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Felix Deanda
Author PubWeight™ 5.63
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Top papers
Rank
Title
Journal
Year
PubWeight™
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1
Dolutegravir (S/GSK1349572) exhibits significantly slower dissociation than raltegravir and elvitegravir from wild-type and integrase inhibitor-resistant HIV-1 integrase-DNA complexes.
Antimicrob Agents Chemother
2011
1.68
2
Optimization of 4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine IGF-1R tyrosine kinase inhibitors towards JNK selectivity.
Bioorg Med Chem Lett
2008
0.88
3
Discovery of 3,5-disubstituted-1H-pyrrolo[2,3-b]pyridines as potent inhibitors of the insulin-like growth factor-1 receptor (IGF-1R) tyrosine kinase.
Bioorg Med Chem Lett
2009
0.83
4
Optimization of a series of 4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidine inhibitors of IGF-1R: elimination of an acid-mediated decomposition pathway.
Bioorg Med Chem Lett
2008
0.80
5
Discovery of bioavailable 4,4-disubstituted piperidines as potent ligands of the chemokine receptor 5 and inhibitors of the human immunodeficiency virus-1.
J Med Chem
2008
0.80
6
Discovery of 4,6-bis-anilino-1H-pyrrolo[2,3-d]pyrimidines: potent inhibitors of the IGF-1R receptor tyrosine kinase.
Bioorg Med Chem Lett
2008
0.75
7
Discovery of novel pyridyl carboxamides as potent CCR5 antagonists and optimization of their pharmacokinetic profile in rats.
Bioorg Med Chem Lett
2011
0.75
8
Aza-stilbenes as potent and selective c-RAF inhibitors.
Bioorg Med Chem Lett
2006
0.75