Cristian G Bologa

Author PubWeight™ 26.22‹?›

Top papers

Rank Title Journal Year PubWeight™‹?›
1 In vivo effects of a GPR30 antagonist. Nat Chem Biol 2009 2.39
2 A crowdsourcing evaluation of the NIH chemical probes. Nat Chem Biol 2009 2.29
3 Drug Repurposing from an Academic Perspective. Drug Discov Today Ther Strateg 2011 1.68
4 Identification of a GPER/GPR30 antagonist with improved estrogen receptor counterselectivity. J Steroid Biochem Mol Biol 2011 1.42
5 Associating Drugs, Targets and Clinical Outcomes into an Integrated Network Affords a New Platform for Computer-Aided Drug Repurposing. Mol Inform 2011 1.35
6 Lead-like, drug-like or "Pub-like": how different are they? J Comput Aided Mol Des 2007 1.21
7 Real-time analysis of conformation-sensitive antibody binding provides new insights into integrin conformational regulation. J Biol Chem 2009 1.14
8 Modulation of bitter taste perception by a small molecule hTAS2R antagonist. Curr Biol 2010 1.09
9 Biomolecular screening of formylpeptide receptor ligands with a sensitive, quantitative, high-throughput flow cytometry platform. Nat Protoc 2006 1.07
10 The CARLSBAD database: a confederated database of chemical bioactivities. Database (Oxford) 2013 1.05
11 Structural simplification of bioactive natural products with multicomponent synthesis. 3. Fused uracil-containing heterocycles as novel topoisomerase-targeting agents. J Med Chem 2011 0.95
12 Strategies for compound selection. Curr Drug Discov Technol 2004 0.95
13 Identification of a small molecule yeast TORC1 inhibitor with a multiplex screen based on flow cytometry. ACS Chem Biol 2012 0.95
14 High-throughput screen for the chemical inhibitors of antiapoptotic bcl-2 family proteins by multiplex flow cytometry. Assay Drug Dev Technol 2011 0.89
15 Microbial efflux pump inhibition: tactics and strategies. Curr Pharm Des 2011 0.88
16 Fluorescent substrates for flow cytometric evaluation of efflux inhibition in ABCB1, ABCC1, and ABCG2 transporters. Anal Biochem 2013 0.88
17 A novel flow cytometric HTS assay reveals functional modulators of ATP binding cassette transporter ABCB6. PLoS One 2012 0.85
18 Conformational mAb as a tool for integrin ligand discovery. Assay Drug Dev Technol 2009 0.84
19 A selective ATP-binding cassette subfamily G member 2 efflux inhibitor revealed via high-throughput flow cytometry. J Biomol Screen 2012 0.82
20 Therapeutic options and emerging alternatives for multidrug resistant staphylococcal infections. Curr Pharm Des 2015 0.79
21 Structural determinants of the alpha2 adrenoceptor subtype selectivity. J Mol Graph Model 2011 0.78
22 Post-high-throughput screening analysis: an empirical compound prioritization scheme. J Biomol Screen 2005 0.77
23 Of possible cheminformatics futures. J Comput Aided Mol Des 2011 0.77
24 Ligand-directed profiling of organelles with internalizing phage libraries. Curr Protoc Protein Sci 2015 0.75