Published in Angew Chem Int Ed Engl on June 08, 2011
Antiplasmodial thiostrepton derivatives: proteasome inhibitors with a dual mode of action. Angew Chem Int Ed Engl (2010) 1.38
Thiostrepton and derivatives exhibit antimalarial and gametocytocidal activity by dually targeting parasite proteasome and apicoplast. Antimicrob Agents Chemother (2011) 1.27
Small molecule transcription factor mimic. J Am Chem Soc (2004) 1.10
Synthesis and structure-activity correlation of natural-product inspired cyclodepsipeptides stabilizing F-actin. J Am Chem Soc (2010) 1.01
Hetero Diels-Alder synthesis of 3-hydroxypyridines: access to the nosiheptide core. J Org Chem (2007) 1.00
A fluorescent probe for the 70 S-ribosomal GTPase-associated center. Chembiochem (2009) 0.99
Total synthesis of chondramide C and its binding mode to F-actin. Angew Chem Int Ed Engl (2008) 0.98
Minimization of a protein-DNA dimerizer. J Am Chem Soc (2007) 0.97
Synthesis and structure-activity correlation of a brunsvicamide-inspired cyclopeptide collection. Chembiochem (2009) 0.97
Biology-oriented synthesis of a natural-product inspired oxepane collection yields a small-molecule activator of the Wnt-pathway. Proc Natl Acad Sci U S A (2011) 0.92
Temperature-sensitive protein-DNA dimerizers. Proc Natl Acad Sci U S A (2005) 0.92
Molecular determinants of microbial resistance to thiopeptide antibiotics. J Am Chem Soc (2010) 0.90
NMR structures of thiostrepton derivatives for characterization of the ribosomal binding site. Angew Chem Int Ed Engl (2011) 0.86
Solid-phase based total synthesis of Jasplakinolide by ring-closing metathesis. Chem Commun (Camb) (2009) 0.84
Small molecules intercept Notch signaling and the early secretory pathway. Nat Chem Biol (2013) 0.83
D-cysteine occurrence in thiostrepton may not necessitate an epimerase. Chem Commun (Camb) (2009) 0.82
Solid-phase based synthesis of jasplakinolide analogs by intramolecular azide-alkyne cycloadditions. Chem Commun (Camb) (2007) 0.81
Regioselective de novo synthesis of cyanohydroxypyridines with a concerted cycloaddition mechanism. J Am Chem Soc (2008) 0.81
Mapping the binding site of thiopeptide antibiotics by proximity-induced covalent capture. J Am Chem Soc (2008) 0.80
Influence of thiostrepton binding on the ribosomal GTPase associated region characterized by molecular dynamics simulation. Bioorg Med Chem (2012) 0.80
Peptide-embedded heterocycles by mild single and multiple Aza-Wittig ring closures. Angew Chem Int Ed Engl (2007) 0.79
Solid-support based total synthesis and stereochemical correction of brunsvicamide A. Org Lett (2008) 0.78
Synthesis and conformational analysis of stevastelin C3 analogues and their activity against the dual-specific vaccina H1-related phosphatase. Chemistry (2008) 0.77
Structure-activity relationships of thiostrepton derivatives: implications for rational drug design. J Comput Aided Mol Des (2014) 0.77
Selective chemical imaging of static actin in live cells. J Am Chem Soc (2012) 0.76
Aza-Wittig-supported synthesis of the A ring of nosiheptide. Angew Chem Int Ed Engl (2009) 0.76
(Z)-Methyl 2-methoxy-imino-3-oxo-butanoate. Acta Crystallogr Sect E Struct Rep Online (2008) 0.75
Biphenomycin B and derivatives: total synthesis and translation inhibition. Chem Asian J (2011) 0.75
Synthesis of (±)-4,5-dia-Parthenolide, an Unnatural Parthenolide Stereoisomer. J Org Chem (2016) 0.75
Flexible total synthesis of biphenomycin B. Chem Commun (Camb) (2008) 0.75
Functional studies of synthetic gramicidin hybrid ion channels in CHO cells. Chembiochem (2007) 0.75
Dynamic combinatorial enrichment of polyconformational D-/L-peptide dimers. Chemistry (2015) 0.75
Aza-Wittig access to chiral imidazol(in)es. Chem Commun (Camb) (2009) 0.75
Iterative antimicrobial candidate selection from informed d-/l-Peptide dimer libraries. Chembiochem (2013) 0.75