Niche-based screening identifies small-molecule inhibitors of leukemia stem cells.

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Published in Nat Chem Biol on October 27, 2013

Authors

Kimberly A Hartwell1,2,3, Peter G Miller2,3, Siddhartha Mukherjee4, Alissa R Kahn5, Alison L Stewart1, David J Logan1, Joseph M Negri1, Mildred Duvet1,4, Marcus Järås2, Rishi Puram2,3, Vlado Dancik1, Fatima Al-Shahrour1,2, Thomas Kindler2, Zuzana Tothova2,3, Shrikanta Chattopadhyay1,6, Thomas Hasaka1, Rajiv Narayan1, Mingji Dai1,7, Christina Huang1, Sebastian Shterental2, Lisa P Chu2, J Erika Haydu2, Jae Hung Shieh5, David P Steensma3,8, Benito Munoz1, Joshua A Bittker1, Alykhan F Shamji1, Paul A Clemons1, Nicola J Tolliday1, Anne E Carpenter1, D Gary Gilliland1,2,8,9, Andrew M Stern1, Malcolm A S Moore10, David T Scadden1,4,6, Stuart L Schreiber1,9,7, Benjamin L Ebert1,2,3,8, Todd R Golub1,3,9,11

Author Affiliations

1: Broad Institute of MIT and Harvard, Cambridge, MA 02142, USA.
2: Division of Hematology, Department of Medicine, Brigham and Women's Hospital and Harvard Medical School, Boston, MA 02115, USA.
3: Harvard Medical School, Boston, MA 02115, USA.
4: Center for Regenerative Medicine and Cancer Center, Massachusetts General Hospital, Boston, MA 02114, USA.
5: Department of Pediatrics, Memorial Sloan-Kettering Cancer Center, New York, NY 10021, USA.
6: Department of Stem Cell and Regenerative Biology, Harvard University, Cambridge, MA 02138, USA.
7: Department of Chemistry and Chemical Biology, Harvard University, Cambridge, MA 02138, USA.
8: Department of Medical Oncology, Dana-Farber Cancer Institute, Harvard Medical School, Boston, MA 02115, USA.
9: Howard Hughes Medical Institute, Harvard Medical School, Chevy Chase, MD 20815, USA.
10: Cell Biology Program, Memorial Sloan-Kettering Cancer Center, New York, NY 10021, USA.
11: Department of Pediatric Oncology, Dana-Farber Cancer Institute, Boston, MA 02115, USA.

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