Published in Chem Soc Rev on May 21, 2009
Organocatalytic cascade reactions as a new tool in total synthesis. Nat Chem (2010) 2.29
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Neurotrophic natural products: chemistry and biology. Angew Chem Int Ed Engl (2013) 0.96
Direct observation of an enamine intermediate in amine catalysis. J Am Chem Soc (2009) 0.94
Multicatalytic, asymmetric Michael/Stetter reaction of salicylaldehydes and activated alkynes. Proc Natl Acad Sci U S A (2010) 0.92
Methods for direct alkene diamination, new & old. Tetrahedron (2012) 0.92
Direct asymmetric vinylogous Michael addition of cyclic enones to nitroalkenes via dienamine catalysis. Proc Natl Acad Sci U S A (2010) 0.91
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Stereoselective synthesis of highly functionalized alpha-diazo-beta-ketoalkanoates via catalytic one-pot Mukaiyama-Aldol reactions. Org Lett (2010) 0.84
N-heterocyclic carbene-catalyzed rearrangements of vinyl sulfones. Chem Sci (2011) 0.83
Organocatalytic asymmetric assembly reactions for the syntheses of carbohydrate derivatives by intermolecular Michael-Henry reactions. Proc Natl Acad Sci U S A (2010) 0.83
A versatile and efficient approach for the synthesis of chiral 1,3-nitroamines and 1,3-diamines via conjugate addition to new (S,E)-γ-aminated nitroalkenes derived from L-α-amino acids. Beilstein J Org Chem (2013) 0.81
Seven Post-synthetic Covalent Reactions in Tandem Leading to Enzyme-like Complexity within Metal-Organic Framework Crystals. J Am Chem Soc (2016) 0.81
Organocatalytic Asymmetric Synthesis of Functionalized 1,3,5-Triarylpyrrolidin-2-ones via an Aza-Michael/Aldol Domino Reaction. Synthesis (Stuttg) (2014) 0.80
Organocatalytic multicomponent reaction for the acquisition of a selective inhibitor of mPTPB, a virulence factor of tuberculosis. Chem Commun (Camb) (2013) 0.80
Developing novel organocatalyzed aldol reactions for the enantioselective synthesis of biologically active molecules. Synthesis (Stuttg) (2011) 0.80
Multivalent polyglycerol supported imidazolidin-4-one organocatalysts for enantioselective Friedel-Crafts alkylations. Beilstein J Org Chem (2015) 0.80
Cross-trienamines in asymmetric organocatalysis. J Am Chem Soc (2012) 0.80
Asymmetric synthesis of highly functionalized tetrahydropyrans via a one-pot organocatalytic Michael/Henry/ketalization sequence. Org Lett (2014) 0.80
A quantitative approach to nucleophilic organocatalysis. Beilstein J Org Chem (2012) 0.79
Kinetic isotope effects in asymmetric reactions. Chemistry (2010) 0.79
An Asymmetric Organocatalytic Quadruple Cascade to Tetraaryl-Substituted 2-Azabicyclo[3.3.0]octadienones. Synthesis (Stuttg) (2014) 0.78
Highly stereoselective and scalable anti-aldol reactions using N-(p-dodecylphenylsulfonyl)-2-pyrrolidinecarboxamide: scope and origins of stereoselectivities. J Org Chem (2010) 0.78
Nonenzymatic enantioselective synthesis of all-carbon quaternary centers through desymmetrization. Tetrahedron Lett (2015) 0.78
A Simple Primary Amine Catalyst for Enantioselective α-Hydroxylations and α-Fluorinations of Branched Aldehydes. Org Lett (2015) 0.77
Diastereoselective and enantioselective conjugate addition reactions utilizing α,β-unsaturated amides and lactams. Beilstein J Org Chem (2015) 0.76
The origin of large molecules in primordial autocatalytic reaction networks. PLoS One (2012) 0.75
Enzyme catalysis: sweet flexibility. Nat Chem (2010) 0.75
Enantioselective cycloaddition of münchnones onto [60]fullerene: organocatalysis versus metal catalysis. J Am Chem Soc (2014) 0.75
Old tricks, new dogs: organocatalytic dienamine activation of α,β-unsaturated aldehydes. Chem Soc Rev (2016) 0.75
Chiral GAP catalysts of phosphonylated imidazolidinones and their applications in asymmetric Diels-Alder and Friedel-Crafts reactions. Org Biomol Chem (2017) 0.75
Synthesis of the tetracyclic core of Illicium sesquiterpenes using an organocatalyzed asymmetric Robinson annulation. Beilstein J Org Chem (2013) 0.75
Enantioselective bifunctional iminophosphorane catalyzed sulfa-Michael addition of alkyl thiols to unactivated β-substituted-α,β-unsaturated esters. Chem Sci (2016) 0.75
Synthesis of chiral sulfoximine-based thioureas and their application in asymmetric organocatalysis. Beilstein J Org Chem (2012) 0.75
Asymmetric synthesis of 1H-pyrrol-3(2H)-ones from 2,3-diketoesters by combination of aldol condensation with benzilic acid rearrangement. Chem Commun (Camb) (2015) 0.75
2,2',2''-Terpyridine-catalyzed synthesis of cyclic carbonates from epoxides and carbon dioxide under solvent-free conditions. Int J Mol Sci (2014) 0.75
N-Heterocyclic Carbene-Promoted Rauhut]Currier Reactions between Vinyl Sulfones and α,β-Unsaturated Aldehydes. Aust J Chem (2011) 0.75
Organocatalytic cascade aza-Michael/hemiacetal reaction between disubstituted hydrazines and α,β-unsaturated aldehydes: Highly diastereo- and enantioselective synthesis of pyrazolidine derivatives. Beilstein J Org Chem (2012) 0.75
From Mechanistic Study to Chiral Catalyst Optimization: Theoretical Insight into Binaphthophosphepine-catalyzed Asymmetric Intramolecular [3 + 2] Cycloaddition. Sci Rep (2017) 0.75
Asymmetric 1,3-Dipolar Cycloaddition Reactions. Chem Rev (1998) 3.73
Allylic Amination. Chem Rev (1998) 1.98
C(2)-symmetric chiral bis(oxazoline) ligands in asymmetric catalysis. Chem Rev (2006) 1.63
Enantioselective organocatalyzed alpha sulfenylation of aldehydes. Angew Chem Int Ed Engl (2005) 1.55
Catalytic asymmetric 1,3-dipolar cycloaddition reactions of azomethine ylides-a simple approach to optically active highly functionalized proline derivatives. Angew Chem Int Ed Engl (2002) 1.45
Direct organocatalytic asymmetric alpha-chlorination of aldehydes. J Am Chem Soc (2004) 1.40
On the origin of the stereoselectivity in organocatalysed reactions with trimethylsilyl-protected diarylprolinol. Chemistry (2008) 1.35
Enantioselective formation of stereogenic carbon-fluorine centers by a simple catalytic method. Angew Chem Int Ed Engl (2005) 1.32
Asymmetric organocatalytic epoxidation of alpha,beta-unsaturated aldehydes with hydrogen peroxide. J Am Chem Soc (2005) 1.23
Catalytic asymmetric Friedel-Crafts alkylation reactions--copper showed the way. Chem Rev (2008) 1.17
The diarylprolinol silyl ether system: a general organocatalyst. Acc Chem Res (2011) 1.11
Asymmetric organocatalysis with sulfones. Angew Chem Int Ed Engl (2010) 1.08
Enantioselective organocatalytic conjugate addition of N heterocycles to alpha,beta-unsaturated aldehydes. Angew Chem Int Ed Engl (2007) 1.07
Highly enantioselective direct organocatalytic alpha-chlorination of ketones. Angew Chem Int Ed Engl (2004) 1.06
Dienamine catalysis: organocatalytic asymmetric gamma-amination of alpha,beta-unsaturated aldehydes. J Am Chem Soc (2006) 1.06
A simple recipe for sophisticated cocktails: organocatalytic one-pot reactions--concept, nomenclature, and future perspectives. Angew Chem Int Ed Engl (2011) 1.04
Squaramides: bridging from molecular recognition to bifunctional organocatalysis. Chemistry (2011) 1.04
Asymmetric organocatalytic alpha-arylation of aldehydes. Angew Chem Int Ed Engl (2007) 1.01
Acyl phosphonates: good hydrogen bond acceptors and ester/amide equivalents in asymmetric organocatalysis. J Am Chem Soc (2010) 1.00
Organocatalytic direct asymmetric alpha-heteroatom functionalization of aldehydes and ketones. Chem Commun (Camb) (2006) 1.00
Organocatalytic asymmetric direct alpha-alkynylation of cyclic beta-ketoesters. J Am Chem Soc (2007) 1.00
Direct organocatalytic asymmetric alpha-sulfenylation of activated C-H bonds in lactones, lactams, and beta-dicarbonyl compounds. Chemistry (2005) 0.98
Catalytic asymmetric direct alpha-amination reactions of 2-keto esters: a simple synthetic approach to optically active syn-beta-amino-alpha-hydroxy esters. J Am Chem Soc (2002) 0.98
Highly efficient aerobic oxidative hydroxylation of arylboronic acids: photoredox catalysis using visible light. Angew Chem Int Ed Engl (2011) 0.96
Direct enantioselective Michael addition of aldehydes to vinyl ketones catalyzed by chiral amines. J Org Chem (2003) 0.96
Mechanisms in aminocatalysis. Chem Commun (Camb) (2010) 0.96
Asymmetric 1,4-addition of oxazolones to nitroalkenes by bifunctional cinchona alkaloid thiourea organocatalysts: synthesis of alpha,alpha-disubstituted alpha-amino acids. Chemistry (2008) 0.96
A general organocatalyst for direct alpha-functionalization of aldehydes: stereoselective C-C, C-N, C-F, C-Br, and C-S bond-forming reactions. Scope and mechanistic insights. J Am Chem Soc (2005) 0.95
Organocatalytic asymmetric synthesis of alpha,alpha-disubstituted alpha-amino acids and derivatives. J Am Chem Soc (2008) 0.94
Asymmetric synthesis of highly functionalized tetrahydrothiophenes by organocatalytic domino reactions. J Am Chem Soc (2006) 0.94
Direct L-proline-catalyzed asymmetric alpha-amination of ketones. J Am Chem Soc (2002) 0.93
Organocatalytic asymmetric conjugate addition of nitroalkanes to alpha,beta-unsaturated enones using novel imidazoline catalysts. J Org Chem (2002) 0.93
A new approach for an organocatalytic multicomponent domino asymmetric reaction. Angew Chem Int Ed Engl (2007) 0.93
Mechanistic investigation of the 2,5-diphenylpyrrolidine-catalyzed enantioselective alpha-chlorination of aldehydes. Chemistry (2005) 0.93
A simple asymmetric organocatalytic approach to optically active cyclohexenones. Chem Commun (Camb) (2006) 0.93
Organocatalytic asymmetric Michael reaction of cyclic 1,3-dicarbonyl compounds and alpha,beta-unsaturated ketones--a highly atom-economic catalytic one-step formation of optically active warfarin anticoagulant. Angew Chem Int Ed Engl (2003) 0.93
Catalytic, highly enantioselective, direct amination of beta-ketoesters. Angew Chem Int Ed Engl (2003) 0.92
Direct catalytic asymmetric aldol reactions of aldehydes. Chem Commun (Camb) (2002) 0.92
Asymmetric multicomponent domino reactions and highly enantioselective conjugated addition of thiols to alpha,beta-unsaturated aldehydes. J Am Chem Soc (2005) 0.91
Trienamines in asymmetric organocatalysis: Diels-Alder and tandem reactions. J Am Chem Soc (2011) 0.91
Catalytic and enantioselective aza-ene and hetero-Diels-Alder reactions of alkenes and dienes with azodicarboxylates. Org Biomol Chem (2005) 0.91
Asymmetric construction of quaternary stereocenters by direct organocatalytic amination of alpha-substituted alpha-cyanoacetates and beta-dicarbonyl compounds. J Am Chem Soc (2004) 0.90
Direct asymmetric Michael reactions of cyclic 1,3-dicarbonyl compounds and enamines catalyzed by chiral bisoxazoline-copper(II) complexes. J Org Chem (2003) 0.90
Optically active aromatic and heteroaromatic alpha-amino acids by a one-pot catalytic enantioselective addition of aromatic and heteroaromatic C-H bonds to alpha-imino esters. J Org Chem (2002) 0.90
Direct organocatalytic enantioselective mannich reactions of ketimines: an approach to optically active quaternary alpha-amino acid derivatives. Angew Chem Int Ed Engl (2004) 0.90
Organocatalytic asymmetric conjugate addition to allenic esters and ketones. J Am Chem Soc (2008) 0.90
Asymmetric organocatalytic beta-hydroxylation of alpha,beta-unsaturated aldehydes. J Am Chem Soc (2007) 0.89
Organocatalysed asymmetric beta-amination and multicomponent syn-selective diamination of alpha,beta-unsaturated aldehydes. Chemistry (2007) 0.89
Organocatalytic asymmetric 1,6-additions of beta-ketoesters and glycine imine. J Am Chem Soc (2007) 0.89
Organocatalytic enantioselective one-pot synthesis and application of substituted 1,4-dihydropyridines--Hhantzsch ester analogues. Chem Asian J (2008) 0.89
Organocatalytic enantioselective nucleophilic vinylic substitution. Angew Chem Int Ed Engl (2006) 0.88
Direct organo-catalytic asymmetric alpha-amination of aldehydes--a simple approach to optically active alpha-amino aldehydes, alpha-amino alcohols, and alpha-amino acids. Angew Chem Int Ed Engl (2002) 0.88
One-pot organocatalytic domino Michael-aldol and intramolecular SN2 reactions. Asymmetric synthesis of highly functionalized epoxycyclohexanone derivatives. J Am Chem Soc (2006) 0.88
Asymmetric organocatalytic formal [2 + 2]-cycloadditions via bifunctional H-bond directing dienamine catalysis. J Am Chem Soc (2012) 0.87
Organocatalytic asymmetric "anti-Michael" reaction of beta-ketoesters. Chem Commun (Camb) (2007) 0.87
Catalytic enantioselective oxaziridination. J Am Chem Soc (2011) 0.87
Organocatalytic preparation of simple β-hydroxy and β-amino esters: low catalyst loadings and gram-scale synthesis. Org Lett (2010) 0.87
Organocatalytic conjugate addition of malonates to alpha,beta-unsaturated aldehydes: asymmetric formal synthesis of (-)-paroxetine, chiral lactams, and lactones. Angew Chem Int Ed Engl (2006) 0.86
Enantioselective one-pot synthesis of α-amino esters by a phosphine-catalyzed [3+2]-cycloaddition reaction. Chemistry (2011) 0.86
Organocatalytic asymmetric desymmetrization-fragmentation of cyclic ketones. Angew Chem Int Ed Engl (2009) 0.86
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Direct organocatalytic and highly enantio- and diastereoselective Mannich reactions of alpha-substituted alpha-cyanoacetates. Angew Chem Int Ed Engl (2005) 0.86
Highly enantioselective approach to geminal bisphosphonates by organocatalyzed Michael-type addition of beta-ketoesters. Chemistry (2008) 0.86
Non-biaryl atropisomers in organocatalysis. Chemistry (2006) 0.86
Update 1 of: C2-symmetric chiral bis(oxazoline) ligands in asymmetric catalysis. Chem Rev (2011) 0.85
Catalytic asymmetric Henry reactions of silyl nitronates with aldehydes. Org Biomol Chem (2003) 0.85
A cleavable azide resin for direct click chemistry mediated enrichment of alkyne-labeled proteins. Chem Commun (Camb) (2014) 0.85
Asymmetric aza-Michael reactions catalyzed by cinchona alkaloids. J Org Chem (2007) 0.85
The first organocatalytic enantioselective inverse-electron-demand hetero-Diels-Alder reaction. Angew Chem Int Ed Engl (2003) 0.85
Development of a chemical probe for identifying protein targets of α-oxoaldehydes. Chem Commun (Camb) (2013) 0.85
Copper-catalyzed enantioselective Henry reactions of alpha-keto esters: an easy entry to optically active beta-nitro-alpha-hydroxy esters and beta-amino-alpha-hydroxy esters. J Org Chem (2002) 0.85
Enantioselective Friedel-Crafts type addition of indoles to nitro-olefins using a chiral hydrogen-bonding catalyst--synthesis of optically active tetrahydro-beta-carbolines. Org Biomol Chem (2005) 0.84
Organocatalytic diastereo- and enantioselective annulation reactions--construction of optically active 1,2-dihydroisoquinoline and 1,2-dihydrophthalazine derivatives. Angew Chem Int Ed Engl (2005) 0.84
A new organocatalytic concept for asymmetric α-alkylation of aldehydes. J Am Chem Soc (2014) 0.83
Highly enantioselective organocatalytic conjugate addition of malonates to acyclic alpha,beta-unsaturated enones. Angew Chem Int Ed Engl (2003) 0.83
Formation of optically active chromanes by catalytic asymmetric tandem oxa-Michael addition-Friedel-Crafts alkylation reactions. Org Biomol Chem (2003) 0.83
Target-directed organocatalysis: a direct asymmetric catalytic approach to chiral propargylic and allylic fluorides. J Am Chem Soc (2009) 0.83
Organocatalytic enantioselective conjugate addition to alkynones. J Am Chem Soc (2004) 0.83
Enantioselective organocatalytic allylic amination. J Am Chem Soc (2005) 0.83
The first catalytic highly enantioselective alkylation of ketimines--a novel approach to optically active quaternary alpha-amino acids. Chemistry (2003) 0.83
Chirally aminated 2-naphthols--organocatalytic synthesis of non-biaryl atropisomers by asymmetric Friedel-Crafts amination. Angew Chem Int Ed Engl (2006) 0.83
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Direct catalytic asymmetric mannich reactions of malonates and beta-keto esters. Chemistry (2003) 0.82
Organocatalytic activation of polycyclic aromatic compounds for asymmetric Diels-Alder reactions. Angew Chem Int Ed Engl (2012) 0.82
Asymmetric trienamine catalysis for the construction of structurally rigid cyclic α,α-disubstituted amino acid derivatives. Chemistry (2011) 0.82
Achieving molecular complexity by organocatalytic one-pot strategies - a fast entry for synthesis of sphingoids, amino sugars, and polyhydroxylated alpha-amino acids. Angew Chem Int Ed Engl (2009) 0.82
Organocatalytic regio- and asymmetric C-selective S(N)Ar reactions-stereoselective synthesis of optically active spiro-pyrrolidone-3,3'-oxoindoles. J Am Chem Soc (2005) 0.81
Asymmetric organocatalytic thio-Diels-Alder reactions via trienamine catalysis. J Am Chem Soc (2013) 0.81
Controlling the formation of 1 out of 64 stereoisomers using organocatalysis. Chem Commun (Camb) (2008) 0.81
Asymmetric one-pot sequential organo- and gold catalysis for the enantioselective synthesis of dihydropyrrole derivatives. Chemistry (2010) 0.81
Enantioselective hydroxylation of nitroalkenes: an organocatalytic approach. Chem Commun (Camb) (2007) 0.81
Asymmetric organocatalysed [1,3]-sigmatropic rearrangements. Chemistry (2008) 0.81
Asymmetric organocatalytic epoxidations: reactions, scope, mechanisms, and applications. Angew Chem Int Ed Engl (2014) 0.81
Beyond classical reactivity patterns: shifting from 1,4- to 1,6-additions in regio- and enantioselective organocatalyzed vinylogous reactions of olefinic lactones with enals and 2,4-dienals. J Am Chem Soc (2013) 0.81
How to make five contiguous stereocenters in one reaction: asymmetric organocatalytic synthesis of pentasubstituted cyclohexanes. Angew Chem Int Ed Engl (2007) 0.81
Hydrogen-bonding in aminocatalysis: from proline and beyond. Chemistry (2013) 0.81
Catalytic asymmetric Mannich reactions of glycine derivatives with imines. A new approach to optically active alpha,beta-diamino acid derivatives. J Org Chem (2003) 0.81
Organocatalytic asymmetric alpha-bromination of aldehydes and ketones. Chem Commun (Camb) (2005) 0.81
Cofactor activation and substrate binding in pyruvate decarboxylase. Insights into the reaction mechanism from molecular dynamics simulations. Biochemistry (2005) 0.81