABCO-derived bromine complex. Org Lett 2014 0.76
85 Total synthesis of halipeptin A: a potent antiinflammatory cyclic depsipeptide. Angew Chem Int Ed Engl 2004 0.76
86 Development of 3-phenyl-N-(2-(3-phenylureido)ethyl)-thiophene-2-sulfonamide compounds as inhibitors of antiapoptotic Bcl-2 family proteins. ChemMedChem 2014 0.76
87 Construction of polycyclic spiro-indolines via an intramolecular oxidative coupling/cyclization cascade reaction process. Org Lett 2012 0.76
88 Studies on the structure-activity relationship of 1,3,3,4-tetra-substituted pyrrolidine embodied CCR5 receptor antagonists. Part 1: Tuning the N-substituents. Bioorg Med Chem Lett 2010 0.76
89 Total synthesis of leucosceptroids A and B. Angew Chem Int Ed Engl 2014 0.76
90 Total syntheses of (±)-spiroquinazoline, (-)-alantryphenone, (+)-lapatin A, and (-)-quinadoline B. Angew Chem Int Ed Engl 2013 0.76
91 Synthesis of 2-thio-substituted benzothiazoles via a domino condensation/S-arylation/heterocyclization process. J Org Chem 2011 0.76
92 Highly efficient catalytic system for enantioselective Michael addition of aldehydes to nitroalkenes in water. Angew Chem Int Ed Engl 2008 0.76
93 Assembly of substituted 3-aminoindazoles from 2-bromobenzonitrile via a CuBr-catalyzed coupling/condensation cascade process. J Org Chem 2013 0.75
94 Cascade annulation of malonic diamides: a concise synthesis of polycyclic pyrroloindolines. Chem Commun (Camb) 2012 0.75
95 Preparation of syn-delta-hydroxy-beta-amino esters via an intramolecular hydrogen bond directed diastereoselective hydrogenation. Total synthesis of (3S,4aS,6R,8S)-hyperaspine. Org Lett 2003 0.75
96 Recent progress on the total synthesis of natural products in China. Nat Prod Rep 2006 0.75
97 Diastereoselective aldol reaction of N,N-dibenzyl-alpha-amino aldehydes with ketones catalyzed by proline. Org Lett 2004 0.75
98 Total synthesis of antimicrobial and antitumor cyclic depsipeptides. Chem Commun (Camb) 2010 0.75
99 A formal [3+2] cycloaddition process with nonactivated aziridines to polysubstituted indolizidines. Org Lett 2005 0.75
100 N,N'-Bisoxalamides Enhance the Catalytic Activity in Cu-Catalyzed Coupling of (Hetero)Aryl Bromides with Anilines and Secondary Amines. J Org Chem 2017 0.75
101 Synthesis and antitumor activity of cyclodepsipeptide zygosporamide and its analogues. Bioorg Med Chem Lett 2008 0.75
102 Assembly of indoline-2-carboxylate-embodied dipeptides via Pd-catalyzed C(sp2)-H bond direct functionalization. Org Lett 2015 0.75
103 Synthesis and SAR study of diphenylbutylpiperidines as cell autophagy inducers. Bioorg Med Chem Lett 2010 0.75
104 Assembly of 3-acyloxindoles via cui/L-proline-catalyzed intramolecular arylation of beta-keto amides. Org Lett 2006 0.75
105 Retraction of "Total Synthesis of Kaitocephalin, the First Naturally Occurring AMPA/KA Receptor Antagonist". J Am Chem Soc 2017 0.75
106 Occurrence of matrix-bound phosphine in polar ornithogenic tundra ecosystems: effects of alkaline phosphatase activity and environmental variables. Sci Total Environ 2011 0.75
107 Potentially biomimetic total synthesis and relative stereochemical assignment of (±)-gracilamine. Angew Chem Int Ed Engl 2012 0.75
108 Organocatalytic and scalable synthesis of the anti-influenza drugs zanamivir, laninamivir, and CS-8958. Angew Chem Int Ed Engl 2014 0.75
109 1H, 13C and 15N backbone resonance assignments of matrilysin (MMP7) complexed with a sulfonamide hydroxamate-type inhibitor. J Biomol NMR 2004 0.75
110 Synthesis of 1,5-benzothiazepine dipeptide mimetics via two CuI-catalyzed cross coupling reactions. Org Lett 2009 0.75