Rank | Title | Journal | Year | PubWeight™‹?› |
---|---|---|---|---|
1 | Discovery of potent, selective, orally active, nonpeptide inhibitors of human mast cell chymase. | J Med Chem | 2007 | 0.92 |
2 | Nonpeptide inhibitors of cathepsin G: optimization of a novel beta-ketophosphonic acid lead by structure-based drug design. | J Am Chem Soc | 2002 | 0.81 |
3 | Facile dephosphonylation of beta-ketophosphonic acids: mechanistic studies. | Org Lett | 2006 | 0.80 |