Published in J Enzyme Inhib Med Chem on April 01, 2010
Induction of autophagy by a novel small molecule improves aβ pathology and ameliorates cognitive deficits. PLoS One (2013) 0.86
First synthesis of meso-substituted pyrrolo[1,2-a]quinoxalinoporphyrins. Beilstein J Org Chem (2014) 0.77
Multidrug resistance reversal agents. J Med Chem (2003) 1.42
Destructive arthritis in a patient with chikungunya virus infection with persistent specific IgM antibodies. BMC Infect Dis (2009) 1.18
Resveratrol inhibits the growth and induces the apoptosis of both normal and leukemic hematopoietic cells. Carcinogenesis (2002) 1.11
Quercetin induces apoptosis of Trypanosoma brucei gambiense and decreases the proinflammatory response of human macrophages. Antimicrob Agents Chemother (2004) 1.09
Therapeutic and preventive properties of quercetin in experimental arthritis correlate with decreased macrophage inflammatory mediators. Biochem Pharmacol (2006) 1.03
Rutoside decreases human macrophage-derived inflammatory mediators and improves clinical signs in adjuvant-induced arthritis. Arthritis Res Ther (2008) 0.96
8-O-Azeloyl-14-benzoylaconine: a new alkaloid from the roots of Aconitum karacolicum Rapcs and its antiproliferative activities. Bioorg Med Chem (2005) 0.95
Synthesis and preliminary in vitro evaluation of antimycobacterial activity of new pyrrolo[1,2-a] quinoxaline-carboxylic acid hydrazide derivatives. J Enzyme Inhib Med Chem (2004) 0.95
Synthesis of new pyrrolo[1,2-a]quinoxaline derivatives as potential inhibitors of Akt kinase. J Enzyme Inhib Med Chem (2008) 0.93
A Love wave immunosensor for whole E. coli bacteria detection using an innovative two-step immobilisation approach. Biosens Bioelectron (2006) 0.92
Synthesis of a novel class of non-peptide NK-2 receptor ligand, derived from 1-phenyl-3-pyrrol-1-ylindan-2-carboxamides. Bioorg Med Chem (2002) 0.92
IgE mediates killing of intracellular Toxoplasma gondii by human macrophages through CD23-dependent, interleukin-10 sensitive pathway. PLoS One (2011) 0.90
Probing the role of the covalent linkage of ferrocene into a chloroquine template. J Med Chem (2006) 0.87
Plasmodium berghei: dehydroepiandrosterone sulfate reverses chloroquino-resistance in experimental malaria infection; correlation with glucose 6-phosphate dehydrogenase and glutathione synthesis pathway. Biochem Pharmacol (2004) 0.86
Type I interferon signature in the initiation of the immune response in vitiligo. Pigment Cell Melanoma Res (2014) 0.86
Synthesis, analytical behaviour and biological evaluation of new 4-substituted pyrrolo[1,2-a]quinoxalines as antileishmanial agents. Bioorg Med Chem (2006) 0.86
Converting potent indeno[1,2-b]indole inhibitors of protein kinase CK2 into selective inhibitors of the breast cancer resistance protein ABCG2. J Med Chem (2014) 0.84
Pharmacomodulation on the 3-acetylursolic acid skeleton: Design, synthesis, and biological evaluation of novel N-{3-[4-(3-aminopropyl)piperazinyl]propyl}-3-O-acetylursolamide derivatives as antimalarial agents. Bioorg Med Chem (2007) 0.83
CD23 mediates antimycobacterial activity of human macrophages. Infect Immun (2009) 0.82
Synthesis and preliminary evaluation of new 1- and 3-[1-(2-hydroxy-3-phenoxypropyl)]xanthines from 2-amino-2-oxazolines as potential A1 and A2A adenosine receptor antagonists. Bioorg Med Chem (2005) 0.81
Synthesis and preliminary evaluation of new ursolic and oleanolic acids derivatives as antileishmanial agents. J Enzyme Inhib Med Chem (2008) 0.81
Hemisynthesis and antiproliferative properties of mono-[O-(14-benzoylaconine-8-yl)]esters and bis-[O-(14-benzoylaconine-8-yl)]esters. Eur J Med Chem (2012) 0.81
1H and 13C NMR assignments of bioactive indeno[1,2-b]indole-10-one derivatives. Magn Reson Chem (2013) 0.80
Synthesis of new 4-[2-(alkylamino) ethylthio]pyrrolo[1,2-a]quinoxaline and 5-[2-(alkylamino) ethylthio]pyrrolo[1,2-a]thieno[3,2-e]pyrazine derivatives, as potential bacterial multidrug resistance pump inhibitors. J Enzyme Inhib Med Chem (2007) 0.80
Phenotypic effects induced by knock-down of the period clock gene in Bombyx mori. Genet Res (2007) 0.79
Synthesis of omeprazole analogues and evaluation of these as potential inhibitors of the multidrug efflux pump NorA of Staphylococcus aureus. Antimicrob Agents Chemother (2006) 0.79
Pharmaceutical development and optimization of azithromycin suppository for paediatric use. Int J Pharm (2012) 0.79
Modulation of cell proliferation in rat liver cell cultures by new calix[4]arenes. J Enzyme Inhib Med Chem (2006) 0.79
A role of IgE and CD23/NO immune pathway in age-related resistance of Lewis rats to Plasmodium berghei Anka? Microbes Infect (2008) 0.78
New ferrocenic pyrrolo[1,2-a]quinoxaline derivatives: synthesis, and in vitro antimalarial activity. Bioorg Med Chem (2008) 0.78
Halo nevi association in nonsegmental vitiligo affects age at onset and depigmentation pattern. Arch Dermatol (2012) 0.78
Antiproliferative effect on HepaRG cell cultures of new calix[4]arenes. J Enzyme Inhib Med Chem (2010) 0.77
New ferrocenic pyrrolo[1,2-a]quinoxaline derivatives: synthesis, and in vitro antimalarial activity--Part II. Eur J Med Chem (2011) 0.77
Basis of a FTIR spectroscopy methodology for automated evaluation of Akt kinase inhibitor on leukemic cell lines used as model. Anal Bioanal Chem (2012) 0.77
Antiproliferative effect on HepaRG cell cultures of new calix[4]arenes. Part II. J Enzyme Inhib Med Chem (2010) 0.76
Development of a nanoparticulate formulation of diminazene to treat African trypanosomiasis. Nanotechnology (2010) 0.76
2-(3H-1,3-Benzothia-zol-2-yl-idene)-propane-dial. Acta Crystallogr Sect E Struct Rep Online (2011) 0.75
1-Allyl-3-phenyl-quinoxalin-2(1H)-one. Acta Crystallogr Sect E Struct Rep Online (2011) 0.75
tert-Butyl N-{[5-(5-oxohexa-namido)-pyridin-2-yl]amino}-carbamate. Acta Crystallogr Sect E Struct Rep Online (2013) 0.75
Synthesis and primary cytotoxicity evaluation of arylmethylenenaphthofuranones derivatives. J Enzyme Inhib Med Chem (2006) 0.75
Tripodal ligand incorporating dual fluorescent ionophore: a coordinative control of photoinduced electron transfer. Photochem Photobiol Sci (2003) 0.75
Efficient synthesis and first regioselective C-3 direct arylation of imidazo[1,2-b]pyrazoles. Chemistry (2012) 0.75
Development of a rapid RP-HPLC method for the determination of clonazepam in human plasma. J Pharm Biomed Anal (2004) 0.75
Enantioselective synthesis of spirocyclic aminochroman derivatives according to the CN(R,S) strategy. J Org Chem (2003) 0.75
Synthesis of new 4-(E)-alkenylpyrrolo[1,2-a]quinoxalines as antileishmanial agents by Suzuki-Miyaura cross-coupling reactions. J Enzyme Inhib Med Chem (2007) 0.75
Intrinsically disordered amphiphilic peptides as potential targets in drug delivery vehicles. Mol Biosyst (2015) 0.75
Potential of immobilized artificial membrane chromatography for lipophilicity determination of arylpropionic acid non-steroidal anti-inflammatory drugs. J Pharm Biomed Anal (2003) 0.75
Synthesis and initial results for MAO-B inhibition by new N-propargyl-3-pyrrol-1-ylindanamine derivatives, analogues of rasagiline. J Enzyme Inhib Med Chem (2003) 0.75
Synthesis and PC3 androgen-independent prostate cells antiproliferative effect of fagaronine derivatives. J Enzyme Inhib Med Chem (2007) 0.75
Highly diastereoselective synthesis of C6-functionalized dihydroimidazotriazines. Org Lett (2003) 0.75
Efficient metal-free synthesis of various pyrido[2',1':2,3]imidazo- [4,5-b]quinolines. Chemistry (2013) 0.75
Antitumor activity of semisynthetic derivatives of Aconitum alkaloids. Invest New Drugs (2013) 0.75
Synthesis and evaluation of the antiproliferative activity of novel isoindolo[2,1-a]quinoxaline and indolo[1,2-a]quinoxaline derivatives. J Enzyme Inhib Med Chem (2011) 0.75
Antispasmodic and antioxidant activities of fractions and bioactive constituent davidigenin isolated from Mascarenhasia arborescens. J Ethnopharmacol (2010) 0.75
Efficient pallado-catalyzed C6-(het)arylation of Imidazo[1,2-b][1,2,4,5]tetrazines under microwave irradiations. J Comb Chem (2010) 0.75
Smiles rearrangement as a tool for the preparation of dihydrodipyridopyrazines. Org Lett (2009) 0.75
Derivatization of (+/-)-5-[(2-methylphenoxy)methyl]-2-amino-2-oxazoline, an imidazoline binding sites ligand, with (+)-(R)-alpha-methylbenzyl isocyanate for drug monitoring purposes. J Enzyme Inhib Med Chem (2002) 0.75
Proceedings of the 16th annual conference of the Groupement des Pharmacochimistes de l'Arc Atlantique (GP2A). J Enzyme Inhib Med Chem (2008) 0.75
Synthesis and in vitro cytostatic activity of new beta-D-arabino furan[1',2':4,5]oxazolo- and arabino-pyrimidinone derivatives. Eur J Med Chem (2009) 0.75
Anti-leukemia activity of 7-hydroxy-2-substituted-methyl-5H-oxazolo[3,2-a]pyrimidin-5-one derivatives. J Enzyme Inhib Med Chem (2002) 0.75
New efficient route to dissymmetric 2,4-di(het)aryl-pyrido[3,2-d]pyrimidines via regioselective cross-coupling reactions. Org Lett (2007) 0.75