Published in Eur J Med Chem on November 07, 2012
Biological evaluation of hydroxynaphthoquinones as anti-malarials. Malar J (2013) 0.87
Potential of 2-hydroxy-3-phenylsulfanylmethyl-[1,4]-naphthoquinones against Leishmania (L.) infantum: biological activity and structure-activity relationships. PLoS One (2014) 0.75
Insights into cytochrome bc1 complex binding mode of antimalarial 2-hydroxy-1,4-naphthoquinones through molecular modelling. Mem Inst Oswaldo Cruz (2017) 0.75
Growing Latin American science. Science (2012) 2.03
Novel 1,2,3-triazole derivatives for use against Mycobacterium tuberculosis H37Rv (ATCC 27294) strain. J Med Chem (2011) 1.57
Synthesis and evaluation of new difluoromethyl azoles as antileishmanial agents. Eur J Med Chem (2007) 1.38
Synthesis, tuberculosis inhibitory activity, and SAR study of N-substituted-phenyl-1,2,3-triazole derivatives. Bioorg Med Chem (2006) 1.13
Exposure of Plasmodium sporozoites to the intracellular concentration of potassium enhances infectivity and reduces cell passage activity. Mol Biochem Parasitol (2007) 1.10
Synthesis and anti-HSV-1 activity of new 1,2,3-triazole derivatives. Bioorg Med Chem (2011) 1.03
Regulation of multidrug resistance-associated protein 2 by calcium signaling in mouse liver. Hepatology (2010) 1.01
Synthesis, biological activity, and molecular modeling studies of 1H-1,2,3-triazole derivatives of carbohydrates as alpha-glucosidases inhibitors. J Med Chem (2010) 0.97
Identification of a potential lead structure for designing new antimicrobials to treat infections caused by Staphylococcus epidermidis-resistant strains. Curr Microbiol (2008) 0.97
Synthesis and antitubercular activity of novel Schiff bases derived from d-mannitol. Carbohydr Res (2009) 0.94
Antiviral evaluation of N-amino-1,2,3-triazoles against Cantagalo virus replication in cell culture. Eur J Med Chem (2009) 0.91
Antiplatelet properties of novel N-substituted-phenyl-1,2,3-triazole-4-acylhydrazone derivatives. Bioorg Med Chem (2003) 0.91
Melatonin and IP3-induced Ca2+ release from intracellular stores in the malaria parasite Plasmodium falciparum within infected red blood cells. J Biol Chem (2010) 0.90
Synthesis and anti-HSV-1 activity of quinolonic acyclovir analogues. Bioorg Med Chem Lett (2006) 0.90
Synthesis, antiplatelet and in silico evaluations of novel N-substituted-phenylamino-5-methyl-1H-1,2,3-triazole-4-carbohydrazides. Bioorg Med Chem (2009) 0.87
Synthesis and anti-Trypanosoma cruzi activity of derivatives from nor-lapachones and lapachones. Bioorg Med Chem (2008) 0.87
Biological evaluation of hydroxynaphthoquinones as anti-malarials. Malar J (2013) 0.87
Involvement of TSSA (trypomastigote small surface antigen) in Trypanosoma cruzi invasion of mammalian cells. Biochem J (2012) 0.86
Influenza A viral nucleoprotein interacts with cytoskeleton scaffolding protein α-actinin-4 for viral replication. FEBS J (2014) 0.86
Synthesis, antitubercular activity, and SAR study of N-substituted-phenylamino-5-methyl-1H-1,2,3-triazole-4-carbohydrazides. Bioorg Med Chem (2011) 0.84
Synthesis and potent antitumor activity of new arylamino derivatives of nor-beta-lapachone and nor-alpha-lapachone. Bioorg Med Chem (2007) 0.84
The compound 6-chloro-1,4-dihydro-4-oxo-1-(beta-D-ribofuranosyl) quinoline-3-carboxylic acid inhibits HIV-1 replication by targeting the enzyme reverse transcriptase. Curr HIV Res (2008) 0.83
Inhibition of HSV-1 replication and HSV DNA polymerase by the chloroxoquinolinic ribonucleoside 6-chloro-1,4-dihydro-4-oxo-1-(beta-D-ribofuranosyl) quinoline-3-carboxylic acid and its aglycone. Antiviral Res (2007) 0.83
Quantitative structure-activity relationship in aziridinyl-1,4-naphthoquinone antimalarials: study of theoretical correlations by the PM3 method. Bioorg Med Chem (2004) 0.83
Synthesis using microwave irradiation and antibacterial evaluation of new N,O-acetals and N,S-acetals derived from 2-amino-1,4-naphthoquinones. Eur J Med Chem (2013) 0.82
Identification of nor-β-lapachone derivatives as potential antibacterial compounds against Enterococcus faecalis clinical strain. Curr Microbiol (2010) 0.81
Synthesis, antiviral activity and molecular modeling of oxoquinoline derivatives. Bioorg Med Chem (2009) 0.81
New oxirane derivatives of 1,4-naphthoquinones and their evaluation against T. cruzi epimastigote forms. Bioorg Med Chem (2012) 0.81
Potent naphthoquinones against antimony-sensitive and -resistant Leishmania parasites: synthesis of novel α- and nor-α-lapachone-based 1,2,3-triazoles by copper-catalyzed azide-alkyne cycloaddition. Eur J Med Chem (2013) 0.80
Nitroxides attenuate carrageenan-induced inflammation in rat paws by reducing neutrophil infiltration and the resulting myeloperoxidase-mediated damage. Free Radic Biol Med (2012) 0.80
Synthesis, biological, and theoretical evaluations of new 1,2,3-triazoles against the hemolytic profile of the Lachesis muta snake venom. Bioorg Med Chem (2009) 0.79
In vivo uptake of a haem analogue Zn protoporphyrin IX by the human malaria parasite P. falciparum-infected red blood cells. Cell Biol Int (2010) 0.79
Novel 1H-1,2,3-, 2H-1,2,3-, 1H-1,2,4- and 4H-1,2,4-triazole derivatives: a patent review (2008 - 2011). Expert Opin Ther Pat (2013) 0.79
Molecular design, synthesis and biological evaluation of 1,4-dihydro-4-oxoquinoline ribonucleosides as TcGAPDH inhibitors with trypanocidal activity. Bioorg Med Chem Lett (2013) 0.79
Naphthoquinoidal [1,2,3]-triazole, a new structural moiety active against Trypanosoma cruzi. Eur J Med Chem (2007) 0.79
Synthesis, HIV-RT inhibitory activity and SAR of 1-benzyl-1H-1,2,3-triazole derivatives of carbohydrates. Eur J Med Chem (2008) 0.79
Synthesis of new 9-hydroxy-α- and 7-hydroxy-β-pyran naphthoquinones and cytotoxicity against cancer cell lines. Org Biomol Chem (2011) 0.79
FRET peptides reveal differential proteolytic activation in intraerythrocytic stages of the malaria parasites Plasmodium berghei and Plasmodium yoelii. Int J Parasitol (2010) 0.79
Synthesis of alpha- and beta-pyran naphthoquinones as a new class of antitubercular agents. Arch Pharm (Weinheim) (2010) 0.78
3-arylamino and 3-alkoxy-nor-beta-lapachone derivatives: synthesis and cytotoxicity against cancer cell lines. J Med Chem (2010) 0.78
Oxyrane derivative of alpha-lapachone is potent growth inhibitor of Trypanosoma cruzi epimastigote forms. Parasitol Res (2006) 0.78
Singlet oxygen production by pyrano and furano 1,4-naphthoquinones in non-aqueous medium. Photochem Photobiol Sci (2012) 0.77
Synthesis of 1H-1,2,3-triazoles and study of their antifungal and cytotoxicity activities. Med Chem (2013) 0.76
Trypanosoma cruzi: insights into naphthoquinone effects on growth and proteinase activity. Exp Parasitol (2010) 0.76
Synthesis of new chlorin e6 trimethyl and protoporphyrin IX dimethyl ester derivatives and their photophysical and electrochemical characterizations. Chemistry (2014) 0.76
Structure-activity relationships of novel inhibitors of glyceraldehyde-3-phosphate dehydrogenase. Bioorg Med Chem Lett (2004) 0.76
Characterization of HIV-1 enzyme reverse transcriptase inhibition by the compound 6-chloro-1,4-dihydro-4-oxo-1-(beta-D-ribofuranosyl) quinoline-3-carboxylic acid through kinetic and in silico studies. Curr HIV Res (2009) 0.76
Antivenom effects of 1,2,3-triazoles against Bothrops jararaca and Lachesis muta snakes. Biomed Res Int (2013) 0.75
Synthesis and anti-Trypanosoma cruzi activity of naphthoquinone-containing triazoles: electrochemical studies on the effects of the quinoidal moiety. Bioorg Med Chem (2013) 0.75
Advances in drug discovery to assess cholinergic neurotransmission: a systematic review. Curr Drug Discov Technol (2008) 0.75
One-pot preparation of substituted pyrroles from alpha-diazocarbonyl compounds. Beilstein J Org Chem (2008) 0.75
Synthesis and evaluation of D-gluconamides as green mineral scales. Carbohydr Res (2012) 0.75
Recent advances in the synthesis of new antimycobacterial agents based on the 1H-1,2,3-triazoles. Curr Top Med Chem (2013) 0.75
New families of hetero-tri-spin 2p-3d-4f complexes: synthesis, crystal structures, and magnetic properties. Inorg Chem (2014) 0.75
Synthesis and antiviral evaluation of isatin ribonucleosides. Nucleosides Nucleotides Nucleic Acids (2003) 0.75
pi-Stacked dimers in 6-methoxy-3,3-dimethyl-3H-benzo[f]chromene, and centrosymmetric dimers containing C-H...pi(arene) hydrogen bonds in racemic 3-bromo-2,2,6,6-tetramethyl-3,4-dihydro-2H,6H-1,5-dioxatriphenylene. Acta Crystallogr C (2007) 0.75
Tuberculosis: finding a new potential antimycobacterium derivative in a aldehyde-arylhydrazone-oxoquinoline series. Curr Microbiol (2012) 0.75
Synthesis and antiviral activities of new pyrazolo[4,3-c]quinolin-3-ones and their ribonucleoside derivatives. Nucleosides Nucleotides Nucleic Acids (2004) 0.75
Synthesis of 1,2,3-triazole glycoconjugates as inhibitors of α-glucosidases. Carbohydr Res (2012) 0.75
Inner reorganization during the radical-biradical transition in a nor-beta-lapachone derivative possessing two redox centers. Org Biomol Chem (2008) 0.75
Oxoquinoline derivatives: identification and structure-activity relationship (SAR) analysis of new anti-HSV-1 agents. Curr Microbiol (2011) 0.75
Synthesis, Anticlotting and Antiplatelet Effects of 1,2,3-Triazoles Derivatives. Med Chem (2016) 0.75
Complete and unambiguous assignments of 1H and 13C chemical shifts of new arylamino derivatives of ortho-naphthofuranquinones. Magn Reson Chem (2008) 0.75
Three ethyl 5-amino-1-aryl-1H-imidazole-4-carboxylates: hydrogen-bonded supramolecular structures in one, two and three dimensions. Acta Crystallogr C (2006) 0.75