Published in Science on August 23, 1985
Qinghaosu (artemisinin): an antimalarial drug from China. Science (1985) 4.95
2-Acetylpyridine thiosemicarbazones. 1. A new class of potential antimalarial agents. J Med Chem (1979) 2.86
2-Acetylpyridine thiosemicarbazones. 4. Complexes with transition metals as antimalarial and antileukemic agents. J Med Chem (1982) 1.28
Inhibition of clinically significant bacterial organisms in vitro by 2-acetylpyridine thiosemicarbazones. Antimicrob Agents Chemother (1980) 1.23
Isolation of artemisinin (qinghaosu) from Artemisia annua growing in the United States. J Nat Prod (1984) 1.17
Antimalarial activity of new water-soluble dihydroartemisinin derivatives. J Med Chem (1987) 1.17
Protoberberine alkaloids as antimalarials. J Med Chem (1988) 1.08
Berberine derivatives as antileishmanial drugs. Antimicrob Agents Chemother (1990) 1.06
2-Acetylpyridine thiosemicarbazones. 9. Derivatives of 2-acetylpyridine 1-oxide as potential antimalarial agents. J Med Chem (1984) 1.00
Antiviral activity of 2-acetylpyridine thiosemicarbazones against herpes simplex virus. Antimicrob Agents Chemother (1981) 0.97
Thiosemicarbazones of 2-acetylpyridine, 2-acetylquinoline, 1-acetylisoquinoline, and related compounds as inhibitors of herpes simplex virus in vitro and in a cutaneous herpes guinea pig model. Antiviral Res (1986) 0.96
In vitro assessment of 2-acetylpyridine thiosemicarbazones against chloroquine-resistant Plasmodium falciparum. Antimicrob Agents Chemother (1982) 0.93
2-Acetylpyridine thiosemicarbazones. 5. 1-[1-(2-Pyridyl)ethyl]-3-thiosemicarbazides as potential antimalarial agents. J Med Chem (1983) 0.90
Correlations between structure and antimycobacterial activity in a series of 2-acetylpyridine thiosemicarbazones. J Gen Microbiol (1982) 0.89
Filariasis testing in a jird model: new drug leads from some old standbys. Am J Trop Med Hyg (1994) 0.88
Antimalarial activity of new water-soluble dihydroartemisinin derivatives. 2. Stereospecificity of the ether side chain. J Med Chem (1989) 0.86
Artemisinin: an endoperoxidic antimalarial from Artemisia annua L. Fortschr Chem Org Naturst (1997) 0.84
Plasmodium berghei: the antimalarial action of artemisinin and sodium artelinate in vivo and in vitro, studied by flow cytometry. Exp Parasitol (1990) 0.84
Conversion of artemisinin (qinghaosu) to iso-artemisitene and to 9-epi-artemisinin1. Planta Med (1987) 0.83
Comparison of beta-artemether and beta-arteether against malaria parasites in vitro and in vivo. Am J Trop Med Hyg (1993) 0.82
Reductive electrochemical HPLC assay for artemisinin (qinghaosu). Planta Med (1985) 0.82
2-Acetylpyridine thiosemicarbazones. 12. Derivatives of 3-acetylisoquinoline as potential antimalarial agents. Arzneimittelforschung (1986) 0.81
Antimalarial activity of new dihydroartemisinin derivatives. 5. Sugar analogues. J Med Chem (1992) 0.80
Antimalarial activity of new water-soluble dihydroartemisinin derivatives. 3. Aromatic amine analogues. J Med Chem (1990) 0.80
2-Acetylpyridine thiosemicarbazones. 6.2-Acetylpyridine and 2-butyrylpyridine thiosemicarbazones as antileukemic agents. Arzneimittelforschung (1983) 0.80
Evaluation of the in vitro antimalarial activity of Picralima nitida extracts. J Ethnopharmacol (1992) 0.80
Artemisitene, a New Sesquiterpene Lactone Endoperoxide from Artemisia annua. Planta Med (1985) 0.80
Production of artemisinin in tissue cultures of Artemisia annua. J Nat Prod (1986) 0.79
Activity of 2-acetylpyridine thiosemicarbazones against Trypanosoma rhodesiense in vitro. Antimicrob Agents Chemother (1980) 0.79
2-Acetylpyridine thiosemicarbazones. 8. Derivatives of 1-acetylisoquinoline as potential antimalarial agents. J Med Chem (1984) 0.79
2-Acetylpyridine thiosemicarbazones. 10. 2-Propionyl-, 2-butyryl-, and 2-(2-methylpropionyl)pyridine thiosemicarbazones as potential antimalarial agents. Arzneimittelforschung (1984) 0.79
Antimalarial activity of dihydroartemisinin derivatives by transdermal application. Am J Trop Med Hyg (1994) 0.78
2-Acetylpyridine thiosemicarbazones and Mycobacterium leprae. Int J Lepr Other Mycobact Dis (1984) 0.78
Evaluation of plant extracts for antileishmanial activity using a mechanism-based radiorespirometric microtechnique (RAM). Planta Med (1992) 0.76
2-Acetylpyridine thiosemicarbazones XI: 2-(alpha-Hydroxyacetyl)pyridine thiosemicarbazones as antimalarial and antibacterial agents. J Pharm Sci (1984) 0.75
2-Amino-2-thiazoline. 3. The differing behavior of phenylisothiocyanate and phenylisocyanate toward 2-amino-2-thiazoline. Tetrahedron Lett (1967) 0.75
Activity of 2-acetylpyridine and 2-acetylquinoline thiosemicarbazones tested in vitro in combination with other antituberculous drugs. Am Rev Respir Dis (1982) 0.75
Antibacterial properties of 2-acetylpyridine-1-oxide thiosemicarbazones. Chemotherapy (1986) 0.75
Potential antiradiation agents. 3. N-substituted aminoethanethiosulfuric acids. J Med Chem (1970) 0.75
2-amino-2-oxazoline formation by cyclization of 1-(2-hydroxyethyl)-2-methyl-2-thiopseudoureas. J Pharm Sci (1970) 0.75
Thiosulfuric acid analog of quinine as a potential antimalarial agent. J Med Chem (1973) 0.75
Charge transfer and oxy radicals in antimalarial action. Quinones, dapsone metabolites, metal complexes, iminium ions, and peroxides. J Free Radic Biol Med (1985) 0.75
The oxidation of selenocystamine to 2-aminoethaneselenenic acid. J Org Chem (1966) 0.75
Potential antiradiation agents. II. Guanidinoalkanethiosulfuric acids. J Med Chem (1969) 0.75
Primaquine analogues: derivatives of 4-amino-2-methoxyacridine. J Med Chem (1979) 0.75
Stability studies of bis(pyridiniumaldoxime) reactivators of organophosphate-inhibited acetylcholinesterase. J Pharm Sci (1986) 0.75
2-amino-2-thiazoline. VI. The formation of a thiazolo-S-triazine from 2-amino-2-thiazoline. Tetrahedron (1969) 0.75
Comparison of mass spectral techniques using organic peroxides related to artemisinin. Anal Chem (1990) 0.75
Potential antiradiation agents. I. Primary aminoalkanethiosulfuric acids. J Med Chem (1969) 0.75
Thiosemicarbazones of 2-acetylpyridine, 2-acetylquinoline, 1- and 3-acetylisoquinoline and related compounds as inhibitors of clinically significant bacteria in vitro. Arzneimittelforschung (1983) 0.75
Peroxides as oxidant antimalarials. Drug Des Deliv (1989) 0.75
The structure of an N-carbamoyl derivative of 2-amino-delta-2-thiazoline. Mass spectrometry of 15N derivatives of 2-amino-delta-2-thiazoline. Acta Chem Scand (1967) 0.75
A new synthesis of selenoureas and selenothiocarbamic esters from thioureas. J Org Chem (1969) 0.75