Published in Pflugers Arch on December 01, 1985
Voltage-dependent magnesium block of adenosine-triphosphate-sensitive potassium channel in guinea-pig ventricular cells. J Physiol (1987) 3.29
A metabolite-regulated potassium channel in rat pancreatic B cells. Proc Natl Acad Sci U S A (1986) 2.27
The effects of magnesium upon adenosine triphosphate-sensitive potassium channels in a rat insulin-secreting cell line. J Physiol (1987) 1.86
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Properties and calcium-dependent inactivation of calcium currents in cultured mouse pancreatic B-cells. J Physiol (1988) 1.69
Properties of single potassium channels modulated by glucose in rat pancreatic beta-cells. J Physiol (1988) 1.63
Dual effects of diazoxide on ATP-K+ currents recorded from an insulin-secreting cell line. Br J Pharmacol (1989) 1.59
Inhibition by glibenclamide of the vasorelaxant action of cromakalim in the rat. Br J Pharmacol (1989) 1.52
Modulation of the bursting properties of single mouse pancreatic beta-cells by artificial conductances. Biophys J (1999) 1.46
Phentolamine and yohimbine inhibit ATP-sensitive K+ channels in mouse pancreatic beta-cells. Br J Pharmacol (1990) 1.45
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Endocytosis of secretory granules in mouse pancreatic beta-cells evoked by transient elevation of cytosolic calcium. J Physiol (1996) 1.28
ATP-sensitive K+ channels that are blocked by hypoglycemia-inducing sulfonylureas in insulin-secreting cells are activated by galanin, a hyperglycemia-inducing hormone. Proc Natl Acad Sci U S A (1988) 1.26
Activators of protein kinase C depolarize insulin-secreting cells by closing K+ channels. EMBO J (1988) 1.25
Role of single-channel stochastic noise on bursting clusters of pancreatic beta-cells. Biophys J (1988) 1.20
Failure of glucose to elicit a normal secretory response in fetal pancreatic beta cells results from glucose insensitivity of the ATP-regulated K+ channels. Proc Natl Acad Sci U S A (1989) 1.19
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Block of ATP-regulated and Ca2(+)-activated K+ channels in mouse pancreatic beta-cells by external tetraethylammonium and quinine. J Physiol (1990) 1.17
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Voltage-activated currents in guinea pig pancreatic alpha 2 cells. Evidence for Ca2+-dependent action potentials. J Gen Physiol (1988) 1.14
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Multiple actions of pinacidil on adenosine triphosphate-sensitive potassium channels in guinea-pig ventricular myocytes. J Physiol (1990) 1.11
Cloning and expression of two brain-specific inwardly rectifying potassium channels. Proc Natl Acad Sci U S A (1995) 1.09
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The effects of cromakalim on ATP-sensitive potassium channels in insulin-secreting cells. Br J Pharmacol (1990) 1.02
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Mg(2+)-dependent inhibition of KATP by sulphonylureas in CRI-G1 insulin-secreting cells. Br J Pharmacol (1994) 0.98
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A model of action potentials and fast Ca2+ dynamics in pancreatic beta-cells. Biophys J (2009) 0.92
Effects of intracellular pH on ATP-sensitive K+ channels in mouse pancreatic beta-cells. J Physiol (1994) 0.92
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Clonidine inhibits ATP-sensitive K+ channels in mouse pancreatic beta-cells. Br J Pharmacol (1991) 0.92
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Activation of transmembrane bile acid receptor TGR5 stimulates insulin secretion in pancreatic β cells. Biochem Biophys Res Commun (2012) 0.90
Glucose increases activity and Ca2+ in insulin-producing cells of adult Drosophila. Neuroreport (2010) 0.89
Block of pancreatic ATP-sensitive K+ channels and insulinotrophic action by the antiarrhythmic agent, cibenzoline. Br J Pharmacol (1996) 0.89
Cross-talk between ATP-regulated K+ channels and Na+ transport via cellular metabolism in frog skin principal cells. J Physiol (1996) 0.87
Significance of Na/Ca exchange for Ca2+ buffering and electrical activity in mouse pancreatic beta-cells. Biophys J (1999) 0.85
Block of ATP-sensitive K+ channels in isolated mouse pancreatic beta-cells by 2,3-butanedione monoxime. Br J Pharmacol (1994) 0.85
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Effects of lactate on pancreatic islets. Lactate efflux as a possible determinant of islet-cell depolarization by glucose. Biochem J (1989) 0.84
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Inhibition of the ATP-sensitive potassium channel by class I antiarrhythmic agent, cibenzoline, in rat pancreatic beta-cells. Br J Pharmacol (1993) 0.82
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Amantadine and sparteine inhibit ATP-regulated K-currents in the insulin-secreting beta-cell line, HIT-T15. Br J Pharmacol (1991) 0.81
Barbiturates inhibit ATP-K+ channels and voltage-activated currents in CRI-G1 insulin-secreting cells. Br J Pharmacol (1991) 0.81
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Potentiation of sulfonylurea action by an EPAC-selective cAMP analog in INS-1 cells: comparison of tolbutamide and gliclazide and a potential role for EPAC activation of a 2-APB-sensitive Ca2+ influx. Mol Pharmacol (2012) 0.78
Cloning of a pore-forming subunit of ATP-sensitive potassium channel from Clonorchis sinensis. Korean J Parasitol (2003) 0.77
Synthesis and characterization of a quinolinonic compound activating ATP-sensitive K(+) channels in endocrine and smooth muscle tissues. Br J Pharmacol (2001) 0.77
Uncoupling of Cav1.2 from Ca(2+)-induced Ca(2+) release and SK channel regulation in pancreatic β-cells. Mol Endocrinol (2014) 0.77
Glibenclamide increases post-fatigue tension in slow skeletal muscle fibers of the chicken. J Comp Physiol B (2010) 0.76
Loperamide mobilizes intracellular Ca2+ stores in insulin-secreting HIT-T15 cells. Br J Pharmacol (2003) 0.75
Activation of insulin-secreting cells by pyruvate and halogenated derivatives. Biochem J (1990) 0.75
Effects of nicorandil on the recovery of reflex potentials after spinal cord ischaemia in cats. Br J Pharmacol (1995) 0.75
Electrophysiology of the pancreatic beta-cell. Prog Biophys Mol Biol (1989) 6.00
Conductance properties of single inwardly rectifying potassium channels in ventricular cells from guinea-pig heart. J Physiol (1984) 4.70
Voltage-dependent inactivation of inward-rectifying single-channel currents in the guinea-pig heart cell membrane. J Physiol (1984) 4.08
Opposite effects of tolbutamide and diazoxide on the ATP-dependent K+ channel in mouse pancreatic beta-cells. Pflugers Arch (1986) 3.51
Calcium and delayed potassium currents in mouse pancreatic beta-cells under voltage-clamp conditions. J Physiol (1986) 3.46
Ro 25-6981, a highly potent and selective blocker of N-methyl-D-aspartate receptors containing the NR2B subunit. Characterization in vitro. J Pharmacol Exp Ther (1997) 2.68
Inward-rectifying channels in isolated patches of the heart cell membrane: ATP-dependence and comparison with cell-attached patches. Pflugers Arch (1984) 2.59
The effect of subunit composition of rat brain GABAA receptors on channel function. Neuron (1990) 2.54
Exocytosis elicited by action potentials and voltage-clamp calcium currents in individual mouse pancreatic B-cells. J Physiol (1993) 2.47
Calcium-independent potentiation of insulin release by cyclic AMP in single beta-cells. Nature (1993) 2.40
Co-localization of L-type Ca2+ channels and insulin-containing secretory granules and its significance for the initiation of exocytosis in mouse pancreatic B-cells. EMBO J (1995) 2.39
Inositol trisphosphate-dependent periodic activation of a Ca(2+)-activated K+ conductance in glucose-stimulated pancreatic beta-cells. Nature (1991) 2.35
Dual effects of ATP on K+ currents of mouse pancreatic beta-cells. Pflugers Arch (1987) 2.19
Modulation of dihydropyridine-sensitive Ca2+ channels by glucose metabolism in mouse pancreatic beta-cells. Nature (1989) 2.07
Protein kinase A-dependent and -independent stimulation of exocytosis by cAMP in mouse pancreatic B-cells. J Physiol (1997) 2.06
Regulation of glucagon release in mouse -cells by KATP channels and inactivation of TTX-sensitive Na+ channels. J Physiol (2000) 2.05
Voltage-gated and resting membrane currents recorded from B-cells in intact mouse pancreatic islets. J Physiol (1999) 2.01
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Tight coupling between electrical activity and exocytosis in mouse glucagon-secreting alpha-cells. Diabetes (2000) 1.88
Fast exocytosis with few Ca(2+) channels in insulin-secreting mouse pancreatic B cells. Biophys J (2001) 1.79
The voltage sensitive Lc-type Ca2+ channel is functionally coupled to the exocytotic machinery. Proc Natl Acad Sci U S A (1999) 1.78
Rapid ATP-dependent priming of secretory granules precedes Ca(2+)-induced exocytosis in mouse pancreatic B-cells. J Physiol (1997) 1.72
Simultaneous recordings of glucose dependent electrical activity and ATP-regulated K(+)-currents in isolated mouse pancreatic beta-cells. FEBS Lett (1990) 1.68
Concentration-dependent effects of tolbutamide, meglitinide, glipizide, glibenclamide and diazoxide on ATP-regulated K+ currents in pancreatic B-cells. Naunyn Schmiedebergs Arch Pharmacol (1988) 1.66
Multivesicular exocytosis in rat pancreatic beta cells. Diabetologia (2011) 1.63
Adrenaline stimulates glucagon secretion in pancreatic A-cells by increasing the Ca2+ current and the number of granules close to the L-type Ca2+ channels. J Gen Physiol (1997) 1.62
Activation of Ca(2+)-dependent K(+) channels contributes to rhythmic firing of action potentials in mouse pancreatic beta cells. J Gen Physiol (1999) 1.59
Activation of protein kinases and inhibition of protein phosphatases play a central role in the regulation of exocytosis in mouse pancreatic beta cells. Proc Natl Acad Sci U S A (1994) 1.59
A novel mechanism of activity-dependent NMDA receptor antagonism describes the effect of ifenprodil in rat cultured cortical neurones. J Physiol (1996) 1.56
Patch-clamp characterisation of somatostatin-secreting -cells in intact mouse pancreatic islets. J Physiol (2000) 1.49
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Cellular regulation of islet hormone secretion by the incretin hormone glucagon-like peptide 1. Pflugers Arch (1998) 1.46
Somatostatin release, electrical activity, membrane currents and exocytosis in human pancreatic delta cells. Diabetologia (2009) 1.46
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Dual effects of glucose on the cytosolic Ca2+ activity of mouse pancreatic beta-cells. FEBS Lett (1984) 1.42
Cooling inhibits exocytosis in single mouse pancreatic B-cells by suppression of granule mobilization. J Physiol (1996) 1.41
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Priming of insulin granules for exocytosis by granular Cl(-) uptake and acidification. J Cell Sci (2001) 1.37
Changes of membrane currents in cardiac cells induced by long whole-cell recordings and tolbutamide. Pflugers Arch (1987) 1.35
Glucagon-like peptide 1 (7-36) amide stimulates exocytosis in human pancreatic beta-cells by both proximal and distal regulatory steps in stimulus-secretion coupling. Diabetes (1998) 1.33
Separate processes mediate nucleotide-induced inhibition and stimulation of the ATP-regulated K(+)-channels in mouse pancreatic beta-cells. Proc Biol Sci (1991) 1.32
Characterisation of sulphonylurea and ATP-regulated K+ channels in rat pancreatic A-cells. Pflugers Arch (1999) 1.32
Single Ca channel currents in mouse pancreatic B-cells. Pflugers Arch (1988) 1.30
Endocytosis of secretory granules in mouse pancreatic beta-cells evoked by transient elevation of cytosolic calcium. J Physiol (1996) 1.28
Effects of external tetraethylammonium ions and quinine on delayed rectifying K+ channels in mouse pancreatic beta-cells. J Physiol (1990) 1.26
Cytosolic ADP enhances the sensitivity to tolbutamide of ATP-dependent K+ channels from pancreatic B-cells. FEBS Lett (1988) 1.24
Glucagon-like peptide I increases cytoplasmic calcium in insulin-secreting beta TC3-cells by enhancement of intracellular calcium mobilization. Diabetes (1995) 1.22
PKC-dependent stimulation of exocytosis by sulfonylureas in pancreatic beta cells. Science (1996) 1.22
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Increased activity of L-type Ca2+ channels exposed to serum from patients with type I diabetes. Science (1993) 1.19
Block of ATP-regulated and Ca2(+)-activated K+ channels in mouse pancreatic beta-cells by external tetraethylammonium and quinine. J Physiol (1990) 1.17
Delayed rectifying and calcium-activated K+ channels and their significance for action potential repolarization in mouse pancreatic beta-cells. J Gen Physiol (1990) 1.16
Multisite regulation of insulin secretion by cAMP-increasing agonists: evidence that glucagon-like peptide 1 and glucagon act via distinct receptors. Pflugers Arch (1997) 1.14
Stimulation of the KATP channel by ADP and diazoxide requires nucleotide hydrolysis in mouse pancreatic beta-cells. J Physiol (1993) 1.13
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