Published in J Org Chem on May 10, 2012
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Toward understanding how the lactone moiety of discodermolide affects activity. J Am Chem Soc (2005) 0.96
Multiple multicomponent macrocyclizations (MiBs): a strategic development toward macrocycle diversity. Chem Rev (2009) 0.91
Multiple multicomponent macrocyclizations including bifunctional building blocks (MiBs) based on Staudinger and Passerini three-component reactions. J Org Chem (2008) 0.88
Enantioselective synthesis and biological activity of (3S,4R)- and (3S,4S)-3-hydroxy-4-hydroxymethyl- 4-butanolides in relation to PGE2. J Med Chem (2004) 0.86
Design, synthesis, and evaluation of carbamate-substituted analogues of (+)-discodermolide. Org Lett (2005) 0.83
Diversity oriented one-pot synthesis of complex macrocycles: very large steroid-peptoid hybrids from multiple multicomponent reactions including bifunctional building blocks. Angew Chem Int Ed Engl (2005) 0.82
Design, synthesis, and biological evaluation of potent discodermolide fluorescent and photoaffinity molecular probes. Org Lett (2005) 0.82
Rapid access to N-substituted diketopiperazines by one-pot Ugi-4CR/deprotection+activation/cyclization (UDAC). J Comb Chem (2009) 0.80
Isolation, structure elucidation, total synthesis, and evaluation of new natural and synthetic ceramides on human SK-MEL-1 melanoma cells. J Med Chem (2006) 0.79
Design, synthesis, and evaluation of analogues of (+)-14-normethyldiscodermolide. Org Lett (2005) 0.78
Synthesis of steroid-biaryl ether hybrid macrocycles with high skeletal and side chain variability by multiple multicomponent macrocyclization including bifunctional building blocks. J Org Chem (2006) 0.77
Freezing imine exchange in dynamic combinatorial libraries with Ugi reactions: versatile access to templated macrocycles. Org Lett (2007) 0.77
New insights into the structure-cytotoxicity relationship of spirostan saponins and related glycosides. Bioorg Med Chem (2012) 0.77
Sesquiterpene lactones from Gonospermum gomerae and G. fruticosum and their cytotoxic activities. J Nat Prod (2008) 0.76
Synthesis of novel spirostanic saponins and their cytotoxic activity. Bioorg Med Chem (2007) 0.76
A new ceramide from Suillus luteus and its cytotoxic activity against human melanoma cells. Chem Biodivers (2008) 0.76
A new lupene triterpenetriol and anticholinesterase activity of Salvia sclareoides. Fitoterapia (2007) 0.76
New quinoline alkaloid from Ruta graveolens aerial parts and evaluation of the antifertility activity. Nat Prod Res (2014) 0.75
A chemotaxonomic study of endemic species of genus Tanacetum from the Canary Islands. Phytochemistry (2013) 0.75
Expanding the Scope of Ugi Multicomponent Bioconjugation to Produce Pneumococcal Multivalent Glycoconjugates as Vaccine Candidates. Bioconjug Chem (2020) 0.75
Organocatalytic asymmetric epoxidation and tandem epoxidation/Passerini reaction under eco-friendly reaction conditions. Org Biomol Chem (2012) 0.75
Secondary metabolites from two species of Pulicaria and their cytotoxic activity. Chem Biodivers (2011) 0.75
A new flavonoid and other constituents from Centaurea nicaeensis All. var. walliana M. Nat Prod Res (2011) 0.75
Multicomponent combinatorial development and conformational analysis of prolyl peptide-peptoid hybrid catalysts: application in the direct asymmetric Michael addition. J Org Chem (2013) 0.75
Chemotaxonomy of Gonospermum and related genera. Phytochemistry (2010) 0.75
Chemical constituents of Tolpis species. Fitoterapia (2009) 0.75
Secondary metabolites from two species of Tolpis and their biological activities. Molecules (2012) 0.75
A multicomponent macrocyclization strategy to natural product-like cyclic lipopeptides: synthesis and anticancer evaluation of surfactin and mycosubtilin analogues. Org Biomol Chem (2017) 0.75
Multicomponent ligation of steroids: creating diversity at the linkage moiety of bis-spirostanic conjugates by Ugi reactions. ACS Comb Sci (2013) 0.75
Combinatorial multicomponent access to natural-products-inspired peptidomimetics: discovery of selective inhibitors of microbial metallo-aminopeptidases. ChemMedChem (2014) 0.75
Effect of C-ring modifications on the cytotoxicity of spirostan saponins and related glycosides. Bioorg Med Chem (2012) 0.75
Bidirectional macrocyclization of peptides by double multicomponent reactions. Org Biomol Chem (2015) 0.75