Published in ACS Comb Sci on February 10, 2012
Stereocontrol in asymmetric γ-lactam syntheses from imines and cyanosuccinic anhydrides. Org Lett (2013) 0.92
Stereoselective synthesis of γ-lactams from imines and cyanosuccinic anhydrides. Org Lett (2013) 0.78
Synthesis of a library of "lead-like" γ-lactams by a one pot, four-component reaction. ACS Comb Sci (2013) 0.75
Diastereoselective synthesis of γ- and δ-lactams from imines and sulfone-substituted anhydrides. J Org Chem (2014) 0.75
A construction of 4,4-spirocyclic γ-lactams by tandem radical cyclization with carbon monoxide. Beilstein J Org Chem (2013) 0.75
Salinosporamide A: a highly cytotoxic proteasome inhibitor from a novel microbial source, a marine bacterium of the new genus salinospora. Angew Chem Int Ed Engl (2003) 4.50
Lead- and drug-like compounds: the rule-of-five revolution. Drug Discov Today Technol (2004) 3.57
Pursuing the leadlikeness concept in pharmaceutical research. Curr Opin Chem Biol (2004) 2.36
Pyrrolidinyl-spirooxindole natural products as inspirations for the development of potential therapeutic agents. Angew Chem Int Ed Engl (2007) 2.07
Discovery and development of the anticancer agent salinosporamide A (NPI-0052). Bioorg Med Chem (2008) 1.77
Cooperative catalysis by carbenes and Lewis acids in a highly stereoselective route to gamma-lactams. Nat Chem (2010) 1.44
Synthesis of diverse lactam carboxamides leading to the discovery of a new transcription-factor inhibitor. Angew Chem Int Ed Engl (2007) 1.38
N-heterocyclic carbene and Brønsted acid cooperative catalysis: asymmetric synthesis of trans-γ-lactams. J Am Chem Soc (2011) 1.36
Azomethine ylide cycloaddition/reductive heterocyclization approach to oxindole alkaloids: asymmetric synthesis of (-)-horsfiline. J Org Chem (2001) 1.34
Cyclic anhydrides in formal cycloadditions and multicomponent reactions. Chem Rev (2009) 1.07
Diastereoselective synthesis of gamma-lactams by a one-pot, four-component reaction. Org Lett (2007) 1.00
Lajollamycin, a nitro-tetraene spiro-beta-lactone-gamma-lactam antibiotic from the marine actinomycete Streptomyces nodosus. J Nat Prod (2005) 0.96
Cycloaddition reactions of imines with 3-thiosuccinic anhydrides: synthesis of the tricyclic core of martinellic acid. Org Lett (2006) 0.94
Amide enolate additions to acylsilanes: in situ generation of unusual and stereoselective homoenolate equivalents. J Am Chem Soc (2009) 0.92
Ammonia synthons for the multicomponent assembly of complex gamma-lactams. Proc Natl Acad Sci U S A (2011) 0.89
New dimeric compounds of avenanthramide phytoalexin in oats. J Org Chem (2007) 0.86
Divergent structural complexity from a linear reaction sequence: synthesis of fused and spirobicyclic gamma-lactams from common synthetic precursors. J Comb Chem (2006) 0.85
Heliotropamide, a novel oxopyrrolidine-3-carboxamide from Heliotropium ovalifolium. J Nat Prod (2003) 0.85
Chemical inhibition of the mitochondrial division dynamin reveals its role in Bax/Bak-dependent mitochondrial outer membrane permeabilization. Dev Cell (2008) 5.67
Synthesis of a stable compound with fivefold bonding between two chromium(I) centers. Science (2005) 1.96
Methylene-bridged glycoluril dimers: synthetic methods. J Org Chem (2002) 1.96
Reversible reactions of ethylene with distannynes under ambient conditions. Science (2009) 1.46
Stereoselective C-glycosylation reactions of ribose derivatives: electronic effects of five-membered ring oxocarbenium ions. J Am Chem Soc (2005) 1.42
Synthesis of antimicrobial natural products targeting FtsZ: (+/-)-dichamanetin and (+/-)-2' ''-hydroxy-5' '-benzylisouvarinol-B. Org Lett (2005) 1.39
Synthesis of diverse lactam carboxamides leading to the discovery of a new transcription-factor inhibitor. Angew Chem Int Ed Engl (2007) 1.38
Potent s-cis-locked bithiazole correctors of DeltaF508 cystic fibrosis transmembrane conductance regulator cellular processing for cystic fibrosis therapy. J Med Chem (2008) 1.29
Synthesis and relaxometric studies of a dendrimer-based pH-responsive MRI contrast agent. Chemistry (2008) 1.28
Isolation of a stable, acyclic, two-coordinate silylene. J Am Chem Soc (2012) 1.23
Diastereoselective magnesium halide-catalyzed anti-aldol reactions of chiral N-acyloxazolidinones. J Am Chem Soc (2002) 1.21
Interpenetrating As20 fullerene and Ni12 icosahedra in the onion-skin [As@Ni12@As20]3- ion. Science (2003) 1.16
Stannous chloride in alcohol: a one-pot conversion of 2-nitro-N-arylbenzamides to 2,3-dihydro-1H-quinazoline-4-ones. J Org Chem (2005) 1.15
Regarding the stability of d(0) monocyclopentadienyl zirconium acetamidinate complexes bearing alkyl substituents with beta-hydrogens. J Am Chem Soc (2002) 1.13
An oxazolo[3,2-b]indazole route to 1H-indazolones. Org Lett (2009) 1.12
Magnetic properties and negative colossal magnetoresistance of the rare earth Zintl phase EuIn2As2. Inorg Chem (2008) 1.09
Cyclic anhydrides in formal cycloadditions and multicomponent reactions. Chem Rev (2009) 1.07
Recent advances in multicomponent reactions for diversity-oriented synthesis. Curr Opin Chem Biol (2010) 1.06
Comparison of small molecule inhibitors of the bacterial cell division protein FtsZ and identification of a reliable cross-species inhibitor. ACS Chem Biol (2012) 1.04
Pyrazolylthiazole as DeltaF508-cystic fibrosis transmembrane conductance regulator correctors with improved hydrophilicity compared to bithiazoles. J Med Chem (2010) 1.04
A structurally diverse library of polycyclic lactams resulting from systematic placement of proximal functional groups. Angew Chem Int Ed Engl (2006) 1.03
Magnesium halide-catalyzed anti-aldol reactions of chiral N-acylthiazolidinethiones. Org Lett (2002) 1.03
Ion channel formation from a calix[4]arene amide that binds HCl. J Am Chem Soc (2002) 1.02
Titanium-catalyzed stereoselective synthesis of spirooxindole oxazolines. Org Lett (2010) 1.01
Inhibitors of bacterial tubulin target bacterial membranes in vivo. Medchemcomm (2012) 1.01
Diastereoselective synthesis of gamma-lactams by a one-pot, four-component reaction. Org Lett (2007) 1.00
Catalytic asymmetric synthesis of substituted 3-hydroxy-2-oxindoles. Angew Chem Int Ed Engl (2010) 1.00
Synthesis of (-)-viriditoxin: a 6,6'-binaphthopyran-2-one that targets the bacterial cell division protein FtsZ. Angew Chem Int Ed Engl (2011) 0.98
Profiling base excision repair glycosylases with synthesized transition state analogs. Bioorg Med Chem Lett (2011) 0.98
Fluoride-selective host based on anion-pi interactions, ion pairing, and hydrogen bonding: synthesis and fluoride-ion sandwich complex. Angew Chem Int Ed Engl (2007) 0.97
Diastereoselective formation of glycoluril dimers: isomerization mechanism and implications for cucurbit[n]uril synthesis. J Am Chem Soc (2002) 0.97
Molecular clips form isostructural dimeric aggregates from benzene to water. J Am Chem Soc (2004) 0.96
A one-pot-three-step route to triazolotriazepinoindazolones from oxazolino-2H-indazoles. Org Lett (2012) 0.96
Lipophilic G-quadruplexes are self-assembled ion pair receptors, and the bound anion modulates the kinetic stability of these complexes. J Am Chem Soc (2003) 0.96
Synthesis of antimicrobial natural products targeting FtsZ: (+)-totarol and related totarane diterpenes. Org Lett (2010) 0.95
Cycloaddition reactions of imines with 3-thiosuccinic anhydrides: synthesis of the tricyclic core of martinellic acid. Org Lett (2006) 0.94
Facile activation of dihydrogen by an unsaturated heavier main group compound. J Am Chem Soc (2005) 0.93
Intramolecular cycloaddition of azomethine ylides in the preparation of pyrrolidino[2',3':3,4]pyrrolidino[1,2- a]benzimidazoles. Org Lett (2007) 0.93
Identification of the molecular target of small molecule inhibitors of HDL receptor SR-BI activity. Biochemistry (2007) 0.93
The correct structure of aquatolide-experimental validation of a theoretically-predicted structural revision. J Am Chem Soc (2012) 0.93
Stereocontrol in asymmetric γ-lactam syntheses from imines and cyanosuccinic anhydrides. Org Lett (2013) 0.92
A new synthetic route to (North)-methanocarba nucleosides designed as A3 adenosine receptor agonists. J Org Chem (2005) 0.92
A new copper acetate-bis(oxazoline)-catalyzed, enantioselective Henry reaction. J Am Chem Soc (2003) 0.91
Heterocycle-heterocycle strategies: (2-nitrophenyl)isoxazole precursors to 4-aminoquinolines, 1H-indoles, and quinolin-4(1H)-ones. Org Lett (2013) 0.91
Antinociceptive properties of coumarins, steroid and dihydrostyryl-2-pyrones from Polygala sabulosa (Polygalaceae) in mice. J Pharm Pharmacol (2006) 0.91
Molecular clips that undergo heterochiral aggregation and self-sorting. Angew Chem Int Ed Engl (2002) 0.90
Diazocinones: synthesis and conformational analysis. J Org Chem (2006) 0.90
Influence of HDL-cholesterol-elevating drugs on the in vitro activity of the HDL receptor SR-BI. J Lipid Res (2007) 0.89
Diastereoselective nucleophilic substitution reactions of oxasilacyclopentane acetals: application of the "inside attack" model for reactions of five-membered ring oxocarbenium ions. J Org Chem (2002) 0.89
Ammonia synthons for the multicomponent assembly of complex gamma-lactams. Proc Natl Acad Sci U S A (2011) 0.89
Oxatriquinane and oxatriquinacene: extraordinary oxonium ions. J Am Chem Soc (2008) 0.89
One-step synthesis of complex nitrogen heterocycles from imines and alkyl-substituted maleic anhydrides. Org Lett (2009) 0.88
Characterization of Caulobacter crescentus FtsZ protein using dynamic light scattering. J Biol Chem (2012) 0.88
Understanding molecular recognition of promiscuity of thermophilic methionine adenosyltransferase sMAT from Sulfolobus solfataricus. FEBS J (2014) 0.88
Efficient syntheses of the unknown quinolino[2,3-c]cinnolines; synthesis of neocryptolepines. Org Lett (2010) 0.88
Four psychrotolerant species with high chemical diversity consistently producing cycloaspeptide A, Penicillium jamesonlandense sp. nov., Penicillium ribium sp. nov., Penicillium soppii and Penicillium lanosum. Int J Syst Evol Microbiol (2006) 0.88
Direct displacement of alkoxy groups of vinylogous esters by Grignard reagents. J Org Chem (2011) 0.87
Synthesis and stereochemical assignment of brasilibactin A. Org Lett (2007) 0.86
Zinc-catalyzed silylation of terminal alkynes. J Org Chem (2008) 0.86
Design and synthesis of propeller-shaped dispiroisoxazolinopiperidinochromanones. J Comb Chem (2008) 0.86
Regulating supramolecular function in membranes: calixarenes that enable or inhibit transmembrane Cl- transport. Angew Chem Int Ed Engl (2006) 0.86
Cucurbit[n]uril analogues: synthetic and mechanistic studies. J Org Chem (2005) 0.86
Second-Generation Synthesis of (-)-Viriditoxin. Synthesis (Stuttg) (2012) 0.85
Two-coordinate, homoleptic manganese(II) primary terphenyl amido complexes: the effects of secondary coordination on geometry and Lewis base complexation. Dalton Trans (2009) 0.85
N-Benzyl-3-sulfonamidopyrrolidines are a New Class of Bacterial DNA Gyrase Inhibitors. ACS Med Chem Lett (2011) 0.85
Parallel Synthesis of bis-heterocyclic isoxazolylmethyl- and isoxazolinylmethylpyrazoles. J Comb Chem (2010) 0.85
Divergent structural complexity from a linear reaction sequence: synthesis of fused and spirobicyclic gamma-lactams from common synthetic precursors. J Comb Chem (2006) 0.85
Catalytic Alkene Cyclization Reactions for the Stereoselective Synthesis of Complex "Terpenoid-like" Heterocycles. Chem Sci (2012) 0.85
Dispersion force stabilized two-coordinate transition metal-amido complexes of the -N(SiMe3)Dipp (Dipp = C6H3-2,6-Pr(i)2) ligand: structural, spectroscopic, magnetic, and computational studies. Inorg Chem (2013) 0.85
Antinociceptive effect of the Polygala sabulosa hydroalcoholic extract in mice: evidence for the involvement of glutamatergic receptors and cytokine pathways. Basic Clin Pharmacol Toxicol (2008) 0.84
Practical synthesis of PC190723, an inhibitor of the bacterial cell division protein FtsZ. J Org Chem (2010) 0.84
Reactions of the heavier group 14 element alkyne analogues Ar'EEAr' (Ar' = C6H3-2,6(C6H3-2,6-Pri2)2; E = Ge, Sn) with unsaturated molecules: probing the character of the EE multiple bonds. J Am Chem Soc (2005) 0.84
Cucurbit[n]uril analogues. Org Lett (2003) 0.84
Selective nucleophilic chemistry in the synthesis of 5-carbamoyl-3-sulfanylmethylisoxazole-4-carboxylic acids. J Comb Chem (2007) 0.83
Asymmetric catalysis: resin-bound hydroxyprolylthreonine derivatives in enamine-mediated reactions. Angew Chem Int Ed Engl (2008) 0.83
Enantioselective intramolecular C-H insertion reactions of donor-donor metal carbenoids. J Am Chem Soc (2014) 0.83
"Matched/mismatched" diastereomeric dirhodium(II) carboxamidate catalyst pairs. Structure-selectivity correlations in diazo decomposition and hetero-Diels-Alder reactions. J Org Chem (2005) 0.82
Designed self-assembly of molecular necklaces using host-stabilized charge-transfer interactions. J Am Chem Soc (2004) 0.82
Diastereoselective synthesis of (±)-heliotropamide by a one-pot, four-component reaction. J Org Chem (2010) 0.82
Azatriquinane as a platform for tripodal metal complexes and calixiform scaffolds. Angew Chem Int Ed Engl (2010) 0.82
Very large changes in bond length and bond angle in a heavy group 14 element alkyne analogue by modification of a remote ligand substituent. J Am Chem Soc (2006) 0.81
Addition of H2 to distannynes under ambient conditions. Chem Commun (Camb) (2008) 0.81
Antinociceptive and gastroprotective actions of ethanolic extract from Pluchea sagittalis (Lam.) Cabrera. J Ethnopharmacol (2011) 0.81
Synthesis of 6,6'-binaphthopyran-2-one natural products: pigmentosin A, talaroderxines A and B. Org Lett (2012) 0.81
Self-sorting molecular clips. J Org Chem (2008) 0.81
Synthesis of kaempferitrin. J Org Chem (2007) 0.80
Linear and nonlinear two-coordinate vanadium complexes: synthesis, characterization, and magnetic properties of V(II) amides. J Am Chem Soc (2013) 0.80
A pirouette on a metallofullerene sphere: interconversion of isomers of N-tritylpyrrolidino I(h) Sc3N@C80. J Am Chem Soc (2006) 0.80
Multicomponent macrocyclization reactions (MCMRs) employing highly reactive acyl ketene and nitrile oxide intermediates. Org Lett (2011) 0.80
Synthesis, structure, and magnetic and electrochemical properties of quasi-linear and linear iron(I), cobalt(I), and nickel(I) amido complexes. Inorg Chem (2014) 0.80